| Compound ID |
Compound Name |
Compound Formula |
|
CP0476826
|
N,N-bis(pyridin-2-ylmethyl)-1-[5-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)naphthalen-2-yl]methanamine
Show/Hide
|
C34H45N7
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0521193
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-4-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0435221
|
N,N-bis(pyridin-2-ylmethyl)-1-[2-[3-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)phenyl]pyridin-4-yl]methanamine
Show/Hide
|
C35H46N8
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0378861
|
(2R)-2-[[(3R,6S,9R,12S,15R,20S,23R,26S,29R,32S)-3,6-bis(4-aminobutyl)-15-[[(2R)-2-[[(2R)-2-[[(2R)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-carbamimidamidopentanoyl]amino]propanoyl]amino]-9,26-bis(3-carbamimidamidopropyl)-23-[3-(carbamoylamino)propyl]-12-[(4-hydroxyphenyl)methyl]-29-[(4-methoxyphenyl)methyl]-2,5,8,11,14,22,25,28,31-nonaoxo-17,18-dithia-1,4,7,10,13,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-20-carbonyl]amino]-5-carbamimidamidopentanoic acid
Show/Hide
|
C81H137N33O18S2
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0442837
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N11O6
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0177564
|
2-[3-[(2R,5S,8S,14R)-5-[3-(diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N11O6
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0493224
|
2-[3-[(4R,7S,10S,13S)-10-[3-(diaminomethylideneamino)propyl]-4-[(4-hydroxyphenyl)methyl]-13-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,3,6,9,12-pentazacyclotetradec-7-yl]propyl]guanidine
Show/Hide
|
C35H45N11O6
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0427154
|
N,N-bis(pyridin-2-ylmethyl)-1-[4-[3-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)pyridin-2-yl]phenyl]methanamine
Show/Hide
|
C35H46N8
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0440699
|
N,N-bis(pyridin-2-ylmethyl)-1-[4-[2-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)phenyl]phenyl]methanamine
Show/Hide
|
C36H47N7
|
1
|
| 1 |
IC50 = 5.7 nM
|
|
|
|
CP0427153
|
N,N-bis(pyridin-2-ylmethyl)-1-[2-[3-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)phenyl]phenyl]methanamine
Show/Hide
|
C36H47N7
|
1
|
| 1 |
IC50 = 7.9 nM
|
|
|
|
CP0442841
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N11O6
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0248152
|
2-[3-[(2S,5S,8S,14R)-5-[3-(diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N11O6
|
2
|
| 1 |
IC50 = 8.4 nM
|
|
|
| 2 |
IC50 = 35 nM
|
|
|
|
CP0497380
|
2-[3-[(3R,9S,12S,15S,17S)-17-(diaminomethylideneamino)-3-[(4-hydroxyphenyl)methyl]-9-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-12-yl]propyl]guanidine
Show/Hide
|
C36H45N11O6
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0498468
|
2-[3-[(3R,9S,12S,15S,17R)-17-(diaminomethylideneamino)-3-[(4-hydroxyphenyl)methyl]-9-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-12-yl]propyl]guanidine
Show/Hide
|
C36H45N11O6
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0427157
|
N,N-bis(pyridin-2-ylmethyl)-1-[6-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)naphthalen-2-yl]methanamine
Show/Hide
|
C34H45N7
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0526667
|
2-[3-[(2S,5R,8R,11R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-11-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0526669
|
2-[3-[(2S,5S,8R,11R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-11-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0847581
|
N-{3-[(2S,5S,11R)-14-(2-Amino-ethyl)-11-(4-hydroxy-benzyl)-5-naphthalen-2-ylmethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-propyl}-guanidine
Show/Hide
|
C34H43N9O6
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0426218
|
(3R)-4-[[(2R)-6-amino-1-[[(2R)-6-amino-1-[[(2R)-1-[[6-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S,3R)-1-[[(2S)-4-amino-1-[[(2S)-4-amino-1-[[(2S)-4-amino-1-[(2S)-2-[[(2S)-5-carbamimidamido-1-[[(2S,3R)-1-[[(1R)-1-carboxy-2-sulfanylethyl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1,4-dioxobutan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-1,4-dioxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxohexan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C122H206N46O33S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0402847
|
(3S)-3-[[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-[6-[[(2R)-2-[[(2R)-6-amino-2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]hexanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoylamino]hexanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]acetyl]amino]-4-[[(2S,3S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
|
C123H207N47O30S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0406622
|
2-[3-[(2S,5S,11R,14S)-14-(3-aminopropyl)-11-[(4-hydroxyphenyl)methyl]-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C35H45N9O6
