| Compound ID |
Compound Name |
Compound Formula |
|
CP0460085
|
2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]acetamide
Show/Hide
|
C31H34N6O5
|
1
|
| 1 |
Ki = 0.1072 nM
|
|
|
|
CP0160764
|
(R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridin-2-yl)-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(3-(methylamino)phenyl)urea
Show/Hide
|
C28H30N6O3
|
1
|
| 1 |
Ki = 0.138 nM
|
|
|
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CP0377905
|
2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]acetamide
Show/Hide
|
C30H34N6O5
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
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CP0486206
|
5-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]furan-2-carboxylic acid
Show/Hide
|
C33H36N4O6
|
1
|
| 1 |
Ki = 0.2455 nM
|
|
|
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CP0434221
|
2-[3-[[2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]acetic acid
Show/Hide
|
C31H36N4O5
|
1
|
| 1 |
Ki = 0.2818 nM
|
|
|
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CP0445844
|
2-[6-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indol-1-yl]acetic acid
Show/Hide
|
C32H37N5O5
|
1
|
| 1 |
Ki = 0.2951 nM
|
|
|
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CP0434220
|
2-[3-[[2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]sulfanylacetic acid
Show/Hide
|
C31H36N4O5S
|
1
|
| 1 |
Ki = 0.3311 nM
|
|
|
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CP0445843
|
3-[3-[[2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]propanoic acid
Show/Hide
|
C32H38N4O5
|
1
|
| 1 |
Ki = 0.3388 nM
|
|
|
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CP0463035
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
|
C32H35N5O6
|
1
|
| 1 |
Ki = 0.3631 nM
|
|
|
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CP0877927
|
2-(1-cycloheptyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-(5-oxo-2,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl)-acetamide
Show/Hide
|
C31H36N6O6
|
1
|
| 1 |
Ki = 0.4266 nM
|
|
|
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CP0445812
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]sulfanylacetic acid
Show/Hide
|
C30H36N4O5S
|
1
|
| 1 |
Ki = 0.6457 nM
|
|
|
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CP0377907
|
4-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]-1,3-thiazole-2-carboxylic acid
Show/Hide
|
C32H35N5O5S
|
1
|
| 1 |
Ki = 0.6607 nM
|
|
|
|
CP0377897
|
2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-(2H-tetrazol-5-ylmethylsulfanyl)phenyl]acetamide
Show/Hide
|
C30H36N8O3S
|
1
|
| 1 |
Ki = 0.7079 nM
|
|
|
|
CP0445846
|
2-[5-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indol-1-yl]acetic acid
Show/Hide
|
C32H37N5O5
|
1
|
| 1 |
Ki = 0.7762 nM
|
|
|
|
CP0463044
|
3-[[2-[5-cyclohexyl-1-(2-cyclohexyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C31H36N4O5
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0435649
|
2-[6-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indazol-1-yl]acetic acid
Show/Hide
|
C31H36N6O5
|
1
|
| 1 |
Ki = 0.8318 nM
|
|
|
|
CP0877928
|
(3-(2-(1-cycloheptyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-acetylamino)-phenylsulfanyl)-acetic acid
Show/Hide
|
C31H38N4O6S
|
1
|
| 1 |
Ki = 0.8913 nM
|
|
|
|
CP0236227
|
2-[2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]pyrrol-1-yl]acetic acid
Show/Hide
|
C34H39N5O5
|
1
|
| 1 |
Ki = 0.912 nM
|
|
|
|
CP0374437
|
3-[[2-[5-cyclohexyl-1-(2-cyclopentyl-2-oxoethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C30H34N4O5
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0377904
|
2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-(2H-tetrazol-5-yl)phenyl]acetamide
Show/Hide
|
C29H34N8O3
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0460084
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]-N-methylanilino]acetic acid
Show/Hide
|
C31H39N5O5
|
1
|
| 1 |
Ki = 1.072 nM
|
|
|
|
CP0435583
|
3-[[2-[5-cyclohexyl-1-[2-(2-methylcyclopentyl)-2-oxoethyl]-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C31H36N4O5
|
1
|
| 1 |
Ki = 1.202 nM
|
|
|
|
CP0873275
|
2-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-(5-oxo-2,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl)-acetamide
Show/Hide
|
C30H34N6O6
|
1
|
| 1 |
Ki = 1.202 nM
|
|
|
|
CP0463042
|
3-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]benzoic acid
Show/Hide
|
C35H38N4O5
|
1
|
| 1 |
Ki = 1.585 nM
|
|
|
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CP0475203
|
3-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]propanoic acid
Show/Hide
|
C31H38N4O5
|
1
|
| 1 |
Ki = 1.862 nM
|
|
|
|
CP0374445
|
2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-[methyl(2H-tetrazol-5-yl)amino]phenyl]acetamide
Show/Hide
|
C30H37N9O3
|
1
|
| 1 |
Ki = 1.95 nM
|
|
|
|
CP0435604
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]acetic acid
Show/Hide
|
C30H36N4O5
|
1
|
| 1 |
Ki = 2.138 nM
|
|
|
|
CP0374448
|
2-[4-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indazol-1-yl]acetic acid;2,2,2-trifluoroacetic acid
