| Compound ID |
Compound Name |
Compound Formula |
|
CP0000324
|
2-acetoxyethyl(trimethyl)ammonium;bromide
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|
C7H16NO2+
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0120956
|
3-amino-5-chloro-N-cyclopropyl-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
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|
C13H14ClN3OS
|
1
|
| 1 |
EC50 = 550 nM
|
|
|
|
CP0120957
|
3-amino-5-chloro-4,6-dimethyl-N-(pyridin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxamide
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|
C16H15ClN4OS
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0000753
|
(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-1-[(2S)-2-[[(2S,3R)-2-[[(2S)-2-(hexadecanoylamino)-3-methylbutanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylpentanoyl]pyrrolidine-2-carboxamide
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|
C88H137N17O18
|
2
|
| 1 |
EC50 > 30000 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0066236
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-8-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0366351
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-5-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0666404
|
Tiotropium bromide
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|
C19H24BrNO5S2
|
4
|
| 1 |
IC50 = 0.03162 nM
|
|
|
| 2 |
IC50 = 0.0631 nM
|
|
|
| 3 |
IC50 = 0.2 nM
|
|
|
| 4 |
IC50 = 0.21 nM
|
|
|
|
CP0696953
|
Aclidinium bromide
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|
C26H30BrNO4S2
|
4
|
| 1 |
IC50 < 0.03981 nM
|
|
|
| 2 |
IC50 = 0.1259 nM
|
|
|
| 3 |
IC50 = 0.17 nM
|
|
|
| 4 |
Ki = 0.43 nM
|
|
|
|
CP0705209
|
(3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 0.14 nM
|
|
|
|
CP0428316
|
AHR-504
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|
C19H28NO3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0852883
|
(3R)-3-{[(2S)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.17 nM
|
|
|
|
CP0666488
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C25H28BrNO3S2
|
1
|
| 1 |
IC50 = 0.18 nM
|
|
|
|
CP0918897
|
(3R)-3-{[Hydroxy(di-3-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C26H30BrNO4S2
|
1
|
| 1 |
IC50 = 0.18 nM
|
|
|
|
CP0431075
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-hydroxy(phenyl)2-thienylacetate
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|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.21 nM
|
|
|
|
CP0418147
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-cyclopentyl(hydroxy)2-thienylacetate
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|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0086732
|
(3R)-1-Azabicyclo[2.2.2]oct-3-ylhydroxy(di-2-thienyl)acetate
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|
C17H19NO3S2
|
1
|
| 1 |
IC50 = 0.26 nM
|
|
|
|
CP0397014
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-hydroxy(phenyl)2-thienylacetate
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|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.26 nM
|
|
|
|
CP0851960
|
(3R)-3-{[(9-Methyl-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C31H34BrNO4
|
1
|
| 1 |
IC50 = 0.27 nM
|
|
|
|
CP0893211
|
(3R)-3-{[(2R)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0868135
|
(3R)-3-[(Di-2-thienylacetyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C26H30BrNO3S2
|
1
|
| 1 |
IC50 = 0.35 nM
|
|
|
|
CP0499035
|
(3R)-1-Heptyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
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|
C24H34BrNO3S2
|
1
|
| 1 |
IC50 = 0.36 nM
|
|
|
|
CP0896422
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C30H32BrNO5
|
1
|
| 1 |
IC50 = 0.36 nM
|
|
|
|
CP0874933
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.38 nM
|
|
|
|
CP0217648
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate
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|
C21H23NO3
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0918903
|
(3R)-3-{[Hydroxy(diphenyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C30H34BrNO4
|
1
|
| 1 |
IC50 = 0.44 nM
|
|
|
|
CP0462649
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-methyl-1-azoniabicyclo[2.2.2]octane bromide
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|
C18H22BrNO3S2
|
1
|
| 1 |
IC50 = 0.46 nM
|
|
|
|
CP0860527
|
GLYCOPYRROLATE
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|
C19H28BrNO3
|
2
|
| 1 |
IC50 = 0.5012 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0439371
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-cyclopentyl(hydroxy)2-thienylacetate
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|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.54 nM
|
|
|
|
CP0868133
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C29H30BrNO4
|
1
|
| 1 |
IC50 = 0.54 nM
|
|
|
|
CP0851406
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0859004
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H29BrN2O2S3
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0851961
|
(3R)-3-[(2,2-Di-2-thienylpropanoyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.73 nM
|
|
|
|
CP0864661
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C25H29BrN2O3S2
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0868134
|
(3R)-3-{[(2R)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 1.01 nM
|
|
|
|
CP0874051
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C30H32BrNO4
|
1
|
| 1 |
IC50 = 1.08 nM
|
|
|
|
CP0846167
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
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|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0462648
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9-hydroxy-9H-fluorene-9-carboxylate
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|
C21H21NO3
|
1
|
| 1 |
IC50 = 1.14 nM
|
|
|
|
CP0472694
|
[9-[(3-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0911595
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0387223
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-dithiophen-2-ylacetamide
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|
C17H20N2O2S2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0456356
|
(R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)carbamate
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|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0891026
|
(3R)-1-(2-Phenylethyl)-3-[(9H-xanthen-9-ylcarbonyl)oxy]-1-azoniabicyclo[2.2.2]octane bromide
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|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 1.82 nM
|
|
|
|
CP0070586
|
Ipratropium Bromide
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|
C20H30BrNO3
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 2.24 nM
|
|
|
|
CP0920325
|
(3R)-3-{[(9-Methyl-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrNO3
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0891027
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 2.24 nM
|
|
|
|
CP0391428
|
[9-[(3-methylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-phenylmethanone
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|
C24H30N2O
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0369702
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carboxylate
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
IC50 = 2.83 nM
|
|
|
|
CP0399574
|
[9-[(2-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0454222
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0891718
|
(R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0501199
|
(R)-quinuclidin-3-yl benzyl(phenyl)carbamate
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|
C21H24N2O2
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0846146
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C29H33BrN2O3
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0497828
|
[9-[(3-chlorophenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-phenylmethanone
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|
C23H27ClN2O
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0909075
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
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|
C30H35BrN2O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0441678
|
(2S)-N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-cyclopentyl-2-hydroxy-2-thiophen-2-ylacetamide
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|
C18H26N2O2S
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0505031
|
(3R)-1-Heptyl-3-{[(9-hydroxy-9H-fluoren-9-yl)carbonyl]-oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H36BrNO3
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0456355
|
(R)-quinuclidin-3-yl phenyl(thiophen-3-ylmethyl)carbamate
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 4.7 nM
|
|
|
|
CP0864662
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O3S2
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0497829
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-phenylmethanone
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|
C23H28N2O
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0916859
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H33BrN2O2S
|
1
|
| 1 |
IC50 = 7.6 nM
|
|
|
|
CP0895086
|
(R)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 8.4 nM
|
|
|
|
CP0917225
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O3
|
1
|
| 1 |
IC50 = 8.9 nM
|
|
|
|
CP0502320
|
[9-[(3-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0891721
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H35BrN2O2S
|
1
|
| 1 |
IC50 = 10.9 nM
|
|
|
|
CP0896423
|
(3R)-1-Benzyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
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|
C24H26BrNO3S2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0454523
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-ethyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H26ClN3O2S
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0502914
|
(R)-quinuclidin-3-yl pentyl(phenyl)carbamate
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|
C19H28N2O2
|
1
|
| 1 |
IC50 = 13.6 nM
|
|
|
|
CP0906344
|
(R)-3-((3-fluorophenyl)(3,4,5-trifluorobenzyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H29BrF4N2O3
|
1
|
| 1 |
IC50 = 14.4 nM
|
|
|
|
CP0802380
|
quinuclidin-4-yl biphenyl-2-ylcarbamate hydrochloride
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|
C20H23ClN2O2
|
1
|
| 1 |
IC50 = 14.5 nM
|
|
|
|
CP0391432
|
(9-benzyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H29N3O2S
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0454220
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-thiophen-3-ylmethanone
Show/Hide
|
C21H26N2OS
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0847622
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H37BrN2O2
|
1
|
| 1 |
IC50 = 17.7 nM
|
|
|
|
CP0521412
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C20H23ClN2O2S
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0501201
|
(R)-quinuclidin-3-yl bis(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C18H22N2O2S2
|
1
|
| 1 |
IC50 = 22.7 nM
|
|
|
|
CP0502913
|
(R)-quinuclidin-3-yl butyl(phenyl)carbamate
Show/Hide
|
C18H26N2O2
|
1
|
| 1 |
IC50 = 22.9 nM
|
|
|
|
CP0447654
|
[9-[(2-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 25.12 nM
|
|
|
|
CP0508162
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(furan-2-yl)methanone
Show/Hide
|
C20H23ClN2O3
|
1
|
| 1 |
IC50 = 25.12 nM
|
|
|
|
CP0488363
|
(R)-quinuclidin-3-yl 3-fluorobenzyl(3-fluorophenyl)carbamate
Show/Hide
|
C21H22F2N2O2
|
1
|
| 1 |
IC50 = 26.8 nM
|
|
|
|
CP0912372
|
(R)-1-(2-phenoxyethyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrF3N2O3
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0912371
|
(R)-1-(3-phenylpropyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrF3N2O2
|
1
|
| 1 |