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0526665
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-1-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0482780
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C128H203N39O35
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0442699
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-4-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0451299
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C136H219N39O39
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0406623
|
2-[3-[(2S,5S,11R,14S)-14-[2-(diaminomethylideneamino)ethyl]-11-[(4-hydroxyphenyl)methyl]-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C35H45N11O6
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0482774
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[2-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[2-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C144H235N39O43
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0372636
|
2-[3-[(2S,5S,8S,14R)-5-[3-(diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-8-(naphthalen-2-ylmethyl)-3,6,12,15-tetraoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H49N11O5
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0435223
|
N,N-bis(pyridin-2-ylmethyl)-1-[4-(1,4,8,11-tetrazacyclotetradec-1-ylmethyl)phenyl]methanamine
Show/Hide
|
C30H43N7
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0069850
|
(6,6-dimethyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-3-yl)methyl N,N'-dicyclohexylimidothiocarbamate
Show/Hide
|
C21H34N4S2
|
1
|
| 1 |
IC50 = 32.5 nM
|
|
|
|
CP0421153
|
2-[3-[(2S,5S,11R,14S)-14-[4-(diaminomethylideneamino)butyl]-11-[(4-hydroxyphenyl)methyl]-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0451266
|
(2R)-N-[(2R)-1-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-1-oxopropan-2-yl]-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carboxamide
Show/Hide
|
C126H203N39O31
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0390594
|
2-[3-[(2S,5S,11R,14S)-11-[(4-hydroxyphenyl)methyl]-13,14-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C34H42N8O6
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0454343
|
2-[3-[(2S,5S,8S,11R)-8-[3-(diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-2-(naphthalen-2-ylmethyl)-3,6,9,12,16-pentaoxo-1,4,7,10,13-pentazacyclohexadec-5-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0145769
|
1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-tetraaza-cyclotetradecane}
Show/Hide
|
C28H54N8
|
2
|
| 1 |
IC50 = 51 nM
|
|
|
| 2 |
IC50 = 65 nM
|
|
|
|
CP0515391
|
2-[3-[(2S,5S,8R,11S)-8-[3-(diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,14-tetraoxo-1,4,7,10-tetrazacyclotetradec-5-yl]propyl]guanidine
Show/Hide
|
C36H48N10O5
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0526664
|
2-[3-[(2S,5S,8R,14S)-8-[(4-hydroxyphenyl)methyl]-5-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0515402
|
2-[3-[(2S,5S,11R,14R)-11-[(4-hydroxyphenyl)methyl]-14-methyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0430359
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]amino]propanoyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]amino]propanoyl]amino]-4-oxobutanoic acid
Show/Hide
|
C124H199N39O35
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0526668
|
2-[3-[(2S,5R,8R,11S,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-11-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0487232
|
2-[3-[(2S,5S,11R,14R)-14-(4-aminobutyl)-11-[(4-hydroxyphenyl)methyl]-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N9O6
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0383343
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-1-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0564711
|
(2R)-N-[2-[2-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[2-[2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carboxamide
Show/Hide
|
C116H185N33O31
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0516517
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-7-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 128 nM
|
|
|
|
CP0383345
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C30H43N11O5
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0530533
|
(2R)-N-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethyl]-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carboxamide
Show/Hide
|
C108H169N33O27
|
1
|
| 1 |
IC50 = 144 nM
|
|
|
|
CP0559510
|
(3R)-4-[[(2R)-6-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[2-[[(2R)-1-[[(2R)-5-amino-1-[[(2R)-6-amino-1-[[(2R)-1-[(2R)-2-[[(2R)-1-[(2R)-2-[[6-[[(2S)-6-amino-1-[[2-[[(2S)-1-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C151H249N45O36S2
|
1
|
| 1 |
IC50 = 147 nM
|
|
|
|
CP0503179
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-7-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 157 nM
|
|
|
|
CP0560168
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-10,14-dimethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C27H43N11O6