Show/Hide
|
C31H36N6O5
|
1
|
| 1 |
Ki = 2.754 nM
|
|
|
|
CP0897678
|
(3-(2-(1-cycloheptyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-acetylamino)-phenyl)-acetic acid
Show/Hide
|
C31H38N4O6
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
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CP0374443
|
3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]-N-methylsulfonylbenzamide
Show/Hide
|
C30H37N5O6S
|
1
|
| 1 |
Ki = 3.89 nM
|
|
|
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CP0437077
|
2-[4-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]imidazol-1-yl]acetic acid;hydrochloride
Show/Hide
|
C33H38N6O5
|
1
|
| 1 |
Ki = 4.074 nM
|
|
|
|
CP0377903
|
2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenyl]sulfonylacetic acid
Show/Hide
|
C30H36N4O7S
|
1
|
| 1 |
Ki = 4.266 nM
|
|
|
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CP0939854
|
2-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-(methyl-(2H-tetrazol-5-yl)-amino)-phenyl)-acetamide
Show/Hide
|
C30H37N9O4
|
1
|
| 1 |
Ki = 4.266 nM
|
|
|
|
CP0377906
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2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]-N-[3-(2H-tetrazol-5-ylmethyl)phenyl]acetamide
Show/Hide
|
C30H36N8O3
|
1
|
| 1 |
Ki = 4.677 nM
|
|
|
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CP0435584
|
3-[[2-[5-cycloheptyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C30H36N4O5
|
1
|
| 1 |
Ki = 4.786 nM
|
|
|
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CP0077676
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3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C29H34N4O5
|
1
|
| 1 |
Ki = 5.129 nM
|
|
|
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CP0374442
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2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]phenoxy]acetic acid
Show/Hide
|
C30H36N4O6
|
1
|
| 1 |
Ki = 5.495 nM
|
|
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CP0885418
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methoxy-phenyl)-acetamide
Show/Hide
|
C29H36N4O4
|
1
|
| 1 |
Ki = 5.495 nM
|
|
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CP0437076
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3-[[2-[1-[2-(1-adamantyl)-2-oxoethyl]-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C35H40N4O5
|
1
|
| 1 |
Ki = 5.623 nM
|
|
|
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CP0384959
|
2-[4-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indol-1-yl]acetic acid
Show/Hide
|
C32H37N5O5
|
1
|
| 1 |
Ki = 6.026 nM
|
|
|
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CP0911236
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(dimethylamino)-phenyl)-acetamide
Show/Hide
|
C30H39N5O3
|
1
|
| 1 |
Ki = 6.026 nM
|
|
|
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CP0918905
|
2-((S)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide
Show/Hide
|
C30H38N4O3
|
1
|
| 1 |
Ki = 6.026 nM
|
|
|
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CP0512402
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2-[3-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]anilino]acetic acid;hydrochloride
Show/Hide
|
C30H37N5O5
|
1
|
| 1 |
Ki = 6.166 nM
|
|
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CP0897677
|
3-(3-(2-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-acetylamino)-phenyl)-propionic acid
Show/Hide
|
C31H38N4O6
|
1
|
| 1 |
Ki = 6.31 nM
|
|
|
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CP0384935
|
3-[[2-[5-cyclohexyl-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C32H32N4O5
|
1
|
| 1 |
Ki = 7.586 nM
|
|
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CP0893510
|
2-(1-cycloheptyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-mtolyl-acetamide
Show/Hide
|
C30H38N4O4
|
1
|
| 1 |
Ki = 7.586 nM
|
|
|
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CP0036767
|
S-L-365,260
Show/Hide
|
C24H22N4O2
|
1
|
| 1 |
Ki = 7.762 nM
|
|
|
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CP0918908
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methylamino-phenyl)-acetamide
Show/Hide
|
C29H37N5O3
|
1
|
| 1 |
Ki = 7.943 nM
|
|
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CP0844737
|
2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-m-tolyl-acetamide
Show/Hide
|
C29H36N4O3
|
1
|
| 1 |
Ki = 8.913 nM
|
|
|
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CP0911239
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(1H-imidazol-1-yl)-phenyl)-acetamide
Show/Hide
|
C31H36N6O3
|
1
|
| 1 |
Ki = 9.12 nM
|
|
|
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CP0460088
|
2-[5-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]indazol-1-yl]acetic acid
Show/Hide
|
C31H36N6O5
|
1
|
| 1 |
Ki = 9.333 nM
|
|
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CP0886040
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2-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-(2-methyl-thiazol-4-yl)-phenyl)-acetamide