IC50 = 29.8 nM
|
|
|
|
CP0847983
|
(R)-1-(3-phenoxypropyl)-3-(9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H33BrN2O3
|
1
|
| 1 |
IC50 = 29.8 nM
|
|
|
|
CP0454223
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0528622
|
1-benzofuran-5-yl-[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]methanone
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0459214
|
(R)-1-methyl-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C20H25BrN2O2S
|
1
|
| 1 |
IC50 = 33.1 nM
|
|
|
|
CP0398693
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-diphenylacetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 35.1 nM
|
|
|
|
CP0391430
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,2,5-thiadiazol-3-yl)methanone
Show/Hide
|
C18H21ClN4O2S
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0482224
|
(R)-quinuclidin-3-yl phenethyl(phenyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 42.1 nM
|
|
|
|
CP0478198
|
(R)-quinuclidin-3-yl m-tolyl(2,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C22H23F3N2O2
|
1
|
| 1 |
IC50 = 45.8 nM
|
|
|
|
CP0391431
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,3-thiazol-4-yl)methanone
Show/Hide
|
C19H22ClN3O2S
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0398144
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(5-methylfuran-2-yl)methanone
Show/Hide
|
C21H25ClN2O3
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0845813
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H33BrN2O2
|
1
|
| 1 |
IC50 = 50.9 nM
|
|
|
|
CP0673968
|
SID50106181
Show/Hide
|
C21H26INO2
|
2
|
| 1 |
IC50 = 55 nM
|
|
|
| 2 |
Ki = 23 nM
|
|
|
|
CP0454522
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(furan-3-yl)methanone
Show/Hide
|
C20H23ClN2O3
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0071487
|
BENZTROPINE
Show/Hide
|
C21H25NO
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0459211
|
(R)-quinuclidin-3-yl butyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C17H26N2O2S
|
1
|
| 1 |
IC50 = 76.2 nM
|
|
|
|
CP0505885
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl 10,11-dihydro-5H-dibenzo-[a,d][7]annulene-5-carboxylate
Show/Hide
|
C23H25NO2
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0055048
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-(furan-2-yl)methanone
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0435479
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,2-oxazol-3-yl)methanone
Show/Hide
|
C19H22ClN3O3
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0454221
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-(2-ethoxyphenyl)methanone
Show/Hide
|
C25H32N2O2
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0504490
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-pyridin-3-ylmethanone
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0375586
|
(R)-quinuclidin-3-yl benzyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C20H24N2O2S
|
1
|
| 1 |
IC50 = 88.9 nM
|
|
|
|
CP0882813
|
(R)-3-(2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 91.5 nM
|
|
|
|
CP0390751
|
(R)-quinuclidin-3-yl 3-fluorophenyl(3,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C21H20F4N2O2
|
1
|
| 1 |
IC50 = 97.3 nM
|
|
|
|
CP0379242
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9-hydroxyfluorene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 101.1 nM
|
|
|
|
CP0390680
|
(R)-quinuclidin-3-yl benzyl(4-fluorophenyl)carbamate
Show/Hide
|
C21H23FN2O2
|
1
|
| 1 |
IC50 = 115.7 nM
|
|
|
|
CP0903846
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O2
|
1
|
| 1 |
IC50 = 120.8 nM
|
|
|
|
CP0391429
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-[5-(hydroxymethyl)furan-2-yl]methanone
Show/Hide
|
C21H25ClN2O4
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0446893
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-phenylmethanone
Show/Hide
|
C22H25ClN2O2
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0502624
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-pyrimidin-2-ylmethanone
Show/Hide
|
C20H23ClN4O2
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0935343
|
(R)-1-(3-(1H-pyrrol-1-yl)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H34BrN3O2
|
1
|
| 1 |
IC50 = 136.6 nM
|
|
|
|
CP0868278
|
(R)-1-(3-(biphenyl-4-yloxy)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C37H39ClN2O3
|
1
|
| 1 |
IC50 = 140.2 nM
|
|
|
|
CP0478197
|
(R)-quinuclidin-3-yl benzyl(p-tolyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 195.6 nM
|
|
|
|
CP0398694
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2OS2
|
1
|
| 1 |
IC50 = 229.6 nM
|
|
|
|
CP0454381
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-pyrimidin-2-ylmethanone
Show/Hide
|
C21H26N4O
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0469803
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-N-methyl-9H-xanthene-9-carboxamide
Show/Hide
|
C22H24N2O2
|
1
|
| 1 |
IC50 = 285.9 nM
|
|
|
|
CP0411467
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9H-xanthene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 347.6 nM
|
|
|
|
CP0459212
|
(R)-quinuclidin-3-yl phenyl(propyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 349.3 nM
|
|
|
|
CP0846145
|
SOLIFENACIN SUCCINATE
Show/Hide
|
C27H32N2O6
|
1
|
| 1 |
IC50 = 573.7 nM
|
|
|
|
CP0477682
|
1-[(2R)-4-(5-fluoro-3-methylpyridin-2-yl)-2-methylpiperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C24H27FN4O
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0470009
|
[9-[(2-methylphenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C23H31N3O2S
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0472695
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-(3H-1,2-oxazol-2-yl)methanone
Show/Hide
|
C20H27N3O2
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0864660
|
(R)-3-(9-hydroxy-9H-fluorene-9-carboxamido)-1-(3-(methyl(phenyl)amino)propyl)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C31H36ClN3O2
|
1
|
| 1 |
IC50 = 804.2 nM
|
|
|
|
CP0390681
|
(R)-quinuclidin-3-yl isopropyl(phenyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 1364.9 nM
|
|
|
|
CP0477681
|
1-[(2S)-4-(5-fluoro-3-methylpyridin-2-yl)-2-methylpiperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C24H27FN4O
|
1
|
| 1 |
IC50 = 1995.26 nM
|
|
|
|
CP0401466
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0390678
|
(R)-quinuclidin-3-yl diphenylcarbamate
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
IC50 = 2779 nM
|
|
|
|
CP0507717
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-4-methylbenzamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 = 6900 nM
|
|
|
|
CP0372793
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]benzamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0469062
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,4-difluorobenzamide
Show/Hide
|
C19H20ClF2N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0493960
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0514007
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C20H21ClF3N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0398146
|
(2-tert-butyl-1,3-thiazol-4-yl)-[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]methanone
Show/Hide
|
C23H30ClN3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0475752
|
(9-benzyl-2,9-diazaspiro[5.5]undecan-2-yl)-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H27N3OS
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0502600
|
[9-[(4-chlorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H26ClN3OS
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0167280
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid ethyl ester
Show/Hide
|
C28H36N2O5S
|
1
|
| 1 |
Ki = 0.11 nM
|
|
|
|
CP0543095
|
[1-[3-(4-chlorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrClNO3
|
1
|
| 1 |
Ki = 0.11 nM
|
|
|
|
CP0366483
|
1-(isopropylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine
Show/Hide
|
C28H38N2O5S2
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0101233
|
2-(4-Hydroxy-phenyl)-2-phenyl-propionic acid 2-diethylamino-ethyl ester
Show/Hide
|
C21H27NO3
|
1
|
| 1 |
Ki = 0.165 nM
|
|
|
|
CP0080609
|
1-Cyclohexyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-piperidine
Show/Hide
|
C26H33NO3S
|
1
|
| 1 |
Ki = 0.17 nM
|
|
|
|
CP0412104
|
[1-[3-[4-(trifluoromethyl)phenyl]propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H33BrF3NO3
|
1
|
| 1 |
Ki = 0.18 nM
|
|
|
|
CP0575275
|
(2-aminophenyl)-[4-[4-[[4-(3-chlorophenyl)sulfonylphenyl]methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C30H34ClN3O3S
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0362174
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-(3-methylthiophen-2-yl)methanone
Show/Hide
|
C29H32N2O6S2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0274359
|
cyclopropyl-[4-[4-[1-[4-(4-methoxyphenyl)sulfonylphenyl]ethenyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C29H36N2O4S
|
1
|
| 1 |
Ki = 0.26 nM
|
|
|
|
CP0540935
|
2-[2-[6-[8-[6-[bis[2-oxo-2-(6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)ethyl]amino]hexyl-methylamino]octyl-methylamino]hexylamino]acetyl]-2,4,9,15-tetrazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-10-one
Show/Hide
|
C63H76N14O6
|
1
|
| 1 |
Ki = 0.2692 nM
|
|
|
|
CP0209448
|
4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)-1-(propylsulfonyl)piperidine
Show/Hide
|
C28H38N2O5S2
|
1
|
| 1 |
Ki = 0.29 nM
|
|
|
|
CP0203331
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid isobutyl ester
Show/Hide
|
C30H40N2O5S
|
1
|
| 1 |
Ki = 0.3 nM
|
|
|
|
CP0058613
|
CAS_132947
Show/Hide
|
C64H77N13O6
|
1
|
| 1 |
Ki = 0.302 nM
|
|
|
|
CP0177376
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid butyl ester
Show/Hide
|
C30H40N2O5S
|
1
|
| 1 |
Ki = 0.35 nM
|
|
|
|
CP0177381
|
1'-Benzenesulfonyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl
Show/Hide
|
C31H36N2O5S2
|
1
|
| 1 |
Ki = 0.36 nM
|
|
|
|
CP0212797
|
1'-(Butane-1-sulfonyl)-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl
Show/Hide
|
C29H40N2O5S2
|
1
|
| 1 |
Ki = 0.38 nM
|
|
|
|
CP0220544
|
1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)butan-1-one
Show/Hide
|
C29H38N2O4S
|
1
|
| 1 |
Ki = 0.38 nM
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CP0336623
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[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-(2,3-dimethylphenyl)methanone
Show/Hide
|
C32H36N2O6S
|
1
|
| 1 |
Ki = 0.4 nM
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CP0562060
|
[1-(2-phenylsulfanylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C29H32BrNO3S
|
1
|
| 1 |
Ki = 0.4 nM
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CP0177380
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid isopropyl ester
Show/Hide
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C29H38N2O5S
|
1
|
| 1 |
Ki = 0.41 nM
|
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CP0167279
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid benzyl ester
Show/Hide
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C33H38N2O5S
|
1
|
| 1 |
Ki = 0.45 nM
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CP0287765
|
1'-Ethanesulfonyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl
Show/Hide
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C27H36N2O5S2
|
1
|
| 1 |
Ki = 0.46 nM
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CP0548006
|
[1-[3-(4-fluorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrFNO3
|
1
|
| 1 |
Ki = 0.49 nM
|
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CP0882281
|
Tiotropium bromide
Show/Hide
|
C19H22BrNO4S2
|
1
|
| 1 |
Ki = 0.49 nM
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CP0061483
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-quinolin-5-ylmethanone
Show/Hide
|
C33H33N3O6S
|
1
|
| 1 |
Ki = 0.5 nM
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CP0184076
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-naphthalen-1-ylmethanone
