Compound ID |
Compound Name |
Compound Formula |
CP0462443
|
2-chloro-4-[5-cyano-6-[4-[(2R)-3,3,3-trifluoro-2-hydroxy-2-phenylpropanoyl]piperazin-1-yl]pyridin-3-yl]-N,N-dimethylbenzamide
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|
C28H25ClF3N5O3
|
1
|
1 |
EC50 = 7 nM
|
|
|
CP0003740
|
N-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide
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|
C17H12F9NO3S
|
1
|
1 |
EC50 = 20 nM
|
|
|
CP0535792
|
2-chloro-N,N-dimethyl-4-[4-[1-[(2R)-3,3,3-trifluoro-2-hydroxy-2-phenylpropanoyl]piperidin-4-yl]piperidin-1-yl]benzamide
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|
C28H33ClF3N3O3
|
1
|
1 |
EC50 = 550 nM
|
|
|
CP0380333
|
tert-butyl 4-[5-[3-chloro-4-(dimethylcarbamoyl)phenyl]-3-cyanopyridin-2-yl]piperazine-1-carboxylate
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|
C24H28ClN5O3
|
1
|
1 |
EC50 = 770 nM
|
|
|
CP0429275
|
2-chloro-4-[4-[1-[(2S)-2-hydroxy-3-methyl-2-(trifluoromethyl)butanoyl]piperidin-4-yl]piperidin-1-yl]-N,N-dimethylbenzamide
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|
C25H35ClF3N3O3
|
1
|
1 |
EC50 = 840 nM
|
|
|