Show/Hide
|
C32H37N5O4S
|
1
|
| 1 |
Ki = 9.55 nM
|
|
|
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CP0914890
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2-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-methylamino-phenyl)-acetamide
Show/Hide
|
C29H37N5O4
|
1
|
| 1 |
Ki = 9.55 nM
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|
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CP0881710
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-hydroxy-phenyl)-acetamide
Show/Hide
|
C28H34N4O4
|
1
|
| 1 |
Ki = 13.18 nM
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CP0915570
|
2-((R)-5-cyclohexyl-2,3-dihydro-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1H-benzo[e][1,4]diazepin-3-yl)-N-(3-(methylamino)phenyl)-acetamide
Show/Hide
|
C30H38N4O3
|
1
|
| 1 |
Ki = 13.18 nM
|
|
|
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CP0911234
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-hydroxymethyl-phenyl)-acetamide
Show/Hide
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C29H36N4O4
|
1
|
| 1 |
Ki = 15.14 nM
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|
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CP0911235
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-pyrrolidin-1-yl-phenyl)-acetamide
Show/Hide
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C32H41N5O3
|
1
|
| 1 |
Ki = 15.85 nM
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|
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CP0437070
|
3-[[2-[5-cyclohexyl-2-oxo-1-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C29H33N5O5
|
1
|
| 1 |
Ki = 16.22 nM
|
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CP0862309
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-morpholin-4-yl-phenyl)-acetamide
Show/Hide
|
C32H41N5O4
|
1
|
| 1 |
Ki = 16.6 nM
|
|
|
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CP0445845
|
2-[6-[[2-[5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzimidazol-1-yl]acetic acid;hydrochloride
Show/Hide
|
C31H36N6O5
|
1
|
| 1 |
Ki = 16.98 nM
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CP0044497
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3-[[5-(1-adamantyloxymethyl)-2-cyclohexyl-1H-imidazole-4-carbonyl]amino]benzoic acid
Show/Hide
|
C28H35N3O4
|
1
|
| 1 |
Ki = 19.5 nM
|
|
|
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CP0486210
|
3-[[2-[5-cyclohexyl-1-(3-methylbutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
Show/Hide
|
C28H34N4O4
|
1
|
| 1 |
Ki = 20.42 nM
|
|
|
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CP0920847
|
4-(1-cyclohexyl-5-(3,3-dimethyl-2-oxo-butyl)-2,4-dioxo-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-(3-(5-oxo-2,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl)-butyramide
Show/Hide
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C32H38N6O6
|
1
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| 1 |
Ki = 20.89 nM
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|
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CP0886067
|
2-(1-cycloheptyl-2,4-dioxo-5-(2-oxo-2-pyrrolidin-1-yl-ethyl)-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-m-tolyl-acetamide
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C30H37N5O4
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1
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| 1 |
Ki = 23.44 nM
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CP0399462
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3-[[2-[5-(1-adamantyl)-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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C33H38N4O5
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1
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| 1 |
Ki = 23.99 nM
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CP0435585
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3-[[2-[5-cyclopentyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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C28H32N4O5
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1
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| 1 |
Ki = 23.99 nM
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CP0926875
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N-(3-amino-phenyl)-2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxobutyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetamide
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C28H35N5O3
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1
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| 1 |
Ki = 26.92 nM
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CP0918904
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(methyl-(2-methylaminoethyl)-amino)-phenyl)-acetamide
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C32H44N6O3
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1
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| 1 |
Ki = 29.51 nM
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CP0918907
