Brief Information of the Cell Line and Protein
Cell Line ID: CL000549 , Namalwa
Synonyms
NAMALWA
Namalwa IV
Namalva
NAMALVA
NWA
NK62a
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0067
Protein ID: PT01654 , Tyrosine-protein kinase Blk
Gene Name BLK
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P51451
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000549  Protein ID: PT01654
 
Compound ID Compound Name Compound Formula
CP0568167
N-[4-methyl-3-[[2-[3-[(1-prop-2-enoylpiperidin-4-yl)amino]anilino]pyrimidin-5-yl]carbamoyl]phenyl]isoquinoline-6-carboxamide
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C36H34N8O3
 1
1
IC50 = 5.5 nM
   TI
   LI
   LO
   TS
CP0550588
N-[3-[[2-[3-[[1-[(E)-4-(dimethylamino)but-2-enoyl]piperidin-4-yl]amino]anilino]pyrimidin-5-yl]carbamoyl]-4-methylphenyl]isoquinoline-6-carboxamide
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C39H41N9O3
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0113747
2-methyl-N-[2-[3-(prop-2-enoylamino)anilino]pyrimidin-5-yl]-5-[[3-(trifluoromethyl)benzoyl]amino]benzamide
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C29H23F3N6O3
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0550589
N-[4-methyl-3-[[2-[3-(prop-2-enoylamino)anilino]pyrimidin-5-yl]carbamoyl]phenyl]isoquinoline-6-carboxamide
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C31H25N7O3
 1
1
IC50 = 63 nM
   TI
   LI
   LO
   TS