Show/Hide
|
C34H34N2O6S
|
1
|
| 1 |
Ki = 0.5 nM
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CP0203327
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid propyl ester
Show/Hide
|
C29H38N2O5S
|
1
|
| 1 |
Ki = 0.59 nM
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CP0426656
|
[1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO4
|
1
|
| 1 |
Ki = 0.68 nM
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CP0528505
|
[1-[3-(3-fluorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrFNO3
|
1
|
| 1 |
Ki = 0.69 nM
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CP0500994
|
methyl 2-[4-[[1-[1-(naphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetate
Show/Hide
|
C31H36N2O3S
|
1
|
| 1 |
Ki = 0.7 nM
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CP0552568
|
[1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO3
|
1
|
| 1 |
Ki = 0.72 nM
|
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CP0425074
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-propyl)-pyrrolidinium
Show/Hide
|
C29H34N3O+
|
1
|
| 1 |
Ki = 0.73 nM
|
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|
CP0245329
|
(2-Amino-3-methyl-phenyl)-{4-[4-(3-chloro-benzenesulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C31H36ClN3O3S
|
1
|
| 1 |
Ki = 0.89 nM
|
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CP0406733
|
naphthalen-1-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C31H38N2OS
|
1
|
| 1 |
Ki = 0.9 nM
|
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CP0540883
|
[1-[3-(4-methoxyphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO4
|
1
|
| 1 |
Ki = 0.91 nM
|
|
|
|
CP0177377
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid methyl ester
Show/Hide
|
C27H34N2O5S
|
1
|
| 1 |
Ki = 0.99 nM
|
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CP0169241
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-quinolin-4-ylmethanone
Show/Hide
|
C33H33N3O6S
|
1
|
| 1 |
Ki = 1 nM
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|
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CP0463215
|
[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]-quinolin-5-ylmethanone
Show/Hide
|
C30H37N3OS
|
1
|
| 1 |
Ki = 1 nM
|
|
|
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CP0540885
|
[(3R)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
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CP0177938
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-[1,4']bipiperidinyl-1'-carboxylic acid phenyl ester
Show/Hide
|
C30H32N2O7S
|
1
|
| 1 |
Ki = 1.1 nM
|
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CP0548236
|
[1-[3-(4-methylphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
|
| 1 |
Ki = 1.1 nM
|
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|
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CP0203329
|
4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(piperidin-4-yl)piperidine
Show/Hide
|
C25H32N2O3S
|
1
|
| 1 |
Ki = 1.14 nM
|
|
|
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CP0516424
|
Flotros
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 1.148 nM
|
|
|
|
CP0421654
|
[1-[3-(3-methylphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0109931
|
ATROPEN
Show/Hide
|
C17H23NO3
|
3
|
| 1 |
Ki = 1.44 nM
|
|
|
| 2 |
Ki = 1.9 nM
|
|
|
| 3 |
Ki = 15.85 nM
|
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CP0212795
|
1-(benzylsulfonyl)-4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidine
Show/Hide
|
C32H38N2O5S2
|
1
|
| 1 |
Ki = 1.45 nM
|
|
|
|
CP0850774
|
METHYLBENACTYZIUM BROMIDE
Show/Hide
|
C21H28BrNO3
|
1
|
| 1 |
Ki = 1.54 nM
|
|
|
|
CP0155384
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-phenylmethanone
Show/Hide
|
C30H32N2O6S
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0345843
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-(propane-1-sulfonyl)-[1,4']bipiperidinyl
Show/Hide
|
C26H34N2O7S2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
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CP0552569
|
[1-[3-(4-bromophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33Br2NO3
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0435669
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
|
| 1 |
Ki = 1.66 nM
|
|
|
|
CP0183105
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-ethanesulfonyl-[1,4']bipiperidinyl
Show/Hide
|
C25H32N2O7S2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0528506
|
[1-[3-(3-chlorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrClNO3
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0855970
|
Mepenzolate
Show/Hide
|
C21H26BrNO3
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
|
CP0203332
|
1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)-2-methylpropan-1-one
Show/Hide
|
C29H38N2O4S
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0552567
|
[1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C29H32BrNO3
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0526055
|
1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
|
| 1 |
Ki = 2.39 nM
|
|
|
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CP0540884
|
[1-[3-[4-(trifluoromethoxy)phenyl]propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H33BrF3NO4
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0567616
|
[4-[4-[[4-(3-chlorophenyl)sulfonylphenyl]methyl]piperidin-1-yl]piperidin-1-yl]-(2-methylphenyl)methanone
Show/Hide
|
C31H35ClN2O3S
|
1
|
| 1 |
Ki = 2.692 nM
|
|
|
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CP0463222
|
ethyl 2-[4-[[1-[1-(6-ethoxynaphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetate
Show/Hide
|
C34H42N2O4S
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
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CP0177378
|
1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)-2-phenylethanone
Show/Hide
|
C33H38N2O4S
|
1
|
| 1 |
Ki = 2.99 nM
|
|
|
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CP0357762
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-[1,4']bipiperidinyl-1'-carboxylic acid isopropyl ester
Show/Hide
|
C27H34N2O7S
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
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CP0849067
|
11-{2-[[(1S,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 3.467 nM
|
|
|
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CP0177379
|
1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)propan-1-one
Show/Hide
|
C28H36N2O4S
|
1
|
| 1 |
Ki = 3.8 nM
|
|
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CP0858320
|
11-{2-[[(1R,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 3.981 nM
|
|
|
|
CP0225899
|
AQ-RA 741
Show/Hide
|
C27H37N5O2
|
1
|
| 1 |
Ki = 4.266 nM
|
|
|
|
CP0524193
|
methyl 2-[4-[[1-[1-(7-fluoronaphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetate
Show/Hide
|
C31H35FN2O3S
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
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CP0849144
|
11-{2-[[(1R,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 4.467 nM
|
|
|
|
CP0849141
|
11-{2-[[(1S,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 5.37 nM
|
|
|
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CP0468712
|
S-[2-(diethylamino)ethyl] 2-hydroxy-2,2-diphenylethanethioate
Show/Hide
|
C20H25NO2S
|
1
|
| 1 |
Ki = 5.38 nM
|
|
|
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CP0873360
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenethyl-pyrrolidinium bromide
Show/Hide
|
C28H32BrN3O
|
1
|
| 1 |
Ki = 5.4 nM
|
|
|
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CP0468678
|
2-[di(propan-2-yl)amino]ethyl 2-hydroxy-2,2-diphenylacetate
Show/Hide
|
C22H29NO3
|
1
|
| 1 |
Ki = 5.85 nM
|
|
|
|
CP0429216
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-[1,4']bipiperidinyl-1'-carboxylic acid ethyl ester
Show/Hide
|
C26H32N2O7S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0217520
|
AF-DX 384
Show/Hide
|
C27H38N6O2
|
1
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| 1 |
Ki = 6.026 nM
|
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CP0487381
|
[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 6.026 nM
|
|
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CP0453567
|
(6-Isopropoxy-naphthalen-1-yl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C34H44N2O2S
|
1
|
| 1 |
Ki = 6.1 nM
|
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CP0472898
|
N-[2-[2-[(dipropylamino)methyl]piperidin-1-yl]ethyl]-5-oxo-6H-pyrido[3,2-c][1,5]benzodiazepine-11-carboxamide
Show/Hide
|
C27H38N6O2
|
1
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| 1 |
Ki = 6.31 nM
|
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CP0200801
|
4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-(butane-1-sulfonyl)-[1,4']bipiperidinyl
Show/Hide
|
C27H36N2O7S2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
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CP0438023
|
[1-(5-phenylpentyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C32H38BrNO3
|
1
|
| 1 |
Ki = 7.1 nM
|
|
|
|
CP0491603
|
2-(diethylamino)ethyl 2-cyclohexyl-2-hydroxy-2-thiophen-2-ylacetate
Show/Hide
|
C18H29NO3S
|
1
|
| 1 |
Ki = 7.93 nM
|
|
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CP0516427
|
1-[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0500897
|
(7-Fluoro-naphthalen-1-yl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C31H37FN2OS
|
1
|
| 1 |
Ki = 8.6 nM
|
|
|
|
CP0505237
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenoxy-propyl)-pyrrolidinium
Show/Hide
|
C29H34N3O2+
|
1
|
| 1 |
Ki = 8.84 nM
|
|
|
|
CP0543094
|
[1-[3-(3-bromophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33Br2NO3
|
1
|
| 1 |
Ki = 9.2 nM
|
|
|
|
CP0175835
|
Isoptpo Hyoscine
Show/Hide
|
C17H21NO4
|
1
|
| 1 |
Ki = 9.5 nM
|
|
|
|
CP0390370
|
1-[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H23NO2
|
1
|
| 1 |
Ki = 9.772 nM
|
|
|
|
CP0379032
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenylcarbamoylmethyl-pyrrolidinium
Show/Hide
|
C28H31N4O2+
|
1
|
| 1 |
Ki = 9.92 nM
|
|
|
|
CP0530138
|
isoquinolin-1-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C30H37N3OS
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0152464
|
[4-[4-[4-(1,3-benzodioxol-5-ylsulfonyl)phenoxy]piperidin-1-yl]piperidin-1-yl]-quinolin-8-ylmethanone
Show/Hide
|
C33H33N3O6S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0511025
|
N,N-dimethyl-2-[4-[[1-[1-(naphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetamide
Show/Hide
|
C32H39N3O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
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CP0426657
|
[1-(4-phenoxybutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO4
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0434673
|
[1-(3-phenylmethoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO4
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0548005
|
[1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0406396
|
N,N-dimethyl-1-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methanamine
Show/Hide
|
C19H22N2
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0472767
|
(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 12.3 nM
|
|
|
|
CP0401540
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(octahydro-quinolin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C25H41NO2
|
1
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| 1 |
Ki = 13 nM
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CP0421081
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1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine
Show/Hide
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C19H29NO2
|
1
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| 1 |
Ki = 13.18 nM
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CP0436551
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1-(bicyclo[2.2.1]hept-5-en-2-yl)-1-phenyl-3-(piperidin-1-yl)propan-1-ol