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2-(5-cyclohexyl-1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-(2-ethoxy-ethylamino)-phenyl)-acetamide
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C32H43N5O4
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1
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| 1 |
Ki = 44.67 nM
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CP0034742
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(R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-amide: 0.1C4H10O
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C25H20N4O2
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1
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| 1 |
Ki = 51.29 nM
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CP0853811
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2-(1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methylamino-phenyl)-acetamide
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C29H31N5O3
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1
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| 1 |
Ki = 74.13 nM
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CP0435586
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3-[[2-[1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-propan-2-yl-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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C26H30N4O5
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1
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| 1 |
Ki = 89.13 nM
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CP0915572
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2-(1-(3,3-dimethyl-2-oxo-butyl)-2-oxo-5-pyridin-2-yl-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-N-(3-methylamino-phenyl)-acetamide
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C28H30N6O3
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1
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| 1 |
Ki = 194.98 nM
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CP0917618
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N-(3-methylamino-phenyl)-2-(2-oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetamide
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C31H28N6O3
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1
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| 1 |
Ki = 288.4 nM
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CP0443146
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3-[[2-[5-cyclohexyl-2-oxo-1-(2-oxopropyl)-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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C26H28N4O5
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1
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| 1 |
Ki = 331.13 nM
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CP0893511
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3-(2-(2,4-dioxo-1-(2-oxo-2-pyrrolidin-1-yl-ethyl)-5-phenyl-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-acetylamino)-benzoic acid
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C29H27N5O6
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1
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| 1 |
Ki = 380.19 nM
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CP0162124
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3-[[2-[5-cyclohexyl-1-(2-ethoxyethyl)-2-oxo-1,3,4-benzotriazepin-3-yl]acetyl]amino]benzoic acid
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C27H32N4O5
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1
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| 1 |
Ki = 489.78 nM
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CP0914889
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2-(2,4-dioxo-1-(2-oxo-2-pyrrolidin-1-yl-ethyl)-5-phenyl-1,2,4,5-tetrahydro-1,3,5-benzotriazepin-3-yl)-N-phenylacetamide
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C28H27N5O4
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1
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| 1 |
Ki = 1000 nM
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CP0384937
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3-[[2-(5-cyclohexyl-1-methyl-2-oxo-1,3,4-benzotriazepin-3-yl)acetyl]amino]benzoic acid
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C24H26N4O4
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1
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| 1 |
Ki = 1202.26 nM
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CP0931190
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N-(3-methylamino-phenyl)-2-(2-oxo-1-(2-oxo-2-pyrrolidin-1-yl-ethyl)-5-pyridin-2-yl-1,2-dihydro-3H-1,3,4-benzotriazepin-3-yl)-acetamide
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C28H29N7O3
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1
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| 1 |
Ki = 2511.89 nM
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