| Compound ID |
Compound Name |
Compound Formula |
|
CP0502246
|
CAS_52906-92-0
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|
C120H188N34O35S
|
1
|
| 1 |
EC50 = 0.97 nM
|
|
|
|
CP0579879
|
N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]-4-[3-[2-oxo-2-(propan-2-ylamino)ethyl]phenoxy]cyclohexane-1-carboxamide
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|
C32H46N4O3
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0578448
|
4-[4-chloro-3-(hydroxymethyl)phenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C28H38ClN3O3
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0580200
|
N-[3-chloro-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]-4-(4-fluorophenoxy)-N-methylcyclohexane-1-carboxamide
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|
C26H33ClFN3O2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0574487
|
4-(4-fluorophenoxy)-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C27H36FN3O2
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0579142
|
CHEMBL5192584
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|
C30H44N4O2
|
1
|
| 1 |
EC50 = 2.6 nM
|
|
|
|
CP0576977
|
4-[3-(2-hydroxy-2-methylpropyl)phenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C31H45N3O3
|
1
|
| 1 |
EC50 = 4.3 nM
|
|
|
|
CP0579424
|
4-(5-fluoropyridin-2-yl)oxy-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C26H35FN4O2
|
1
|
| 1 |
EC50 = 4.6 nM
|
|
|
|
CP0579878
|
4-[3-(2-hydroxyethyl)phenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C29H41N3O3
|
1
|
| 1 |
EC50 = 4.7 nM
|
|
|
|
CP0579258
|
4-[3-(hydroxymethyl)phenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C28H39N3O3
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0579594
|
4-[5-(hydroxymethyl)-2-methylphenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C29H41N3O3
|
1
|
| 1 |
EC50 = 5.6 nM
|
|
|
|
CP0579593
|
4-[4-fluoro-3-(hydroxymethyl)phenoxy]-N-methyl-N-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C28H38FN3O3
|
1
|
| 1 |
EC50 = 7.5 nM
|
|
|
|
CP0579425
|
4-(2-cyanopyridin-4-yl)oxy-N-[4-[[(3S)-3-ethylpiperazin-1-yl]methyl]-3-methylphenyl]-N-methylcyclohexane-1-carboxamide
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|
C28H37N5O2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0574486
|
N-(3-fluorophenyl)-1-[3-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]pyridin-2-yl]piperidin-4-amine
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|
C28H34FN5
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0579257
|
4-(4-fluorophenoxy)-N-methyl-N-[3-methyl-4-(piperazin-1-ylmethyl)phenyl]cyclohexane-1-carboxamide
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|
C26H34FN3O2
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0320332
|
[3-[4-[[(3S,5R)-3,5-dimethylpiperazin-1-yl]methyl]phenyl]pyridin-2-yl]-[4-[(4-fluorophenyl)methyl]piperidin-1-yl]methanone
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|
C31H37FN4O
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0579877
|
4-(4-fluorophenoxy)-N-methyl-N-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C26H34FN3O2
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0576976
|
4-(4-fluorophenoxy)-N-methyl-N-[2-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C27H36FN3O2
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0551815
|
N-[4-[[(3S)-3-ethylpiperazin-1-yl]methyl]-3-methylphenyl]-4-(4-fluorophenoxy)-N-methylcyclohexane-1-carboxamide
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|
C28H38FN3O2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0136735
|
1-[4-(3-fluoroanilino)piperidin-1-yl]-2-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]ethanone
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|
C25H33FN4O
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
|
CP0579423
|
4-(4-fluorophenoxy)-N-[4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]cyclohexane-1-carboxamide
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|
C25H32FN3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0579577
|
3-[4-[methyl-[3-methyl-4-[[(3S)-3-methylpiperazin-1-yl]methyl]phenyl]carbamoyl]cyclohexyl]oxybenzoic acid
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|
C28H37N3O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