Show/Hide
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C21H29NO
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1
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| 1 |
Ki = 13.7 nM
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CP0521081
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[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium
Show/Hide
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C20H32NO2+
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1
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| 1 |
Ki = 13.8 nM
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CP0178308
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4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-(propane-2-sulfonyl)-[1,4']bipiperidinyl
Show/Hide
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C26H34N2O7S2
|
1
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| 1 |
Ki = 14 nM
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CP0451233
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(6-Ethoxy-naphthalen-1-yl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C33H42N2O2S
|
1
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| 1 |
Ki = 14 nM
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CP0185570
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4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-phenylmethanesulfonyl-[1,4']bipiperidinyl
Show/Hide
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C30H34N2O7S2
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1
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| 1 |
Ki = 15 nM
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CP0420726
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2-(diethylamino)ethyl 2-(1-hydroxycyclohexyl)-2-phenylacetate
Show/Hide
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C20H31NO3
|
1
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| 1 |
Ki = 15.1 nM
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CP0375774
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N,N-dimethyl-2-[3-(2-pyridin-2-ylpropan-2-yl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2
|
1
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| 1 |
Ki = 15.49 nM
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CP0483108
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naphthalen-1-yl-[4-[4-[(4-propan-2-ylsulfonylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
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C31H38N2O3S
|
1
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| 1 |
Ki = 17 nM
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CP0183976
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1-{4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-[1,4']bipiperidinyl-1'-yl}-2-ethoxy-ethanone
Show/Hide
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C27H34N2O7S
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1
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| 1 |
Ki = 17.9 nM
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CP0459309
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2-{4-[1'-(Naphthalene-1-carbonyl)-[1,4']bipiperidinyl-4-ylmethyl]-phenylsulfanyl}-acetamide
Show/Hide
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C30H35N3O2S
|
1
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| 1 |
Ki = 18 nM
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CP0502411
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(2-Amino-3-methyl-phenyl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C28H39N3OS
|
1
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| 1 |
Ki = 20 nM
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CP0521168
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[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]-quinolin-4-ylmethanone
Show/Hide
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C30H37N3OS
|
1
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| 1 |
Ki = 20 nM
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CP0540886
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(1-benzyl-1-azoniabicyclo[2.2.2]octan-3-yl) 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
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C28H30BrNO3
|
1
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| 1 |
Ki = 21 nM
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CP0435668
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1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-phenethyl-pyrrolidinium
Show/Hide
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C28H30F2N3O+
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1
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| 1 |
Ki = 21.9 nM
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CP0453319
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(6-Fluoro-naphthalen-1-yl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C31H37FN2OS
|
1
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| 1 |
Ki = 22 nM
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CP0535695
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(4-Fluoro-naphthalen-1-yl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C31H37FN2OS
|
1
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| 1 |
Ki = 22 nM
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CP0381106
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(Adamantan-1-ylamino)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C26H41NO2
|
1
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| 1 |
Ki = 26 nM
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CP0511312
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[4-[4-[[4-(2-hydroxyethylsulfanyl)phenyl]methyl]piperidin-1-yl]piperidin-1-yl]-naphthalen-1-ylmethanone
Show/Hide
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C30H36N2O2S
|
1
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| 1 |
Ki = 26 nM
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CP0511887
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1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-oxiranylmethyl)-pyrrolidinium
Show/Hide
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C29H32N3O2+
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1
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| 1 |
Ki = 27.4 nM
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CP0271112
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N,N-dimethyl-2-[3-[(1S)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
Show/Hide
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C20H24N2
|
1
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| 1 |
Ki = 30.2 nM
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CP0479764
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N-[3-[1-[2-(8-chloro-6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-2-oxoethyl]piperidin-4-yl]propyl]-N-ethyl-2,2-dimethylpentanamide
Show/Hide
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C31H42ClN5O3
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1
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| 1 |
Ki = 30.2 nM
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CP0433507
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(1-methylpiperidin-4-yl) 3-hydroxy-2-[3-(trifluoromethyl)phenyl]propanoate
Show/Hide
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C16H20F3NO3
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1
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| 1 |
Ki = 30.8 nM
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CP0442398
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1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium
Show/Hide
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C28H30N3O2+
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1
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| 1 |
Ki = 31.5 nM
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CP0296594
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(3S,3aR,4R,4aS,8aR,9aS)-4-[2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-ethyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO2
|
1
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| 1 |
Ki = 32.2 nM
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CP0436507
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N-(2-fluoroethyl)-N-methyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H25FN2
|
1
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| 1 |
Ki = 32.36 nM
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CP0403962
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2-[6-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
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C20H23ClN2
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1
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| 1 |
Ki = 33.11 nM
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CP0465680
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(3S)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
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C24H29NO3
|
1
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| 1 |
Ki = 33.11 nM
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CP0183455
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4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-1'-(naphthalene-1-sulfonyl)-[1,4']bipiperidinyl
Show/Hide
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C33H34N2O7S2
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1
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| 1 |
Ki = 34.7 nM
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CP0448858
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ethyl 2-[4-[[1-[1-(naphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetate
Show/Hide
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C32H38N2O3S
|
1
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| 1 |
Ki = 40 nM
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CP0564271
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[(2R,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H32INO2
|
1
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| 1 |
Ki = 43.65 nM
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CP0372479
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N,N-diethyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C22H28N2
|
1
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| 1 |
Ki = 44.67 nM
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CP0405401
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1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-benzyloxy-ethyl)-pyrrolidinium
Show/Hide
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C29H34N3O2+
|
1
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| 1 |
Ki = 47.8 nM
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CP0406734
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propan-2-yl 2-[4-[[1-[1-(naphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetate
Show/Hide
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C33H40N2O3S
|
1
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| 1 |
Ki = 48 nM
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CP0054849
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methyl-6-(S)-methyl-piperidin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H35NO2
|
1
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| 1 |
Ki = 48.4 nM
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CP0453174
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-morpholin-4-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C20H33NO3
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1
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| 1 |
