Brief Information of the Cell Line and Protein
Cell Line ID: CL000030 , LCL Orang Asli K28
Synonyms
K28
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_C8AT
Protein ID: PT01846 , Neuronal acetylcholine receptor subunit alpha-7
Gene Name CHRNA7
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID P36544
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000030  Protein ID: PT01846
 
Compound ID Compound Name Compound Formula
CP0004216
(S)-3-(azetidin-2-ylmethoxy)pyridine
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C9H12N2O
 1
1
Ki = 148 nM
   TI
   LI
   LO
   TS
CP0304433
3-((R)-1-Azetidin-2-ylmethoxy)-pyridine
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C9H12N2O
 1
1
Ki = 1275 nM
   TI
   LI
   LO
   TS
CP0005847
3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridine
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C11H16N2O
 1
1
Ki = 1530 nM
   TI
   LI
   LO
   TS
CP0000063
CAS_29790-52-1
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C10H14N2
 1
1
Ki = 1610 nM
   TI
   LI
   LO
   TS
CP0009737
(S)-1-Methyl-2-(3-methyl-isoxazol-5-yl)-pyrrolidinium
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C9H14N2O
 1
1
Ki = 4050 nM
   TI
   LI
   LO
   TS
CP0002027
2-Methyl-3-((S)-1-pyrrolidin-2-ylmethoxy)-pyridine
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C11H16N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0002657
2-Methyl-3-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-pyridine
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C12H18N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0514441
2-Methyl-3-((R)-1-pyrrolidin-2-ylmethoxy)-pyridine
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C11H16N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0535603
2-Methyl-3-((R)-1-methyl-pyrrolidin-2-ylmethoxy)-pyridine
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C12H18N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS