Compound ID |
Compound Name |
Compound Formula |
CP0443260
|
2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide
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|
C21H26N4O2
|
1
|
1 |
Ki = 6.68 nM
|
|
|
CP0443262
|
N,N-diethyl-2-[2-(4-methoxyphenyl)-5,7-dimethylimidazo[4,5-b]pyridin-3-yl]acetamide
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|
C21H26N4O2
|
1
|
1 |
Ki = 144.33 nM
|
|
|
CP0508581
|
N,N-diethyl-2-[2-(4-methoxyphenyl)-4,6-dimethylbenzimidazol-1-yl]acetamide
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|
C22H27N3O2
|
1
|
1 |
Ki = 398.18 nM
|
|
|
CP0443261
|
N,N-diethyl-2-[2-(4-methoxyphenyl)-4,6-dimethylindol-1-yl]acetamide
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|
C23H28N2O2
|
1
|
1 |
Ki = 806 nM
|
|
|
CP0458452
|
N,N-diethyl-2-[8-(4-methoxyphenyl)-2,6-dimethylpurin-9-yl]acetamide
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|
C20H25N5O2
|
1
|
1 |
Ki > 10000 nM
|
|
|