| Compound ID |
Compound Name |
Compound Formula |
|
CP0016718
|
8-[6-(2-methoxyethylcarbamoyl)-2-methylpyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C20H20N4O4S2
|
1
|
| 1 |
EC50 = 0.35 nM
|
|
|
|
CP0027462
|
8-(6-acetamidopyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C17H14N4O3S2
|
1
|
| 1 |
EC50 = 0.4 nM
|
|
|
|
CP0016912
|
8-[6-(methylamino)pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H14N4O2S2
|
1
|
| 1 |
EC50 = 0.58 nM
|
|
|
|
CP0024578
|
8-phenoxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H12N2O2S2
|
1
|
| 1 |
EC50 = 0.77 nM
|
|
|
|
CP0023952
|
8-[6-(2-methoxyethylcarbamoyl)pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C19H18N4O4S2
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0030415
|
8-(6-carbamoylpyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H12N4O3S2
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0016917
|
8-[6-(2-ethoxyethylcarbamoyl)pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C20H20N4O4S2
|
1
|
| 1 |
EC50 = 1.5 nM
|
|
|
|
CP0027478
|
8-(2-methylpyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3O2S2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0016918
|
8-(6-aminopyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C15H12N4O2S2
|
1
|
| 1 |
EC50 = 2.3 nM
|
|
|
|
CP0029602
|
8-[6-(methylcarbamoyl)pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C17H14N4O3S2
|
1
|
| 1 |
EC50 = 2.6 nM
|
|
|
|
CP0029592
|
8-(6-methylpyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3O2S2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0030416
|
8-pyridin-3-yloxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C15H11N3O2S2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0022922
|
8-[6-[(2-hydroxy-2-methylpropyl)carbamoyl]pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C20H20N4O4S2
|
1
|
| 1 |
EC50 = 7.4 nM
|
|
|
|
CP0016911
|
8-(2-methyl-1-oxidopyridin-1-ium-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3O3S2
|
1
|
| 1 |
EC50 = 8.3 nM
|
|
|
|
CP0021499
|
8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C11H10N2OS3
|
1
|
| 1 |
EC50 = 8.9 nM
|
|
|
|
CP0024801
|
8-methoxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C11H10N2O2S2
|
1
|
| 1 |
EC50 = 9.1 nM
|
|
|
|
CP0016919
|
8-(4-methylpyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3O2S2
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0027468
|
8-[6-(dimethylcarbamoyl)pyridin-3-yl]oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C18H16N4O3S2
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0022319
|
1-methyl-8-methylsulfanyl-4,5-dihydrothieno[3,4-g]indazole-6-carboxamide
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|
C12H13N3OS2
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0023949
|
8-(5-methylpyridin-3-yl)oxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3O2S2
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0022318
|
8-pyridin-2-yloxy-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C15H11N3O2S2
|
1
|
| 1 |
EC50 = 66 nM
|
|
|
|
CP0027460
|
8-methylsulfinyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C11H10N2O2S3
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0029601
|
N-methyl-8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C12H12N2OS3
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0020244
|
8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzoxazole-6-carboxamide
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|
C11H10N2O2S2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0032209
|
8-methylsulfonyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C11H10N2O3S3
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0030137
|
8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carbonitrile
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|
C11H8N2S3
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0016915
|
8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2,3]benzothiadiazole-6-carboxamide
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|
C10H9N3OS3
|
1
|
| 1 |
EC50 = 550 nM
|
|
|
|
CP0027461
|
8-methylsulfanyl-N-(1,2-thiazol-3-yl)-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C14H11N3OS4
|
1
|
| 1 |
EC50 = 620 nM
|
|
|
|
CP0027479
|
8-methylsulfanyl-N-(1,2-oxazol-3-yl)-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C14H11N3O2S3
|
1
|
| 1 |
EC50 = 890 nM
|
|
|
|
CP0016916
|
8-methylsulfanyl-4,5-dihydro-1H-thieno[3,4-g]indazole-6-carboxamide
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|
C11H11N3OS2
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0023950
|
N-(1-methylpyrazol-3-yl)-8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C15H14N4OS3
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0030140
|
N,N-dimethyl-8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C13H14N2OS3
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0020240
|
8-methylsulfanyl-N-pyridin-2-yl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
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|
C16H13N3OS3
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0022561
|
2-methyl-8-methylsulfanyl-4,5-dihydrothieno[3,4-g]indazole-6-carboxamide
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|
C12H13N3OS2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0023951
|
8-methylsulfanyl-N-phenyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxamide
Show/Hide
|
C17H14N2OS3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0029593
|
8-methylsulfanyl-4,5-dihydrothieno[3,4-g][1,2]benzothiazole-6-carboxylic acid
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|
C11H9NO2S3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0001577
|
N-methyl-3-[(1-methylindazol-5-yl)methyl]-2H-indazole-5-carboxamide
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|
C18H17N5O
|
1
|
| 1 |
IC50 = 49 nM
|
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|