Ki = 51 nM
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CP0403951
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N-methyl-N-[[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methyl]propan-2-amine
Show/Hide
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C21H26N2
|
1
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| 1 |
Ki = 51.29 nM
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CP0414398
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[(2R,5R)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H32INO2
|
1
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| 1 |
Ki = 54.95 nM
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CP0471590
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(3R)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
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C24H29NO3
|
1
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| 1 |
Ki = 57.54 nM
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CP0260958
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1-{4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenoxy]-[1,4']bipiperidinyl-1'-yl}-2-phenoxy-ethanone
Show/Hide
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C31H34N2O7S
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1
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| 1 |
Ki = 59.5 nM
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CP0473020
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[(2R,5S)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H32INO2
|
1
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| 1 |
Ki = 60.26 nM
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CP0489025
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(3S)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
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C24H29NO3
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1
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| 1 |
Ki = 61.66 nM
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CP0473019
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1-[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
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C19H29NO2
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1
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| 1 |
Ki = 67.61 nM
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CP0540888
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[(3S)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
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C30H34BrNO3
|
1
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| 1 |
Ki = 68 nM
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CP0425077
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-thiophen-3-ylethyl)-pyrrolidinium
Show/Hide
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C26H26F2N3O2S+
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1
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| 1 |
Ki = 88.5 nM
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CP0425078
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium
Show/Hide
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C28H28F2N3O2+
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1
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| 1 |
Ki = 94.5 nM
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CP0386733
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[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
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C24H27NO4
|
1
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| 1 |
Ki = 95.5 nM
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CP0475081
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1-[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
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C19H23NO2
|
1
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| 1 |
Ki = 95.5 nM
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CP0436921
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N,N-dimethyl-2-[3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2
|
1
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| 1 |
Ki = 97.72 nM
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CP0459246
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(2-Amino-3-methyl-phenyl)-{4-[4-(propane-2-sulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C28H39N3O3S
|
1
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| 1 |
Ki = 104 nM
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CP0164673
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2,2-Diphenyl-propionic acid 2-diethylamino-ethyl ester
Show/Hide
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C21H27NO2
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1
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| 1 |
Ki = 107 nM
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CP0416602
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2-[6-chloro-3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
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C21H25ClN2
|
1
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| 1 |
Ki = 107.15 nM
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CP0501154
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(4-methoxyphenyl)-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C28H38N2O2S
|
1
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| 1 |
Ki = 108 nM
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CP0405402
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-[2-(3-fluoro-phenyl)-2-oxo-ethyl]-pyrrolidinium
Show/Hide
|
C28H27F3N3O2+
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1
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| 1 |
Ki = 108 nM
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CP0397929
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2-[5-fluoro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H23FN2
|
1
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| 1 |
Ki = 112.2 nM
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CP0433352
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3-(diethylamino)propyl (3S)-3-methyl-2-phenylpentanoate
Show/Hide
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C19H31NO2
|
1
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| 1 |
Ki = 116 nM
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CP0371787
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5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine; oxalic acid
Show/Hide
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C14H23N3OS
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1
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| 1 |
Ki = 120 nM
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CP0002227
|
SOLIFENACIN
Show/Hide
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C23H26N2O2
|
1
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| 1 |
Ki = 120.23 nM
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CP0457284
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4-[4-(4-Isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-carbonyl]-benzenesulfonamide
Show/Hide
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C27H37N3O3S2
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1
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| 1 |
Ki = 129 nM
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CP0448671
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(2,4-Dichloro-phenyl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C27H34Cl2N2OS
|
1
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| 1 |
Ki = 134 nM
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CP0510998
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1,2-oxazol-5-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
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C24H33N3O2S
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1
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| 1 |
Ki = 134 nM
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CP0453595
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4-[4-(4-Methoxy-benzenesulfonyl)-phenoxy]-1'-(propane-1-sulfonyl)-[1,4']bipiperidinyl
Show/Hide
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C26H36N2O6S2
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1
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| 1 |
Ki = 138.8 nM
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CP0449839
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N-methyl-N-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]propan-2-amine
Show/Hide
|
C22H28N2
|
1
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| 1 |
Ki = 144.54 nM
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CP0455460
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3-Hydroxy-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C21H35NO3
|
1
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| 1 |
Ki = 148 nM
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CP0425073
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1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
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| 1 |
Ki = 157 nM
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CP0386735
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[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 158.49 nM
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CP0056034
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11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C19H21N5O2
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1
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| 1 |
Ki = 173.78 nM
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CP0516425
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[(2R)-5,5-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 177.83 nM
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CP0481591
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C25H35NO2
|
1
|
| 1 |
Ki = 184 nM
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CP0502977
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-thiomorpholin-4-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C20H33NO2S
|
1
|
| 1 |
Ki = 189 nM
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CP0443865
|
(2-Chloro-phenyl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C27H35ClN2OS
|
1
|
| 1 |
Ki = 192 nM
|
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CP0472770
|
trimethyl-[[(2R,6R)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 194.98 nM
|
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CP0390368
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 199.53 nM
|
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CP0472768
|
trimethyl-[[(2R,5R)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 199.53 nM
|
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CP0479720
|
[(2R,6R)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO4S
|
1
|
| 1 |
Ki = 199.53 nM
|
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CP0399359
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2-Ethyl-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 209 nM
|
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CP0466978
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,3-Dimethyl-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C23H39NO2
|
1
|
| 1 |
Ki = 224 nM
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CP0397949
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N,N-dimethyl-2-[3-[phenyl(pyridin-2-yl)methyl]-1H-inden-2-yl]ethanamine
Show/Hide
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C25H26N2
|
1
|
| 1 |
Ki = 229.09 nM
