alpha-borano-2-Mes-ATP

({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid

US9120798, 7

US9120798, 15

US9120798, Comparator 2

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(5-pyrazin-2-yl-1,3,4-thiadiazol-2-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[[5-(2,5-dimethylpyrazol-3-yl)-1,3,4-thiadiazol-2-yl]amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

US9120798, Comparator 4

US9120798, Comparator 3

US9120798, 9

1-[2-(1H-indol-2-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

US9120798, 14

1-[2-(1H-indol-2-yl)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

US9120798, Comparator 1

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

(2R,3S,4S)-2-Ethyl-3-methyl-N-[3,5-(chloro)phenyl]-4-(phenylamino)-3,4-dihydro-1(2H)-quinolinecarboxamide

1-(2-(2-isopropylphenyl)benzofuran-7-yl)-3-(4-pentylphenyl)urea

((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(4-methoxyphenyl)methanone

(4-bromophenyl)((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)methanone

(2R,3S,4S)-N-(3,5-dimethoxyphenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

(2R,3S,4S)-N-(3-bromophenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

(2R,3S,4S)-N-(3-chlorophenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(4-(trifluoromethoxy)phenyl)methanone

(4-chlorophenyl)((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)methanone

1-(4-tert-butylphenyl)-3-(2-(2-isopropylphenyl)benzofuran-7-yl)urea

((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(4-nitrophenyl)methanone

(2R,3S,4S)-2-ethyl-3-methyl-N-phenyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

(2R,3S,4S)-2-ethyl-N-(3-methoxyphenyl)-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

1-(2-(2-isopropylphenyl)benzofuran-7-yl)-3-(4-methyl-3-(trifluoromethyl)phenyl)urea

(2R,3S,4S)-N-(4-chlorophenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

1-(4-chlorophenyl)-3-(2-(2-isopropylphenyl)benzofuran-7-yl)urea

1-(4-butoxyphenyl)-3-(2-(2-isopropylphenyl)benzofuran-7-yl)urea

[(2R,4S)-4-anilino-2-ethyl-3,4-dihydro-2H-quinolin-1-yl]-(4-methoxyphenyl)methanone

1-(2-(2-isopropylphenyl)benzofuran-7-yl)-3-(4-(trifluoromethoxy)phenyl)urea

1-(2-(2-tert-butylphenyl)benzofuran-7-yl)-3-(4-(trifluoromethoxy)phenyl)urea

1-(2-(2-isopropylphenyl)benzofuran-7-yl)-3-(3-(trifluoromethyl)phenyl)urea

(2R,3S,4S)-2-ethyl-N-(4-methoxyphenyl)-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

1-(4-(trifluoromethoxy)phenyl)-3-(2-(2-(trifluoromethyl)phenyl)benzofuran-7-yl)urea

(4-methoxyphenyl)((3R,4S)-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)methanone

1-(4-(dimethylamino)phenyl)-3-(2-(2-isopropylphenyl)benzofuran-7-yl)urea

(2S,3R,4R)-N-(3,5-dichlorophenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

((2R,3R,4S)-2-ethyl-3-methyl-4-(methyl(phenyl)amino)-3,4-dihydroquinolin-1(2H)-yl)(4-methoxyphenyl)methanone

(2R,3S,4S)-N-(2-chlorophenyl)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinoline-1(2H)-carboxamide

((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(phenyl)methanone

(S)-(4-methoxyphenyl)(4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)methanone

((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(3-(trifluoromethoxy)phenyl)methanone

[(2R,4R)-4-anilino-2-ethyl-3,4-dihydro-2H-quinolin-1-yl]-(4-methoxyphenyl)methanone

1-(2-(2-isopropoxyphenyl)benzofuran-7-yl)-3-(4-(trifluoromethoxy)phenyl)urea

1-(2-(2-chlorophenyl)benzofuran-7-yl)-3-(4-(trifluoromethoxy)phenyl)urea

1-(4-(trifluoromethoxy)phenyl)-3-(2-(3-(trifluoromethyl)phenyl)benzofuran-7-yl)urea

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[1'-(2,2-dimethylpropyl)spiro[2,3-dihydroquinoline-4,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

ethyl 2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-4-(trifluoromethyl)-1,3-thiazole-5-carboxylate

