| Compound ID |
Compound Name |
Compound Formula |
|
CP0474030
|
US10118915, Compound 542
Show/Hide
|
C20H29N5O2
|
1
|
| 1 |
IC50 = 2410 nM
|
|
|
|
CP0421582
|
methyl 5-bromo-2-[(3R,4R)-4-(cyclohexylamino)-3-hydroxypiperidin-1-yl]pyridine-3-carboxylate
Show/Hide
|
C18H26BrN3O3
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0473326
|
US10118915, Compound 233
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 = 4410 nM
|
|
|
|
CP0426012
|
1-[6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C25H32FN5O2
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0439916
|
Btrx-335140
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|
C25H32FN5O2
|
1
|
| 1 |
IC50 = 6500 nM
|
|
|
|
CP0391081
|
1-[6-ethyl-8-fluoro-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-(oxan-4-yl)piperidin-4-amine
Show/Hide
|
C24H30FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0391082
|
1-[6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C24H30FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0391085
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(2S)-3-methylbutan-2-yl]piperidin-4-amine
Show/Hide
|
C24H33N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0391086
|
N-(cyclopropylmethyl)-1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]piperidin-4-amine
Show/Hide
|
C23H29N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0391087
|
1-[6-ethyl-8-fluoro-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C24H30FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0426009
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0473979
|
1-[6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C25H32FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0474031
|
(1S,2S)-2-[[1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]piperidin-4-yl]amino]cyclohexan-1-ol
Show/Hide
|
C25H33N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530129
|
US10118915, Compound 355
Show/Hide
|
C23H31N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530130
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530151
|
US10118915, Compound 285
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530152
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530153
|
US10118915, Compound 433
Show/Hide
|
C22H27N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530197
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0530198
|
1-[6-ethyl-8-fluoro-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C23H28FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0538020
|
1-[6-ethyl-8-fluoro-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3R)-oxan-3-yl]piperidin-4-amine
Show/Hide
|
C24H30FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0538021
|
1-[6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C24H30FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0538022
|
US10118915, Compound 324
Show/Hide
|
C22H29N5O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0545565
|
1-[6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3-methyloxetan-3-yl)methyl]piperidin-4-amine
Show/Hide
|
C24H31N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0550955
|
1-[6-ethyl-8-fluoro-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-[(3S)-oxolan-3-yl]piperidin-4-amine
Show/Hide
|
C23H28FN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417818
|
3-O-ethyl 5-O-methyl 2-[4-[(2-hydroxycyclohexyl)amino]piperidin-1-yl]-6-methylpyridine-3,5-dicarboxylate
Show/Hide
|
C22H33N3O5
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