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CP0397931
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N,N-dimethyl-2-[3-(pyridin-2-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C19H22N2
|
1
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| 1 |
Ki = 234.42 nM
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CP0463221
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(2-Chloro-6-methoxy-phenyl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C28H37ClN2O2S
|
1
|
| 1 |
Ki = 237 nM
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CP0517270
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[(2R,5S,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO2
|
1
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| 1 |
Ki = 239.88 nM
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CP0521249
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naphthalen-2-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
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C31H38N2OS
|
1
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| 1 |
Ki = 241 nM
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CP0385601
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2-(diethylamino)ethyl 2,2-diphenylbutanoate
Show/Hide
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C22H29NO2
|
1
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| 1 |
Ki = 243 nM
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CP0468112
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Biphenyl-2-yl-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C33H40N2OS
|
1
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| 1 |
Ki = 250 nM
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CP0128076
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8-Chloro-11-piperazin-1-yl-5H-dibenzo[b,e][1,4]diazepine
Show/Hide
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C17H17ClN4
|
1
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| 1 |
Ki = 250 nM
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CP0505806
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[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]-pyrazin-2-ylmethanone
Show/Hide
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C25H34N4OS
|
1
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| 1 |
Ki = 254 nM
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CP0511061
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[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]-quinolin-8-ylmethanone
Show/Hide
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C30H37N3OS
|
1
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| 1 |
Ki = 256 nM
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CP0530357
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cinnolin-4-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
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C29H36N4OS
|
1
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| 1 |
Ki = 256 nM
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CP0449403
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N,N-dimethyl-2-[3-(1-phenylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H25N
|
1
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| 1 |
Ki = 257.04 nM
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CP0501153
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(2-Fluoro-phenyl)-[4-(4-isopropylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
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C27H35FN2OS
|
1
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| 1 |
Ki = 260 nM
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CP0372485
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N,N-dimethyl-3-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]propan-1-amine
Show/Hide
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C21H26N2
|
1
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| 1 |
Ki = 263.03 nM
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CP0435671
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-2-ylethyl)-pyrrolidinium
Show/Hide
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C27H27F2N4O2+
|
1
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| 1 |
Ki = 268 nM
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CP0441004
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(2-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO2
|
1
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| 1 |
Ki = 275 nM
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CP0875549
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1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-piperidinium iodide
Show/Hide
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C22H30INO
|
1
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| 1 |
Ki = 275.42 nM
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CP0432187
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2-(diethylamino)ethyl 2-(2,6-dimethylphenyl)-2-hydroxy-2-phenylacetate
Show/Hide
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C22H29NO3
|
1
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| 1 |
Ki = 281.5 nM
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CP0437730
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(4-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO2
|
1
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| 1 |
Ki = 283 nM
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CP0378379
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(3-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO2
|
1
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| 1 |
Ki = 312 nM
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CP0305211
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1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
Show/Hide
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C25H32N4O
|
1
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| 1 |
Ki = 320 nM
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CP0842192
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2-(2,2-diphenylacetoxy)-N,N,Ntrimethylethanaminiumbromide
Show/Hide
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C19H24BrNO2
|
1
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| 1 |
Ki = 348 nM
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CP0428746
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-piperidin-1-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C21H35NO2
|
1
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| 1 |
Ki = 352 nM
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CP0410687
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(3R)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
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C24H29NO3
|
1
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| 1 |
Ki = 354.81 nM
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CP0403738
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2-[5-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
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C20H23ClN2
|
1
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| 1 |
Ki = 363.08 nM
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CP0851174
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1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium-4-yl]-1-methylpiperidin-1-ium diiodide
Show/Hide
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C44H58I2N2O2
|
1
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| 1 |
Ki = 363.08 nM
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CP0493835
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2,6-Dimethyl-morpholin-4-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO3
|
1
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| 1 |
Ki = 376 nM
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CP0372523
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2-[1-[2-(2-pyrrolidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
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C22H26N2
|
1
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| 1 |
Ki = 398.11 nM
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CP0473018
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[(2R,5R)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
|
1
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| 1 |
Ki = 407.38 nM
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CP0479629
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[(2R,5S)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
|
1
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| 1 |
Ki = 416.87 nM
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CP0479715
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[(2R,6R)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
|
1
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| 1 |
Ki = 416.87 nM
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CP0410686
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
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| 1 |
Ki = 426.58 nM
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CP0524558
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4-[3-((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-1-oxo-dodecahydro-naphtho[2,3-c]furan-4-yl)-propyl]-piperazine-1-carboxylic acid tert-butyl ester
Show/Hide
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C25H42N2O4
|
1
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| 1 |
Ki = 485 nM
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CP0428329
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8,8-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-8-azonia-bicyclo[3.2.1]octane
Show/Hide
|
C24H30N3O+
|
1
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| 1 |
Ki = 498 nM
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CP0437729
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C26H44N2O2
|
1
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| 1 |
Ki = 520 nM
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CP0425882
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(2-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H24FNO3
|
1
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| 1 |
Ki = 540 nM
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CP0511886
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1-methoxyethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
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C30H36N3O3+
|
1
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| 1 |
Ki = 552 nM
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CP0381564
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2,5-Dimethyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H38N2O2
|
1
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| 1 |
Ki = 570 nM
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CP0441146
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N,N-dimethyl-2-[6-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2
|
1
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| 1 |
Ki = 588.84 nM
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CP0432842
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(4-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C21H36N2O2
|
1
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| 1 |
Ki = 595 nM
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CP0381409
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11-[2-[(4aS,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
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C23H27N5O2
|
1
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| 1 |
Ki = 645.65 nM
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CP0467583