1'-(2,2-dimethylpropyl)-4-fluoro-1-[2-[[5-[4-(trifluoromethoxy)phenyl]-1,3,4-thiadiazol-2-yl]amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-indole-3,3'-pyrrolidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(2-spiro[2H-indole-3,1'-cyclohexane]-1-ylphenyl)-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(3-phenyl-1,2,4-thiadiazol-5-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(5-phenyl-1,3,4-oxadiazol-2-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-(2-spiro[2H-indole-3,1'-cyclopentane]-1-ylphenyl)-3-[4-(trifluoromethoxy)phenyl]urea

1-(4-tert-butylphenyl)-3-[2-(2-propan-2-ylphenoxy)pyridin-3-yl]urea

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-(4-methylphenyl)urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[4-(trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(2-fluorophenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-4-(trifluoromethyl)-1,3-thiazol-2-amine

1-[2-(4,4-dimethyl-2,3-dihydroquinolin-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(2-spiro[2H-indole-3,1'-cyclobutane]-1-ylphenyl)-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-(4-tert-butylphenyl)urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(3-methoxyphenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(4-methoxyphenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(4-methylphenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

1-[2-[4-chloro-1'-(2,2-dimethylpropyl)-7-hydroxyspiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-(5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl)urea

methyl 1-[2-[[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)-7-hydroxyspiro[2H-indole-3,4'-piperidine]-4-carboxylate

1-[2-(3,3-dimethyl-2H-indol-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1'-(2,2-dimethylpropyl)-1-[2-[(5-phenyl-1,3,4-thiadiazol-2-yl)amino]phenyl]-4-(trifluoromethyl)spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-[[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)-7-hydroxyspiro[2H-indole-3,4'-piperidine]-4-carbonitrile

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[4-(trifluoromethoxy)phenyl]-1,3,4-thiadiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,3,4-thiadiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-(2-methylphenyl)-4-(trifluoromethyl)-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-methyl-4-(trifluoromethyl)-1,3-thiazol-2-amine

1-[2-[[2-(2,2-dimethylpropyl)-3,4-dihydro-1H-isoquinolin-5-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-pyrrolo[2,3-c]pyridine-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[3-[3-(dimethylamino)-2,2-dimethylpropoxy]phenyl]-4-(trifluoromethyl)-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-4-ethyl-5-phenyl-1,3-thiazol-2-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[4-(trifluoromethoxy)phenyl]-4-(trifluoromethyl)-1,3-thiazol-2-amine

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-indole-3,3'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

4-[2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-4-(trifluoromethyl)-1,3-thiazol-5-yl]benzonitrile

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[[5-[4-(trifluoromethoxy)phenyl]-1,3,4-thiadiazol-2-yl]amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

4-chloro-1-[2-[[5-(4-chlorophenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-7-ol

methyl 1-[2-[[4-(trifluoromethoxy)phenyl]carbamoylamino]phenyl]spiro[2H-indole-3,4'-piperidine]-1'-carboxylate

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethyl)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,3-thiazol-2-amine

1-[2-(2-propan-2-ylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[2-[1-(2,2-dimethylpropyl)piperidin-4-yl]phenoxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(4,4-dimethyl-2,3-dihydroquinolin-1-yl)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

4-chloro-1-[2-[[5-(3-chlorophenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-7-ol

1'-(2,2-dimethylpropyl)-4-(trifluoromethyl)-1-[2-[[5-[4-(trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-yl]amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(5-phenyl-1,3-thiazol-2-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-(2,4-difluorophenyl)urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-naphthalen-2-yl-1,3,4-thiadiazol-2-amine

1-[2-(1'-benzylspiro[2H-indole-3,4'-piperidine]-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,2-oxazol-3-amine

1-[2-(2-tert-butylphenyl)sulfanylpyridin-3-yl]-3-(4-methylphenyl)urea

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(4-phenyl-1,3-thiazol-2-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-(3,3-dimethyl-2H-indol-1-yl)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[1'-(2-methylpropyl)spiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(4-methoxyphenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-pyridin-2-yl-1,3,4-thiadiazol-2-amine

2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-4-(trifluoromethyl)-1,3-thiazole-5-carbonitrile

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-phenyl-1,2-oxazol-5-amine

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-phenyl-1,2,4-thiadiazol-5-amine

1-(2-spiro[2H-indole-3,1'-cyclopropane]-1-ylphenyl)-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)-4-(trifluoromethyl)spiro[2H-indole-3,4'-piperidine]-7-ol

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[4-(dimethylamino)phenyl]-1,3,4-thiadiazol-2-amine