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0457621
|
2-[3-[(2S,5S,8R,11S,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-11-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0497749
|
3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hydroxy-benzyl)-8-naphthalen-2-ylmethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-propionamide
Show/Hide
|
C35H43N9O7
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0421256
|
2-[3-[(2R,5S,8S,11S,12E)-8-[3-(diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,15-tetraoxo-1,4,7,10-tetrazacyclopentadec-12-en-5-yl]propyl]guanidine
Show/Hide
|
C37H48N10O5
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0391066
|
2-[3-[(2S,5S,8R,14R)-5-[3-(diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C36H47N11O6
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0562552
|
(3R)-4-[[(2R)-6-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[2-[[(2R)-1-[[(2R)-5-amino-1-[[(2R)-6-amino-1-[[(2R)-1-[(2R)-2-[[(2R)-1-[(2R)-2-[[6-[[(2S)-6-amino-1-[[(2R)-6-amino-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[(2R)-1-[[2-[[(2R)-1-[[(2R)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-6-oxohexyl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-carbamimidamido-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C168H265N49O38S2
|
1
|
| 1 |
IC50 = 193 nM
|
|
|
|
CP0457622
|
2-[3-[(2S,5R,8R,14S)-8-[(4-hydroxyphenyl)methyl]-5-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0497746
|
2-[3-[(2S,5S,11R,14S)-11-[(4-hydroxyphenyl)methyl]-14-methyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0377354
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-13-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0521192
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-10-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0515403
|
2-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hydroxy-benzyl)-8-naphthalen-2-ylmethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-acetamide
Show/Hide
|
C34H41N9O7
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0454342
|
2-[3-[(2S,5S,8R,11R)-8-[3-(diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-2-(naphthalen-2-ylmethyl)-3,6,9,12,16-pentaoxo-1,4,7,10,13-pentazacyclohexadec-5-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0446671
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(2S)-1-amino-6-[3-[2-[2-[2-[[(2S)-5-carbamimidamido-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]pentanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-1-oxohexan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C119H196N34O33
|
1
|
| 1 |
IC50 = 407 nM
|
|
|
|
CP0497752
|
2-[3-[(3R,9S,12S,15R)-3-[(4-hydroxyphenyl)methyl]-9-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-12-yl]propyl]guanidine
Show/Hide
|
C35H42N8O6
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0578919
|
(3R)-4-[[(2R)-6-amino-1-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C104H157N35O26
|
1
|
| 1 |
IC50 = 462 nM
|
|
|
|
CP0426217
|
(3R)-4-[[(2R)-6-amino-1-[[(2R)-6-amino-1-[[(2R)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C64H104N24O15
|
1
|
| 1 |
IC50 = 474 nM
|
|
|
|
CP0497378
|
2-[3-[(2S,5S,11R,14R)-11-[(4-hydroxyphenyl)methyl]-13,14-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C34H42N8O6
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0562253
|
(3R)-4-[[(2R)-6-amino-1-[[(2R)-1-amino-6-[[(2S)-5-carbamimidamido-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]pentanoyl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C101H162N32O25
|
1
|
| 1 |
IC50 = 502 nM
|
|
|
|
CP0499960
|
(4S,7S,10S,13R)-13-(3-Guanidino-propionylamino)-10-(3-guanidino-propyl)-7-naphthalen-2-ylmethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid [2-(4-hydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C37H49N11O6S2
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0419682
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-13-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C37H49N11O6
|
1
|
| 1 |
IC50 = 563 nM
|
|
|
|
CP0498467
|
3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hydroxy-benzyl)-8-naphthalen-2-ylmethyl-3,6,9,12,15-pentaoxo-1,4,7,10,13pentaaza-cyclopentadec-2-yl]-propionic acid
Show/Hide
|
C35H42N8O8
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0526666
|
2-[3-[(3R,6R,9S,12S,15S)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.4.0]nonadecan-9-yl]propyl]guanidine
Show/Hide
|
C40H53N11O6
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0391560
|
(R)-13-(3-Guanidino-propionylamino)-10-(3-guanidino-propyl)-7-((S)-(R)-1-naphthalen-2-ylmethyl)-6,9-dioxo-12-(R)-oxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid amide
Show/Hide
|
C29H41N11O5S2
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0540665
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(2S)-1-amino-6-[3-[2-[2-[2-[2-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-1-oxohexan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C108H183N29O32