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(3S,3aR,4R,4aS,8aR,9aS)-4-(3-[1,4']Bipiperidinyl-1'-yl-propyl)-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C26H44N2O2
|
1
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| 1 |
Ki = 650 nM
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CP0392151
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N,N-dimethyl-2-[3-(1-pyridin-2-ylbutyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C22H28N2
|
1
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| 1 |
Ki = 676.08 nM
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CP0415329
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
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| 1 |
Ki = 707.95 nM
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CP0673820
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2-(2,2-diphenylacetoxy)-N,N,N-triethylethanaminiumiodide
Show/Hide
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C22H30INO2
|
1
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| 1 |
Ki = 738 nM
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CP0372527
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2-[1-[2-(2-piperidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
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C23H28N2
|
1
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| 1 |
Ki = 851.14 nM
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CP0455599
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1,1-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium
Show/Hide
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C21H26N3O+
|
1
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| 1 |
Ki = 862 nM
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CP0851169
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1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)piperidin-1-ium-4-yl]piperidin-1-ium dichloride
Show/Hide
|
C42H54Cl2N2O2
|
1
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| 1 |
Ki = 870.96 nM
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CP0473022
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[(2R,5S)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C21H28INO2
|
1
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| 1 |
Ki = 870.96 nM
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CP0511888
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1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-benzyl-pyrrolidinium
Show/Hide
|
C27H30N3O+
|
1
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| 1 |
Ki = 884 nM
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CP0406408
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N,N-dimethyl-2-[5-methylsulfanyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2S
|
1
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| 1 |
Ki = 912.01 nM
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CP0511060
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furan-2-yl-[4-[4-[(4-propan-2-ylsulfanylphenyl)methyl]piperidin-1-yl]piperidin-1-yl]methanone
Show/Hide
|
C25H34N2O2S
|
1
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| 1 |
Ki = 923 nM
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CP0029624
|
4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one
Show/Hide
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C20H31NO
|
1
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| 1 |
Ki = 980 nM
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CP0381581
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11-[2-[(4aR,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C23H27N5O2
|
1
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| 1 |
Ki = 1000 nM
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CP0425076
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-3-ylethyl)-pyrrolidinium
Show/Hide
|
C27H27F2N4O2+
|
1
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| 1 |
Ki = 1014 nM
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CP0220610
|
Bietamiverine
Show/Hide
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C19H30N2O2
|
1
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| 1 |
Ki = 1020 nM
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CP0403766
|
2-[5-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O
|
1
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| 1 |
Ki = 1023.29 nM
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CP0372477
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2-[6-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O
|
1
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| 1 |
Ki = 1071.52 nM
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CP0139207
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
|
C23H24N2O4
|
1
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| 1 |
Ki = 1096.48 nM
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CP0425606
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-(4-methoxy-phenyl)-ethyl ester; oxalic acid
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
Ki = 1100 nM
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CP0532167
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1-cyanomethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C29H31N4O2+
|
1
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| 1 |
Ki = 1152 nM
|
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CP0418483
|
2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H25NO3
|
1
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| 1 |
Ki = 1170 nM
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CP0139209
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N,N-dimethyl-2-[3-[(1R)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 1230.27 nM
|
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CP0386736
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 1230.27 nM
|
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CP0156301
|
2-(diethylamino)ethyl 2-(4-chlorophenyl)sulfanylbenzoate
Show/Hide
|
C19H22ClNO2S
|
1
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| 1 |
Ki = 1340 nM
|
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CP0487384
|
[(2R,5R)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C21H28INO2
|
1
|
| 1 |
Ki = 1348.96 nM
|
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CP0473017
|
trimethyl-[[(2R,5S)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 1380.38 nM
|
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|
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CP0404155
|
4-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]morpholine
Show/Hide
|
C22H26N2O
|
1
|
| 1 |
Ki = 1445.44 nM
|
|
|
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CP0542858
|
2-[4-[[1-[1-(naphthalene-1-carbonyl)piperidin-4-yl]piperidin-4-yl]methyl]phenyl]sulfanylacetic acid
Show/Hide
|
C30H34N2O3S
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
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CP0386734
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 1548.82 nM
|
|
|
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CP0425075
|
1,1-dimethyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-piperidinium
Show/Hide
|
C22H28N3O+
|
1
|
| 1 |
Ki = 1810 nM
|
|
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CP0437455
|
[(2R,5S,6S)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 1905.46 nM
|
|
|
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CP0492466
|
N,N-dimethyl-2-[5-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 1949.84 nM
|
|
|
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CP0379030
|
1-benzyl-1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium
Show/Hide
|
C27H30N3O+
|
1
|
| 1 |
Ki = 2010 nM
|
|
|
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CP0425883
|
3-(4-methoxyphenyl)propyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 2030 nM
|
|
|
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CP0487380
|
trimethyl-[[(2R,5S)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C26H30INO2
|
1
|
| 1 |
Ki = 2137.96 nM
|
|
|
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CP0026924
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C24H29N3O3
|
1
|
| 1 |
Ki = 2200 nM
|
|
|
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CP0487382
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[(2R,5R)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C21H28INO2
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1
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| 1 |
Ki = 2238.72 nM
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CP0516426
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[(2R,5R,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 2238.72 nM
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CP0862114
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1,4-Bis-(4-hydroxy-4,4-diphenyl-butyl)-1-methyl-piperazin-1-ium iodide
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C37H45IN2O2
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1
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| 1 |
Ki = 2290.87 nM
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CP0386732
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C24H27NO4
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1
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| 1 |
Ki = 2290.87 nM
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CP0851168
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DIPHENIDOL HYDROCHLORIDE
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C21H28ClNO
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1
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| 1 |
Ki = 2818.38 nM
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CP0491695
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[(2R,6S)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO3S
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1
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| 1 |
Ki = 3019.95 nM
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CP0516423
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[(2R,5R)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO3S
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1
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| 1 |
Ki = 3019.95 nM
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CP0479627
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trimethyl-[[(2R,5S)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 3235.94 nM
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CP0472769
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trimethyl-[[(2R,6S)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2S
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1
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| 1 |
Ki = 3388.44 nM
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CP0862120
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1-(4-hydroxy-4,4-diphenylbutyl)-4-(1-methylpiperidin-1-ium-4-yl)piperidin-1-ium dichloride
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C27H40Cl2N2O
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1
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| 1 |
Ki = 3981.07 nM
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CP0913741
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4-(1,1-dimethylpiperidin-1-ium-4-yl)-1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium diiodide
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C29H44I2N2O
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1
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| 1 |
Ki = 4365.16 nM
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CP0479714
