| Compound ID |
Compound Name |
Compound Formula |
|
CP0489436
|
5-[3-(4-fluorophenyl)-4-oxo-7-spiro[1,3-dihydroindene-2,5'-4H-1,2-oxazole]-3'-ylquinazolin-2-yl]pentanoic acid
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|
C30H26FN3O4
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0388964
|
5-[7-(5-butyl-5-phenyl-4H-1,2-oxazol-3-yl)-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C32H32FN3O4
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0461325
|
5-[7-(5-ethyl-5-phenyl-4H-1,2-oxazol-3-yl)-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O4
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0489432
|
5-[3-(4-fluorophenyl)-4-oxo-7-(5-phenyl-5-propyl-4H-1,2-oxazol-3-yl)quinazolin-2-yl]pentanoic acid
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|
C31H30FN3O4
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0073144
|
5-[7-[(5S)-5-(1,3-benzoxazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H25FN4O5
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0473199
|
5-[3-(4-fluorophenyl)-7-[5-(methoxymethyl)-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O5
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0481766
|
5-[7-[(5R)-5-(4-chlorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H25ClFN3O4
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0388965
|
5-[7-[(5S)-5-(1,3-benzothiazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H25FN4O4S
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0443724
|
5-[3-(4-fluorophenyl)-7-[(5S)-5-[(R)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O5
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0461374
|
5-[3-(4-fluorophenyl)-7-[5-(hydroxymethyl)-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H26FN3O5
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0478950
|
5-[7-[(5S)-5-(4-chlorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H25ClFN3O4
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0443723
|
5-[7-[(5S)-5-(3-cyanophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H25FN4O4
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0481765
|
5-[7-[(5S)-5-(3,5-difluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H24F3N3O4
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0395524
|
5-[3-(4-fluorophenyl)-7-[(5S)-5-methyl-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H26FN3O4
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0443728
|
5-[3-(4-fluorophenyl)-7-[(5S)-5-[(S)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O5
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0389632
|
5-[3-(4-fluorophenyl)-7-[(5S)-5-(4-fluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H25F2N3O4
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0388963
|
5-[3-(4-fluorophenyl)-7-(5-methyl-5-phenyl-4H-1,2-oxazol-3-yl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H26FN3O4
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
|
CP0389633
|
5-[7-[(5R)-5-(1,3-benzothiazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H25FN4O4S
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0461376
|
5-[3-(4-fluorophenyl)-7-[(5R)-5-(4-fluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H25F2N3O4
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0432909
|
5-[7-[(5S)-5-benzyl-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O4
|
1
|
| 1 |
Ki = 7.4 nM
|
|
|
|
CP0461375
|
5-[7-[(5R)-5-benzyl-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C30H28FN3O4
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0568644
|
5-[7-[(5R)-5-(3,5-difluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C29H24F3N3O4
|
1
|
| 1 |
Ki = 10.5 nM
|
|
|
|
CP0395522
|
5-[7-(5,5-diphenyl-4H-1,2-oxazol-3-yl)-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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|
C34H28FN3O4
|
1
|
| 1 |
Ki = 13.7 nM
|
|
|
|
CP0432908
|
5-[3-(4-fluorophenyl)-7-[(5R)-5-[(R)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O5
|
1
|
| 1 |
Ki = 18.3 nM
|
|
|
|
CP0528920
|
5-[7-[(5R)-5-(1,3-benzoxazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H25FN4O5
|
1
|
| 1 |
Ki = 19.6 nM
|
|
|
|
CP0478951
|
5-[7-[(5R)-5-(3-cyanophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H25FN4O4
|
1
|
| 1 |
Ki = 22.3 nM
|
|
|
|
CP0473200
|
5-[3-(4-fluorophenyl)-7-[(5R)-5-methyl-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H26FN3O4
|
1
|
| 1 |
Ki = 24.9 nM
|
|
|
|
CP0443725
|
5-[3-(4-fluorophenyl)-7-[(5R)-5-[(S)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O5
|
1
|
| 1 |
Ki = 41.7 nM
|
|
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