|
1
|
| 1 |
IC50 = 737 nM
|
|
|
|
CP0552664
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[2-[2-[3-[[(2S)-1-amino-6-[3-[2-[2-[2-[2-[2-[[(2S)-5-carbamimidamido-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]pentanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-1-oxohexan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C127H212N34O37
|
1
|
| 1 |
IC50 = 747 nM
|
|
|
|
CP0509773
|
(4S,7S,10S,13R)-10-(3-Guanidino-propyl)-13-(3-guanidino-propylamino)-7-naphthalen-2-ylmethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid amide
Show/Hide
|
C29H43N11O4S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0526018
|
(4S,7S,10S,13R)-10-(3-Guanidino-propyl)-13-(3-guanidino-propylamino)-7-naphthalen-2-ylmethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid [2-(4-hydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C37H51N11O5S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0383950
|
(3R)-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-4-[[(2R)-1,6-diamino-1-oxohexan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
|
C52H80N18O13
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0523058
|
5-((S)-2-Guanidino-4-methyl-pentanoylamino)-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C30H40N10O2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0528547
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(2S)-1-amino-6-[3-[2-[2-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-1-oxohexan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C101H170N28O28
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0497751
|
2-[3-[(3R,9S,12S,15S)-3-[(4-hydroxyphenyl)methyl]-9-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-12-yl]propyl]guanidine
Show/Hide
|
C35H42N8O6
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0554615
|
5-((S)-2-Guanidino-3-phenyl-propionylamino)-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C33H38N10O2
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0572946
|
(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoic acid
Show/Hide
|
C52H79N17O14
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0554616
|
5-((R)-2-Guanidino-4-methyl-pentanoylamino)-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C30H40N10O2
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0540667
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C67H109N21O18
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0438878
|
N-[2-[2-(diaminomethylideneamino)ethyl]-1-(2-naphthalen-2-ylethyl)indol-5-yl]-3-(4-hydroxyphenyl)propanamide
Show/Hide
|
C32H33N5O2
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0387541
|
5-(2-Guanidino-acetylamino)-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C26H32N10O2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0489417
|
5-[(1-Carbamimidoyl-piperidine-4-carbonyl)-amino]-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C30H38N10O2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0430827
|
5-((R)-2-Guanidino-3-phenyl-propionylamino)-1-(3-guanidino-propyl)-1H-indole-2-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C33H38N10O2
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0468563
|
1-(3-Guanidino-propyl)-5-[2-(4-hydroxy-phenyl)-acetylamino]-1H-indole-2-carboxylic acid naphthalen-1-ylamide
Show/Hide
|
C31H30N6O3
|
1
|
| 1 |
IC50 = 4800 nM
|
|
|
|
CP0649585
|
1-butyl-3-(2-methylpropyl)-9-(6-phenylhexyl)-1,4,9-triazaspiro-[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C28H46ClN3O2
|
1
|
| 1 |
IC50 = 6700 nM
|
|
|
|
CP0511994
|
(6,6-dimethyl-5H-imidazo[2,1-b][1,3]thiazol-3-yl)methyl N'-[4-[[[2-[2-[4-[[2-[2-[[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethoxy]acetyl]amino]butylamino]-2-oxoethoxy]acetyl]amino]methyl]cyclohexyl]carbamimidothioate
Show/Hide
|
C48H69N9O9S2
|
1
|
| 1 |
IC50 = 8300 nM
|
|
|
|
CP0402848
|
(2R)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-1-[(2S)-4-amino-2-[[(2S)-4-amino-2-[[(2S)-4-amino-2-[[(2S,3R)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-(6-aminohexanoylamino)hexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]-3-hydroxybutanoyl]amino]-4-oxobutanoyl]amino]-4-oxobutanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-hydroxybutanoyl]amino]-3-sulfanylpropanoic acid
Show/Hide
|
C58H105N23O18S
|
1
|
| 1 |
IC50 = 9120 nM
|
|
|
|
CP0651200
|
9-(1,4-benzodioxane-6-yl)-1-butyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C25H38ClN3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0657856
|
(+/-)-1-butyl-3-(cyclohexylmethyl)-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride
Show/Hide
|
C32H44ClN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0662025
|
(3R)-3-cyclohexylmethyl-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C30H48ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0662064
|
