| Compound ID |
Compound Name |
Compound Formula |
|
CP0443742
|
N-[3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-methylindol-5-yl]acetamide
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|
C21H19N7O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0204628
|
N-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]-N-methylacetamide
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|
C21H19N7O
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0489848
|
N-[1-[3-cyano-7-(oxetan-3-ylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
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|
C20H17N7O2
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0237741
|
N-[3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1H-indol-5-yl]acetamide
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|
C20H17N7O
|
1
|
| 1 |
IC50 = 77 nM
|
|
|
|
CP0482074
|
7-(cyclopropylamino)-5-[6-(methylsulfonylmethyl)indol-1-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
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|
C20H18N6O2S
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0504780
|
N-[1-[3-cyano-7-(4-hydroxybutylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
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|
C21H21N7O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0521662
|
N-[3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-(3-hydroxypropyl)indol-5-yl]acetamide
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|
C23H23N7O2
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0526090
|
N-[1-[3-cyano-7-(2-morpholin-4-ylethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
Show/Hide
|
C23H24N8O2
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0420972
|
N-[3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-(2-hydroxyethyl)indol-5-yl]acetamide
Show/Hide
|
C22H21N7O2
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0489850
|
N-[1-[3-cyano-7-(2-pyrrolidin-1-ylethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
Show/Hide
|
C23H24N8O
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0459320
|
7-(cyclopropylamino)-5-[6-(hydroxymethyl)indol-1-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
Show/Hide
|
C19H16N6O
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0482075
|
N-[1-[3-cyano-7-(3-pyrrolidin-1-ylpropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
Show/Hide
|
C24H26N8O
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0262754
|
N-[1-[3-cyano-7-[3-(dimethylamino)propylamino]pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamide
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0246588
|
3-[5-acetamido-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-1-yl]propanoic acid
Show/Hide
|
C23H21N7O3
|
1
|
| 1 |
IC50 = 3100 nM
|
|
|
