(S)-(-)-N-(1-(3-(2-(4-isopropoxyphenoxy)thiazol-5-yl)isoxazol-5-yl)ethyl)acetamide

N-[4-[4-(4-propan-2-yloxyphenoxy)phenyl]but-3-yn-2-yl]acetamide

N-[4-[2-[4-(cyclopropylmethoxy)phenoxy]-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[1-[3-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]-1,2-oxazol-5-yl]ethyl]acetamide

2-tert-butyl-1'-(7-methyl-1H-indazole-5-carbonyl)spiro[6H-pyrano[3,2-c]pyrazole-5,4'-piperidine]-7-one

1-(4-(2-(4-(cyclopropylmethoxy)phenoxy)thiazol-5-yl)but-3-yn-2-yl)-3-methylurea

N-[4-[2-(4-phenoxyphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[4-[2-[3-chloro-4-(cyclopropylmethylamino)phenoxy]-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[1-[4-[4-(4-propoxyphenoxy)phenyl]phenyl]ethyl]acetamide

N-[4-[2-(6-propan-2-yloxypyridin-3-yl)oxy-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[(1S)-1-[3-[4-(4-phenoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

N-[4-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[1-[4-[4-[3-(cyclopropylmethoxy)phenoxy]phenoxy]phenyl]ethyl]acetamide

4-[2-(4-phenoxyphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-ylurea

methyl N-[4-[2-[4-(cyclopropylmethoxy)phenoxy]-1,3-thiazol-5-yl]but-3-yn-2-yl]carbamate

N-[1-[2-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]-1,3-thiazol-5-yl]ethyl]acetamide

1-(4-(2-(4-isopropoxyphenoxy)thiazol-5-yl)but-3-yn-2-yl)-3-methylurea

(3R)-1'-(9-anthrylcarbonyl)-3-(morpholin-4-ylcarbonyl)-1,4'-bipiperidine

(S)-(-)-{3-[2-(4-isopropoxy-phenoxy)-thiazol-4-yl]-1-methyl-prop-2ynyl}-acetamide

N-[4-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]propanamide

N-[1-[3-[4-(4-phenoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

CHEMBL1818291

N-[4-[2-(4-propan-2-ylsulfanylphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[4-[2-(4-propan-2-yloxyphenyl)sulfanyl-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

1-hydroxy-1-(4-(2-(4-phenoxyphenoxy)thiazol-5-yl)but-3-yn-2-yl)urea

tert-butyl N-[[4-[[[2-[4-(2-aminoethyl)piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

N-[(2S)-1-[[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1,3-oxazol-5-yl]oxy]propan-2-yl]acetamide

methyl N-[4-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]carbamate

N-[1-[4-[4-[3-(2-methoxyethyl)phenoxy]phenyl]phenyl]ethyl]acetamide

tert-butyl N-[[4-[[[2-[4-[2-(3-hydroxyazetidin-1-yl)ethyl]piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

N-[1-[3-[4-(4-propan-2-yloxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

tert-butyl N-[[4-[[[2-[4-[2-(dimethylamino)ethyl]piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

2,2-dimethylpropyl N-[[4-[[[2-[4-[2-(dimethylamino)ethyl]piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

N-[4-[2-[4-(propan-2-ylamino)phenoxy]-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-[1-[4-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]phenyl]ethyl]acetamide

N-[1-[2-[6-[3-(cyclopropylmethoxy)phenoxy]pyridin-3-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

tert-butyl N-[[4-[[(2-phenylquinoline-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

tert-butyl N-[[4-[[(2-pyridin-4-ylquinoline-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

N-[1-[4-[4-(3-butoxyphenoxy)phenyl]phenyl]ethyl]acetamide

N-[(1S)-1-[3-(4-phenoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]acetamide

CHEMBL1818295

tert-butyl N-[[4-[[[2-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

N-[1-[3-[4-(4-hexoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

N-[1-[3-(4-phenoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl]acetamide

N-[(2S)-1-[[2-[6-[3-(cyclopropylmethoxy)phenoxy]pyridin-3-yl]-1,3-oxazol-5-yl]oxy]propan-2-yl]acetamide

tert-butyl N-[[4-[[[2-[4-(aminomethyl)phenyl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

8-(2-phenyl-3H-benzimidazole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

N-[1-[3-[4-(4-ethoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

CHEMBL1818195

4-[2-(4-phenoxy-phenoxy)-thiazol-5-yl]-but-3-yn-2-ol

N-[1-[3-[4-(4-propoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

(R)-(+)-N-(1-(3-(2-(4-isopropoxyphenoxy)thiazol-5-yl)isoxazol-5-yl)ethyl)acetamide

tert-butyl N-[[4-[[[2-[3-[2-(dimethylamino)ethoxy]azetidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

oxan-4-yl N-[[4-[[[2-[4-[2-(dimethylamino)ethyl]piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

tert-butyl N-[[4-[[[2-[4-(aminomethyl)piperidin-1-yl]quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

tert-butyl N-[[4-[[(2-phenylquinolin-4-yl)sulfonylamino]methyl]cyclohexyl]methyl]carbamate

CHEMBL1818294

4-[4-[[4-[[(2-methylpropan-2-yl)oxycarbonylamino]methyl]cyclohexyl]methylcarbamoyl]quinolin-2-yl]benzoic acid

8-[2-(4-propan-2-ylphenyl)-3H-benzimidazole-5-carbonyl]-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

tert-butyl N-[[4-[[(6-phenyl-1H-pyrrolo[2,3-b]pyridine-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

N-[1-cyclopropyl-3-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]prop-2-ynyl]acetamide