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trimethyl-[[(2R,5R)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C26H30INO2
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1
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| 1 |
Ki = 4365.16 nM
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CP0404384
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2-(dimethylamino)ethyl 3-(pyridin-2-ylmethyl)-1H-indene-2-carboxylate
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C20H22N2O2
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1
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| 1 |
Ki = 4897.79 nM
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CP0399353
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N,N-dimethyl-2-[3-(pyridin-3-ylmethyl)-1H-inden-2-yl]ethanamine
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C19H22N2
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1
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| 1 |
Ki = 5370.32 nM
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CP0479654
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trimethyl-[[(2R,6R)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 5370.32 nM
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CP0862110
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N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N3-dimethylpropane-1,3-diaminium chloride
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C37H48Cl2N2O2
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1
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| 1 |
Ki = 5495.41 nM
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CP0424269
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2-(dimethylamino)ethyl 3-(pyridin-3-ylmethyl)-1H-indene-2-carboxylate
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C20H22N2O2
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1
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| 1 |
Ki = 6025.6 nM
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CP0505786
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N,N-dimethyl-2-[3-(pyridin-4-ylmethyl)-1H-inden-2-yl]ethanamine
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C19H22N2
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1
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| 1 |
Ki = 6760.83 nM
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CP0851172
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4-(4-hydroxy-4,4-diphenylbutyl)piperazine-1,4-diium dichloride
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C20H28Cl2N2O
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1
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| 1 |
Ki = 7244.36 nM
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CP0479708
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[(2R,6S)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO4S
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1
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| 1 |
Ki = 7413.1 nM
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CP0851569
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1-(3,5-dichlorophenyl)piperazine
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C10H12Cl2N2
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1
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| 1 |
Ki = 7943.28 nM
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CP0479711
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trimethyl-[[(2R,6S)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 8709.64 nM
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CP0479717
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trimethyl-[[(2R,5R)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C14H22INO2
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1
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| 1 |
Ki = 8709.64 nM
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CP0387007
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[(2R,5S)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO4S
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1
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| 1 |
Ki > 10000 nM
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CP0421082
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trimethyl-[[(2R,5S)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C14H22INO2
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1
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| 1 |
Ki > 10000 nM
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CP0473016
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[(2R,5S)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C21H28INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479628
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trimethyl-[[(2R,5R)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0862121
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N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N3,N3-tetramethylpropane-1,3-diaminium iodide
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C39H52I2N2O2
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1
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| 1 |
Ki = 12022.64 nM
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CP0404254
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N-[2-(dimethylamino)ethyl]-3-(pyridin-2-ylmethyl)-1H-indene-2-carboxamide
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C20H23N3O
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1
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| 1 |
Ki = 14791.08 nM
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CP0069240
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4-(piperazin-1-yl)-1H-indole
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C12H15N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0184743
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4-methyl-2-piperazin-1-ylquinoline
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C14H17N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0364794
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1-(2,3-dichlorophenyl)piperazine
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C10H12Cl2N2
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1
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| 1 |
Ki > 19952.62 nM
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CP0875550
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4-(4-Hydroxy-4,4-diphenyl-butyl)-1,1-dimethyl-piperazin-1-ium iodide
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C22H31IN2O
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1
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| 1 |
Ki = 23442.29 nM
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CP0851173
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1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-4-phenyl-piperazin-1-ium iodide
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C27H33IN2O
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1
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| 1 |
Ki = 25703.96 nM
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CP0851171
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4-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperazine-1,4-diium dichloride
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C21H30Cl2N2O
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1
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| 1 |
Ki = 35481.34 nM
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CP0416829
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N-[2-(dimethylamino)ethyl]-3-(pyridin-3-ylmethyl)-1H-indene-2-carboxamide
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C20H23N3O
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1
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| 1 |
Ki = 39810.72 nM
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CP0862112
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N1,N2-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N2,N2-tetramethylethane-1,2-diaminium iodide
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C38H50I2N2O2
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1
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| 1 |
Ki = 47863.01 nM
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CP0375776
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N-[2-(dimethylamino)ethyl]-3-(pyridin-4-ylmethyl)-1H-indene-2-carboxamide
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C20H23N3O
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1
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| 1 |
Ki = 93325.43 nM
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CP0418482
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2-naphthalen-1-ylethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C25H25NO2
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1
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| 1 |
Ki > 100000 nM
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CP0425884
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2-(3,4-dimethoxyphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C23H27NO4
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1
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| 1 |
Ki > 100000 nM
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CP0471231
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2-(3,4-dimethoxyphenyl)ethyl 4-(3-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C23H26FNO4
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1
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| 1 |
Ki > 100000 nM
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CP0484746
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C24H27NO3
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1
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| 1 |
Ki > 100000 nM
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CP0406685
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-piperazin-1-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
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C20H34N2O2
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1
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| 1 |
Ki > 42 nM
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CP0392943
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
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C21H35NO3
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1
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| 1 |
Ki > 280 nM
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CP0392927
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-((S)-3-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
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C21H36N2O2
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1
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| 1 |
Ki > 500 nM
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CP0441685
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-((R)-3-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
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C21H36N2O2
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1
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| 1 |
Ki > 500 nM
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CP0490487
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,5-Dimethyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
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C22H38N2O2
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1
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| 1 |
Ki > 500 nM
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