Brief Information of the Cell Line and Protein
Cell Line ID: CL000941 , CHO-DUKX-A2
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_1977
Protein ID: PT01658 , Oxytocin receptor
Gene Name OXTR
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P30559
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000941  Protein ID: PT01658
 
Compound ID Compound Name Compound Formula
CP0117986
(2S)-1-[(4R,7S,10S,13S,16S,19R)-19-amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-[(2S)-butan-2-yl]-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
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C43H66N12O12S2
 2
1
EC50 = 3 nM
   TI
   LI
   LO
   TS
2
Ki = 0.8 nM
   TI
   LI
   LO
   TS
CP0219136
4-[(3,5-dihydroxyphenyl)methyl]-N-[[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,3-c][1,5]benzodiazepine-5-carbonyl)phenyl]methyl]piperazine-1-carboxamide
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C32H35N7O4
 4
1
EC50 = 61 nM
   TI
   LI
   LO
   TS
2
EC50 = 61.3 nM
   TI
   LI
   LO
   TS
3
Ki = 58 nM
   TI
   LI
   LO
   TS
4
Ki = 58.4 nM
   TI
   LI
   LO
   TS