Compound ID |
Compound Name |
Compound Formula |
CP0476680
|
1,10-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-ylsulfanyl]decane
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|
C26H40N6S4
|
1
|
1 |
EC50 = 0.6 nM
|
|
|
CP0383357
|
1,12-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-ylsulfanyl]dodecane
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|
C28H44N6S4
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0460884
|
1,12-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]dodecane
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|
C28H44N6O2S2
|
1
|
1 |
EC50 = 1.4 nM
|
|
|
CP0449083
|
1,11-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-ylsulfanyl]undecane
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|
C27H42N6S4
|
1
|
1 |
EC50 = 4.7 nM
|
|
|
CP0376259
|
1-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]-2-[2-(2-{2-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]ethoxy}ethoxy)ethoxy]ethane
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|
C24H36N6O5S2
|
1
|
1 |
EC50 = 5.2 nM
|
|
|
CP0635477
|
(2-Carbamoyloxy-ethyl)-trimethyl-ammonium chloride
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|
C6H15ClN2O2
|
1
|
1 |
EC50 = 290 nM
|
|
|
CP0471023
|
1,10-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]decane
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|
C26H40N6O2S2
|
1
|
1 |
EC50 = 1100 nM
|
|
|
CP0460747
|
1,2-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]ethane
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|
C18H24N6O2S2
|
1
|
1 |
EC50 = 3900 nM
|
|
|
CP0399528
|
1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]nonane
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|
C25H38N6O2S2
|
1
|
1 |
EC50 = 20000 nM
|
|
|
CP0376490
|
1,8-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]octane
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|
C24H36N6O2S2
|
1
|
1 |
EC50 > 100000 nM
|
|
|
CP0401666
|
1,6-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]hexane
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|
C22H32N6O2S2
|
1
|
1 |
EC50 > 100000 nM
|
|
|
CP0534589
|
1,7-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]heptane
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|
C23H34N6O2S2
|
1
|
1 |
EC50 > 100000 nM
|
|
|