Compound ID |
Compound Name |
Compound Formula |
CP0420961
|
4-[(R)-amino(phenyl)methyl]-N-(6-hydroxy-1,3-benzothiazol-2-yl)benzamide
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|
C21H17N3O2S
|
2
|
1 |
IC50 = 9 nM
|
|
|
2 |
IC50 = 200 nM
|
|
|
CP0040598
|
2-[6-[4-(2-chloro-5-fluorophenoxy)piperidin-1-yl]pyridazin-3-yl]-5-methyl-1,3,4-oxadiazole
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|
C18H17ClFN5O2
|
1
|
1 |
IC50 < 10 nM
|
|
|
CP0420962
|
4-[(R)-amino(phenyl)methyl]-N-(6-methoxy-1,3-benzothiazol-2-yl)benzamide
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|
C22H19N3O2S
|
3
|
1 |
IC50 = 27 nM
|
|
|
2 |
IC50 = 2100 nM
|
|
|
3 |
IC50 > 10000 nM
|
|
|
CP0532063
|
4-[(R)-amino(phenyl)methyl]-N-(1,3-benzothiazol-2-yl)benzamide
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|
C21H17N3OS
|
2
|
1 |
IC50 = 1200 nM
|
|
|
2 |
IC50 = 6700 nM
|
|
|