| Compound ID |
Compound Name |
Compound Formula |
|
CP0384614
|
4-cyclopentyl-2-((4-(piperidin-1-ylmethyl)phenoxy)methyl)morpholine
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|
C22H34N2O2
|
2
|
| 1 |
Kd = 1.549 nM
|
|
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| 2 |
Ki = 10 nM
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|
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CP0441522
|
4-cyclopentyl-2-((4-(pyrrolidin-1-ylmethyl)phenoxy)methyl)morpholine
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|
C21H32N2O2
|
2
|
| 1 |
Kd = 1.585 nM
|
|
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| 2 |
Ki = 9.8 nM
|
|
|
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CP0446007
|
(S)-4-cyclopentyl-2-((4-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C21H32N2O3
|
2
|
| 1 |
Kd = 2.138 nM
|
|
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| 2 |
Ki = 9.7 nM
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CP0106703
|
1-((2R,4S)-2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-4-(4-fluorophenoxy)pyrrolidin-1-yl)ethanone
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|
C22H30FN3O3
|
1
|
| 1 |
Kd = 2.291 nM
|
|
|
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CP0325312
|
((2R,4S)-4-(3-chlorophenoxy)pyrrolidin-2-yl)(4-cyclobutyl-1,4-diazepan-1-yl)methanone
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|
C20H28ClN3O2
|
1
|
| 1 |
Kd = 2.57 nM
|
|
|
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CP0158344
|
4-((3S,5R)-5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)pyrrolidin-3-yloxy)benzonitrile
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|
C22H30N4O2
|
1
|
| 1 |
Kd = 3.09 nM
|
|
|
|
CP0046809
|
(4-cyclobutyl-1,4-diazepan-1-yl)(6-(4-fluorophenoxy)pyridin-3-yl)methanone
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|
C21H24FN3O2
|
1
|
| 1 |
Kd = 3.548 nM
|
|
|
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CP0400799
|
(4-cyclobutyl-1,4-diazepan-1-yl)(6-phenoxypyridin-3-yl)methanone
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|
C21H25N3O2
|
1
|
| 1 |
Kd = 3.715 nM
|
|
|
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CP0246919
|
(6-(4-chlorophenoxy)pyridin-3-yl)(4-cyclobutyl-1,4-diazepan-1-yl)methanone
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|
C21H24ClN3O2
|
1
|
| 1 |
Kd = 3.981 nM
|
|
|
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CP0265410
|
(4-cyclobutyl-1,4-diazepan-1-yl)(6-(3-fluorophenoxy)pyridin-3-yl)methanone
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|
C21H24FN3O2
|
1
|
| 1 |
Kd = 4.169 nM
|
|
|
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CP0095277
|
4-(3-(4-(piperidin-1-yl)but-1-ynyl)benzyl)morpholine
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|
C20H28N2O
|
2
|
| 1 |
Kd = 4.677 nM
|
|
|
| 2 |
Ki = 7.079 nM
|
|
|
|
CP0441524
|
4-cyclopentyl-2-((4-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C21H32N2O3
|
2
|
| 1 |
Kd = 4.786 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
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CP0228017
|
((2R,4S)-4-(4-chlorophenoxy)pyrrolidin-2-yl)(4-cyclobutyl-1,4-diazepan-1-yl)methanone
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|
C20H28ClN3O2
|
1
|
| 1 |
Kd = 5.012 nM
|
|
|
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CP0333672
|
(6-(3-chlorophenoxy)pyridin-3-yl)(4-cyclobutyl-1,4-diazepan-1-yl)methanone
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|
C21H24ClN3O2
|
1
|
| 1 |
Kd = 5.012 nM
|
|
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CP0115802
|
1-((2R,4S)-2-(4-cyclobutyl-1,4-diazepane-1-carbonyl)-4-(3-fluorophenoxy)pyrrolidin-1-yl)ethanone
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|
C22H30FN3O3
|
1
|
| 1 |
Kd = 6.026 nM
|
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|
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CP0158337
|
(4-cyclopentyl-1,4-diazepan-1-yl)((2R,4S)-4-(4-fluorophenoxy)pyrrolidin-2-yl)methanone
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|
C21H30FN3O2
|
1
|
| 1 |
Kd = 6.166 nM
|
|
|
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CP0374240
|
(4-cyclobutyl-1,4-diazepan-1-yl)(6-(3,4-dichlorophenoxy)pyridin-3-yl)methanone
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|
C21H23Cl2N3O2
|
1
|
| 1 |
Kd = 6.918 nM
|
|
|
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CP0158336
|
(4-cyclobutyl-1,4-diazepan-1-yl)((2R,4S)-4-(3-fluorophenoxy)pyrrolidin-2-yl)methanone
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|
C20H28FN3O2
|
1
|
| 1 |
Kd = 8.128 nM
|
|
|
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CP0125374
|
3-(5-(4-cyclobutyl-1,4-diazepane-1-carbonyl)pyridin-2-yloxy)benzonitrile
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|
C22H24N4O2
|
1
|
| 1 |
Kd = 9.55 nM
|
|
|
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CP0506136
|
(6-(3-chlorophenoxy)pyridin-3-yl)(4-cyclopropyl-1,4-diazepan-1-yl)methanone
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|
C20H22ClN3O2
|
1
|
| 1 |
Kd = 11.48 nM
|
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CP0096441
|
(4-cyclobutyl-1,4-diazepan-1-yl)((2R,4S)-4-(4-fluorophenoxy)pyrrolidin-2-yl)methanone
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|
C20H28FN3O2
|
1
|
| 1 |
Kd = 11.75 nM
|
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|
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CP0095968
|
4-((3S,5R)-5-(4-cyclobutyl-1,4-diazepane-1-carbonyl)pyrrolidin-3-yloxy)benzonitrile
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|
C21H28N4O2
|
1
|
| 1 |
Kd = 12.59 nM
|
|
|
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CP0446004
|
4-cyclobutyl-2-((4-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C20H30N2O3
|
2
|
| 1 |
Kd = 19.05 nM
|
|
|
| 2 |
Ki = 75 nM
|
|
|
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CP0037773
|
(4-cyclobutyl-1,4-diazepan-1-yl)(5-(4-fluorophenoxy)pyridin-2-yl)methanone
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|
C21H24FN3O2
|
1
|
| 1 |
Kd = 26.3 nM
|
|
|
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CP0403088
|
(R)-4-cyclopentyl-2-((4-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C21H32N2O3
|
2
|
| 1 |
Kd = 43.65 nM
|
|
|
| 2 |
Ki = 121 nM
|
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|
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CP0462298
|
4-cyclobutyl-2-((3-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C20H30N2O3
|
2
|
| 1 |
Kd = 79.43 nM
|
|
|
| 2 |
Ki = 277 nM
|
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|
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CP0399177
|
4-isopropyl-2-((3-(morpholinomethyl)phenoxy)methyl)morpholine
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|
C19H30N2O3
|
2
|
| 1 |
Kd = 251.19 nM
|
|
|
| 2 |
Ki = 562 nM
|
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|
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CP0056575
|
1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piperidine
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|
C20H32N2O
|
1
|
| 1 |
Ki = 0.4571 nM
|
|
|
|
CP0399176
|
4-isopropyl-2-((4-(morpholinomethyl)phenoxy)methyl)morpholine
Show/Hide
|
C19H30N2O3
|
1
|
| 1 |
Ki = 92 nM
|
|
|