9-(1,4-benzodioxane-6-yl)-1-butyl-3-cyclohexyl-1,4,9-triazaspiro-[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C28H42ClN3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0662079
|
(3S)-3-cyclohexylmethyl-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C30H48ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0720738
|
(+/-)-1-butyl-3-isobutyl-9-(4-phenoxybenzyl)-1,4,9-triazaspiro[5.5]undecane-2,5-dione hydrochloride
Show/Hide
|
C29H40ClN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0837909
|
9-(4-allyloxyphenylmethyl)-1-butyl-3-cyclohexyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C29H44ClN3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0878091
|
(3R)-3-(2-methylpropyl)-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C27H44ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0878092
|
(3S)-3-(2-methylpropyl)-9-(6-phenylhexyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C27H44ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0497750
|
(4S,7S,10S,13R)-13-(3-Guanidino-propionylamino)-10-(3-guanidino-propyl)-11-methyl-7-naphthalen-2-ylmethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid amide
Show/Hide
|
C30H43N11O5S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0499961
|
(4S,7S,10S,13R)-13-(3-Guanidino-propionylamino)-10-(3-guanidino-propyl)-11-methyl-7-naphthalen-2-ylmethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid [2-(4-hydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C38H51N11O6S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0449094
|
(Z)-(2S,5S,8R,14S)-14-(3-Guanidino-propionylamino)-2-(3-guanidino-propyl)-5-naphthalen-2-ylmethyl-3,6,15-trioxo-1,4,7triaza-cyclopentadec-11-ene-8-carboxylic acid amide
Show/Hide
|
C32H45N11O5
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0486077
|
(Z)-(2S,5S,8R,15S)-15-(3-Guanidino-propionylamino)-2-(3-guanidino-propyl)-5-naphthalen-2-ylmethyl-3,6,16-trioxo-1,4,7triaza-cyclohexadec-11-ene-8-carboxylic acid amide
Show/Hide
|
C33H47N11O5
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0861243
|
(Z)-(2S,5S,8R,13S)-13-(3-Guanidino-propionylamino)-2-(3-guanidino-propyl)-5-naphthalen-2-ylmethyl-3,6,14-trioxo-1,4,7triaza-cyclotetradec-10-ene-8-carboxylic acid amide
Show/Hide
|
C31H43N11O5
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0911862
|
(Z)-(2S,5S,8R,13S)-13-(3-Guanidino-propionylamino)-2-(3-guanidino-propyl)-5-naphthalen-2-ylmethyl-3,6,14-trioxo-1,4,7triaza-cyclotetradec-10-ene-8-carboxylic acid [2-(4-hydroxy-phenyl)-ethyl]-amide
Show/Hide
|
C39H51N11O6
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0502395
|
2-[3-[(3S,6R,12R,13Z,15S)-15-[3-(diaminomethylideneamino)propyl]-6-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclopentadec-13-en-3-yl]propyl]guanidine
Show/Hide
|
C37H48N10O5
|
1
|
| 1 |
IC50 = 21000 nM
|
|
|
|
CP0651202
|
1-butyl-3-cyclohexylmethyl-9-(4-methoxyphenylmethyl)-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C27H42ClN3O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0651215
|
9-benzyl-1-butyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]-undeca-2,5-dione hydrochloride
Show/Hide
|
C23H36ClN3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0699196
|
3-(2-methylpropyl)-9-(4-phenoxyphenylmethyl)-1-propyl-1,4,9-triazaspiro[5.5]undeca-2,5-dione hydrochloride
Show/Hide
|
C28H38ClN3O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0850182
|
(3R)-1,9-dibenzyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]-undeca-2,5-dione hydrochloride
Show/Hide
|
C26H34ClN3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0856132
|
(3S)-1,9-dibenzyl-3-(2-methylpropyl)-1,4,9-triazaspiro[5.5]-undeca-2,5-dione hydrochloride
Show/Hide
|
C26H34ClN3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0515389
|
2-[3-[(4R,7S,10S,11Z,13S)-7-[3-(diaminomethylideneamino)propyl]-4-[(4-hydroxyphenyl)methyl]-13-(naphthalen-2-ylmethyl)-2,5,8,14-tetraoxo-1,3,6,9-tetrazacyclotetradec-11-en-10-yl]propyl]guanidine
Show/Hide
|
C36H46N10O5
|
1
|
| 1 |
IC50 = 31000 nM
|
|
|
|
CP0384173
|
(3S)-3-[[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-(6-aminohexanoylamino)hexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]amino]acetyl]amino]-4-[[(2S,3S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
|
C59H106N24O15S
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0564856
|
(6,6-dimethyl-5H-imidazo[2,1-b][1,3]thiazol-3-yl)methyl N-cyclohexyl-N'-[4-[[[2-[2-[4-[[2-[2-(methylamino)-2-oxoethoxy]acetyl]amino]butylamino]-2-oxoethoxy]acetyl]amino]methyl]cyclohexyl]carbamimidothioate
Show/Hide
|
C35H58N8O6S2
|
1
|
| 1 |
IC50 = 53000 nM
|
|
|
|
CP0444195
|
(6,6-dimethyl-5H-imidazo[2,1-b][1,3]thiazol-3-yl)methyl N-cyclohexyl-N'-[4-[[[2-[2-[6-[[2-[2-(methylamino)-2-oxoethoxy]acetyl]amino]hexylamino]-2-oxoethoxy]acetyl]amino]methyl]cyclohexyl]carbamimidothioate
Show/Hide
|
C37H62N8O6S2
|
1
|
| 1 |
IC50 = 74000 nM
|
|
|
|
CP0421366
|
2-[3-[(4R,7S,10S,13S)-10-[3-(diaminomethylideneamino)propyl]-4-[(4-hydroxyphenyl)methyl]-13-(naphthalen-2-ylmethyl)-2,5,8,14-tetraoxo-1,3,6,9,12-pentazacyclotetradec-7-yl]propyl]guanidine