1-(2,4-difluorophenyl)-3-[2-(2-propan-2-ylphenoxy)pyridin-3-yl]urea

1-(4-phenylphenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

4-chloro-1-[2-[[5-(2-chlorophenyl)-1,3,4-thiadiazol-2-yl]amino]phenyl]-1'-(2,2-dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-pyrrolo[3,2-b]pyridine-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[[2-(2,2-dimethylpropyl)-1,3-dihydroisoindol-4-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(4-methyl-3,4-dihydro-2H-quinolin-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(4-tert-butylphenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

4-tert-butyl-N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,3-thiazol-2-amine

1-[2-(3-tert-butylphenoxy)pyridin-3-yl]-3-(2,4-difluorophenyl)urea

1-[2-(3,4-dihydro-2H-quinolin-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

benzyl 1-[2-[[4-(trifluoromethoxy)phenyl]carbamoylamino]phenyl]spiro[2H-indole-3,4'-piperidine]-1'-carboxylate

1-[2-(2,2-dimethyl-3H-1,4-benzoxazin-4-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-phenylurea

2-(2-tert-butylphenoxy)-N-(1-methyl-5-phenylpyrazol-3-yl)pyridin-3-amine

1-(2-fluorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-(4-methylphenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(5-phenylpyrazin-2-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[3-(dimethylamino)phenyl]-1,3,4-thiadiazol-2-amine

1-[2-[(2-benzyl-3,4-dihydro-1H-isoquinolin-5-yl)oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[(3-tert-butyl-2-methyl-1,3-dihydroisoindol-4-yl)oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,3-oxazol-2-amine

1-[2-[[2-(2-methylpropyl)-3,4-dihydro-1H-isoquinolin-5-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(2,3-dihydro-1,4-benzoxazin-4-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[(5-phenyl-1,2-oxazol-3-yl)amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-[[2-(2-methylpropyl)-1,3-dihydroisoindol-4-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(4-chlorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,3,4-oxadiazol-2-amine

1-(2,4-difluorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-(2,4-difluorophenyl)-3-[2-(2-ethylphenoxy)pyridin-3-yl]urea

1-(3,4-dichlorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

ethyl 5-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-1,3,4-thiadiazole-2-carboxylate

1-[2-(4-methyl-2,3-dihydroquinoxalin-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[2-(1-benzylpiperidin-4-yl)phenoxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(3-chlorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-(4-fluorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-[2-[2-[1-(2-methylpropyl)piperidin-4-yl]phenoxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-(3,5-dichlorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-phenyl-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-(2,4-difluorophenyl)-3-[2-[2-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

1-[2-(2-tert-butylanilino)pyridin-3-yl]-3-(4-methylphenyl)urea

2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-N,N-dimethyl-5-phenyl-1,3-thiazole-4-carboxamide

1-[2-[[2-(3,3-dimethylbutyl)-3,4-dihydro-1H-isoquinolin-5-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

3-[2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-4-(trifluoromethyl)-1,3-thiazol-5-yl]phenol

N-propan-2-yl-1-[2-[[4-(trifluoromethoxy)phenyl]carbamoylamino]phenyl]spiro[2H-indole-3,4'-piperidine]-1'-carboxamide

3-[2-[[2-(2-tert-butylphenoxy)pyridin-3-yl]amino]-5-phenyl-1,3-thiazol-4-yl]-3-methylbutanoic acid

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-[4-[(dimethylamino)methyl]phenyl]-1,3,4-thiadiazol-2-amine

1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-pyrrolo[2,3-b]pyridine-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-[[2-[(2-hydroxyphenyl)methyl]-3,4-dihydro-1H-isoquinolin-5-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-pyridin-4-yl-1,3,4-thiadiazol-2-amine

1-[2-[[2-(2-phenylethyl)-3,4-dihydro-1H-isoquinolin-5-yl]oxy]pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[2-(1'-propan-2-ylspiro[2H-indole-3,4'-piperidine]-1-yl)phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

1-[4-(trifluoromethoxy)phenyl]-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-pyridin-3-yl-1,3,4-thiadiazol-2-amine

4-chloro-1'-(2,2-dimethylpropyl)-1-[2-[[5-(4-methylphenyl)pyridin-2-yl]amino]phenyl]spiro[2H-indole-3,4'-piperidine]-7-ol

1-[2-[1'-(2-methoxyethyl)spiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea

N-[2-(2-tert-butylphenoxy)pyridin-3-yl]-5-phenyl-1,2,4-oxadiazol-3-amine