Compound ID |
Compound Name |
Compound Formula |
CP0094782
|
2-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-propyl}-2H-naphtho[1,8-cd]isothiazole 1,1-dioxide
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|
C23H24FN3O2S
|
1
|
1 |
Ki = 0.06 nM
|
|
|
CP0075436
|
(2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-4-yl}-methanol
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|
C22H28FNO3
|
1
|
1 |
Ki = 0.1 nM
|
|
|
CP0040626
|
1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperidine
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|
C19H21F2NO2S
|
1
|
1 |
Ki = 0.18 nM
|
|
|
CP0511470
|
4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-phenyl)-ethyl]-piperidine
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|
C19H20ClF2NO2S
|
1
|
1 |
Ki = 0.25 nM
|
|
|
CP0376926
|
1-(4-fluorophenyl)-4-[6-methoxyspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-1-yl]-1-butanone
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|
C24H28FNO3
|
1
|
1 |
Ki = 0.38 nM
|
|
|
CP0245024
|
1-(4-Fluorophenyl)-2-[4-(phenylsulfonyl)-1-piperidinyl]-ethanone
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|
C19H20FNO3S
|
1
|
1 |
Ki = 0.51 nM
|
|
|
CP0430154
|
3-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
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|
C20H20F2N2O2S
|
1
|
1 |
Ki = 0.54 nM
|
|
|
CP0371095
|
1'-phenethylspiro[1,2,3,4-tetrahydronaphthalene-2,4'-(hexahydropyridine)]-1-ol; hydrochloride
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|
C22H27NO
|
1
|
1 |
Ki = 0.59 nM
|
|
|
CP0345192
|
1'-[2-(2,4-Difluorophenyl)ethyl]-3,4-dihydrospiro[2H-1-benzothiopyran-2,4'-piperidine]-1,1-dioxide
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|
C21H23F2NO2S
|
1
|
1 |
Ki = 0.61 nM
|
|
|
CP0371094
|
1'-(2,4-difluorophenethyl)-6-methoxyspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C22H25F2NO2
|
1
|
1 |
Ki = 0.69 nM
|
|
|
CP0039097
|
1'-(2,4-difluorophenethyl)spiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C21H23F2NO
|
1
|
1 |
Ki = 0.72 nM
|
|
|
CP0371096
|
4-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzamide
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|
C20H22F2N2O3S
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0347888
|
4-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
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|
C20H20F2N2O2S
|
1
|
1 |
Ki = 1.5 nM
|
|
|
CP0460835
|
1'-phenethylspiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C21H25NO
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0376936
|
1'-(2,4-difluorophenethyl)-8-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C21H22F3NO
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0437526
|
1'-(2,4-difluorophenethyl)-7-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C21H22F3NO
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0460927
|
4-(4-Benzenesulfonyl-piperidin-1-yl)-1-(4-fluoro-phenyl)-butan-1-one
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|
C21H24FNO3S
|
1
|
1 |
Ki = 3.3 nM
|
|
|
CP0448560
|
1'-(2,4-difluorophenethyl)-5-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]
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|
C21H22F3NO
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0039100
|
2-[[1-(2-(2,4-Difluorophenyl)ethyl)-4-piperidinyl]sulfonyl]benzonitrile
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|
C20H20F2N2O2S
|
1
|
1 |
Ki = 4.8 nM
|
|
|
CP0126146
|
6-[[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]methyl]-6,7-dihydro-5H-1-benzofuran-4-one
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|
C21H21FN2O3
|
1
|
1 |
Ki = 5.495 nM
|
|
|
CP0802170
|
6-Fluoro-3-(4-fluoro-piperidin-3-yl)-2-phenyl-1H-indole
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|
C19H18F2N2
|
1
|
1 |
Ki = 12 nM
|
|
|
CP0376502
|
6-chloro-1'-phenethylspiro[1,2,3,4-tetrahydronaphthalene-2,4'-(hexahydropyridine)]-1-one
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|
C22H24ClNO
|
1
|
1 |
Ki = 25 nM
|
|
|
CP0448533
|
1-[6-fluorospiro[3,4-dihydro-2H-chromene-2,4'-(hexahydropyridine)]-1-yl]-4-phenyl-2-butanol
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|
C23H28FNO2
|
1
|
1 |
Ki = 29 nM
|
|
|