Show/Hide
|
C35H47N11O5
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0424785
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-methyl-14-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C30H43N11O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0424786
|
2-[3-[(2S,5S,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-14-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C26H41N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0441862
|
2-[3-[(3R,6S,9S,12S,15S)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidine
Show/Hide
|
C39H51N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0441865
|
2-[3-[(2R,5R,11S,14S)-5-[(4-hydroxyphenyl)methyl]-14-methyl-11-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0442838
|
2-[3-[(3R,6R,9S,12S,15R)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidine
Show/Hide
|
C39H51N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0442844
|
2-[3-[(2S,5R,11S,14S)-5-[(4-hydroxyphenyl)methyl]-14-methyl-11-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C33H40N8O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0454115
|
2-[3-[(3R,6R,9S,12S,15R)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.4.0]nonadecan-9-yl]propyl]guanidine
Show/Hide
|
C40H53N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0502747
|
2-[3-[(3R,6S,9S,12S,15R)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidine
Show/Hide
|
C39H51N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0514352
|
2-[3-[(3R,6S,9S,12S,15R)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.4.0]nonadecan-9-yl]propyl]guanidine
Show/Hide
|
C40H53N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0514353
|
2-[3-[(3R,6S,9S,12S,15S)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.4.0]nonadecan-9-yl]propyl]guanidine
Show/Hide
|
C40H53N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0526662
|
2-[3-[(3R,6R,9S,12S,15S)-6-[3-(diaminomethylideneamino)propyl]-3-[(4-hydroxyphenyl)methyl]-12-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidine
Show/Hide
|
C39H51N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0526663
|
2-[3-[(2S,5R,8R,14S)-5-[3-(diaminomethylideneamino)propyl]-8-[(4-hydroxyphenyl)methyl]-14-methyl-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidine
Show/Hide
|
C26H41N11O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0391559
|
2-[3-[(2S,5R,8R,11S)-8-[3-(diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,14-tetraoxo-1,4,7,10-tetrazacyclotetradec-5-yl]propyl]guanidine
Show/Hide
|
C36H48N10O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0485216
|
2-[3-[(2S,5S,8R,11R,12Z)-8-[3-(diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,14-tetraoxo-1,4,7,10-tetrazacyclotetradec-12-en-5-yl]propyl]guanidine
Show/Hide
|
C36H46N10O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0487201
|
2-[3-[(2S,5R,8R,11R,12Z)-8-[3-(diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,14-tetraoxo-1,4,7,10-tetrazacyclotetradec-12-en-5-yl]propyl]guanidine
Show/Hide
|
C36H46N10O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0430351
|
(2S)-2,6-bis[3-[2-[2-[2-[2-[2-[2-[2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C62H119N11O23
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0430352
|
(2S)-2,6-bis[3-[2-[2-[2-[2-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C102H163N23O31
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0530532
|
(3R)-4-[[(2R)-1-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]propanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxopropan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C122H189N37O35
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0534894
|
(3R)-4-[[(2R)-6-amino-1-[2-[2-[2-[3-[[(5S)-6-amino-5-[3-[2-[2-[2-[[(2R)-6-amino-2-[[(2R)-2-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]hexanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-6-oxohexyl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-1-oxohexan-2-yl]amino]-3-[[(2R)-1-[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoic acid
Show/Hide
|
C122H189N33O35
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0540666
|
(2S)-2,6-bis[3-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C52H97N13O19
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0564710
|
(2S)-2,6-bis[3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C110H179N23O35
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0564712
|
(2S)-2,6-bis[3-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C86H131N23O23
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0565270
|
(2S)-2,6-bis[3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[(2R)-2-[[(2R)-2-[[2-[[(2R)-2-amino-4-methylpentanoyl]amino]acetyl]amino]propanoyl]amino]-3-hydroxypropanoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexanamide
Show/Hide
|
C76H145N13O31
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
