Compound ID |
Compound Name |
Compound Formula |
CP0043316
|
3-[5-(cyclohexylamino)-6-(1-methylpyrazol-4-yl)-1H-indazol-3-yl]benzenesulfonamide
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|
C23H26N6O2S
|
1
|
1 |
IC50 = 20.5 nM
|
|
|
CP0043317
|
N-[3-[5-(cyclohexylamino)-6-(1-methylpyrazol-4-yl)-1H-indazol-3-yl]phenyl]acetamide
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|
C25H28N6O
|
1
|
1 |
IC50 = 30.4 nM
|
|
|
CP0153938
|
3-[5-cyclohexyloxy-6-(1-methylpyrazol-4-yl)-1H-indazol-3-yl]benzenesulfonamide
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|
C23H25N5O3S
|
1
|
1 |
IC50 = 74 nM
|
|
|
CP0066304
|
3-[5-ethoxy-6-(1-methylpyrazol-4-yl)-1H-indazol-3-yl]benzenesulfonamide
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|
C19H19N5O3S
|
1
|
1 |
IC50 = 85.8 nM
|
|
|
CP0153937
|
5-[5-ethoxy-6-(1-methylpyrazol-4-yl)-1H-indazol-3-yl]-2-methylbenzenesulfonamide
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|
C20H21N5O3S
|
1
|
1 |
IC50 = 198 nM
|
|
|
CP0166315
|
3-[5-ethoxy-6-(1H-pyrazol-4-yl)-1H-indazol-3-yl]benzenesulfonamide
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|
C18H17N5O3S
|
1
|
1 |
IC50 = 2070 nM
|
|
|
CP0095170
|
3-(5-ethoxy-1H-indazol-3-yl)benzenesulfonamide
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|
C15H15N3O3S
|
1
|
1 |
IC50 = 2740 nM
|
|
|
CP0085315
|
3-(6-cyano-5-ethoxy-1H-indazol-3-yl)benzenesulfonamide
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|
C16H14N4O3S
|
1
|
1 |
IC50 = 3350 nM
|
|
|
CP0266351
|
3-[5-ethoxy-6-[1-(2-methylpropyl)pyrazol-4-yl]-1H-indazol-3-yl]benzenesulfonamide
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|
C22H25N5O3S
|
1
|
1 |
IC50 = 4110 nM
|
|
|
CP0043325
|
N-[3-(6-cyano-5-ethoxy-1H-indazol-3-yl)phenyl]acetamide
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|
C18H16N4O2
|
1
|
1 |
IC50 = 9720 nM
|
|
|
CP0153939
|
3-(5-ethoxy-6-phenyl-1H-indazol-3-yl)benzenesulfonamide
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|
C21H19N3O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
|