N-[4-[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1,3-oxazol-5-yl]butan-2-yl]acetamide

N-[(2S)-1-[[2-[5-[3-(cyclopropylmethoxy)phenoxy]pyridin-2-yl]-1,3-oxazol-5-yl]oxy]propan-2-yl]acetamide

8-(7-methyl-1H-indazole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-[2-(furan-2-yl)-3H-benzimidazole-5-carbonyl]-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

tert-butyl N-[[4-[[(2-phenylquinoline-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

N-[[3-[4-(4-propan-2-yloxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]acetamide

8-(6,7,8,9-tetrahydro-5H-carbazole-3-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-(2-pyridin-4-yl-3H-benzimidazole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

tert-butyl N-[[4-[[(2-piperazin-1-ylquinoline-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

CHEMBL1818301

N-[1-[2-[5-[3-(cyclopropylmethoxy)phenoxy]pyridin-2-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

(R)-(+)-{3-[2-(4-isopropoxy-phenoxy)-thiazol-5-yl]-1-methyl-prop-2-ynyl}-carbamic acid methyl ester

CHEMBL1817676

N-[3-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]prop-2-ynyl]acetamide

methyl 4-[8-(7-methyl-1H-indazole-5-carbonyl)-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzoate

8-(7-methyl-2-propyl-3H-benzimidazole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

6-(4-aminophenyl)-N-(6-fluoro-1H-indazol-5-yl)-1-propan-2-ylpyrrolo[3,2-b]pyridine-3-carboxamide

6-(4-aminophenyl)-N-(1H-indazol-5-yl)-1-propan-2-ylpyrrolo[3,2-b]pyridine-3-carboxamide

1-methyl-3-[2-(4-phenoxy-phenoxy)-thiazol-5-yl]-prop-2-ynylamine

tert-butyl N-[[4-[(naphthalen-2-ylsulfonylamino)methyl]cyclohexyl]methyl]carbamate

8-(1H-indazole-6-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

tert-butyl N-[[4-[[[2-(3,5-dimethyl-1,2-oxazol-4-yl)quinoline-4-carbonyl]amino]methyl]cyclohexyl]methyl]carbamate

8-(2-methyl-3H-benzimidazole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-(1,2,3,4-tetrahydrocyclopenta[b]indole-7-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-(2-phenylquinolin-4-yl)methanone

1-ethyl-N-(1H-indazol-5-yl)-6-phenylpyrrolo[3,2-b]pyridine-3-carboxamide

2-methyl-4-[8-(7-methyl-1H-indazole-5-carbonyl)-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile

CHEMBL1818192

N-(1H-indazol-5-yl)-1-methyl-6-phenylpyrrolo[3,2-b]pyridine-3-carboxamide

tert-butyl N-[[4-[[(2-phenylpyridine-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

4-[8-(7-methyl-1H-indazole-5-carbonyl)-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzoic acid

N-[(2R)-1-[[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1,3-oxazol-5-yl]oxy]propan-2-yl]acetamide

tert-butyl N-[[4-[[(2-methyl-6-phenylpyridine-4-carbonyl)amino]methyl]cyclohexyl]methyl]carbamate

N-[1-[2-[3-[3-(cyclopropylmethoxy)phenoxy]azetidin-1-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

N-(1H-indazol-5-yl)-6-phenyl-1-propan-2-ylpyrrolo[3,2-b]pyridine-3-carboxamide

N-[(1R)-1-[3-[4-(4-phenoxyphenoxy)phenyl]-1,2,4-oxadiazol-5-yl]ethyl]acetamide

N-[1-[2-[6-[3-(cyclopropylmethoxy)phenoxy]pyridin-3-yl]-1,3-benzothiazol-5-yl]ethyl]acetamide

N-[1-[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1-benzothiophen-5-yl]ethyl]acetamide

N-[1-[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1,3-benzoxazol-6-yl]ethyl]acetamide

[(2S)-1-[[2-[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]-1,3-oxazol-5-yl]oxy]propan-2-yl]urea

N-[1-[3-[[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]methoxy]phenyl]ethyl]acetamide

N-[1-[2-[3-(3-butoxyphenoxy)azetidin-1-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

N-[1-[2-[3-(3-methylphenoxy)azetidin-1-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

N-[1-[2-[4-[3-(cyclopropylmethoxy)phenoxy]piperidin-1-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

N-[1-[2-[3-(3-pentylphenoxy)azetidin-1-yl]-1,3-benzoxazol-6-yl]ethyl]acetamide

N-[1-[6-[[4-[3-(cyclopropylmethoxy)phenoxy]-2,6-difluorophenyl]methoxy]pyridin-3-yl]ethyl]acetamide

N-[1-[4-[[6-[3-(cyclopropylmethoxy)phenoxy]pyridin-3-yl]methoxy]phenyl]ethyl]acetamide

N-[1-[6-[[4-[3-(cyclopropylmethoxy)phenoxy]-2,6-difluorophenyl]methoxy]pyridazin-3-yl]ethyl]acetamide

N-[1-[4-[[4-[3-(cyclopropylmethoxy)phenoxy]phenyl]methoxy]phenyl]ethyl]acetamide

N-[1-[4-[[4-[3-(cyclopropylmethoxy)phenoxy]-2-fluorophenyl]methoxy]phenyl]ethyl]acetamide

N-[1-[5-[[4-[3-(cyclopropylmethoxy)phenoxy]-2,6-difluorophenyl]methoxy]pyrazin-2-yl]ethyl]acetamide

N-[1-[4-[[5-[3-(cyclopropylmethoxy)phenoxy]pyridin-2-yl]methoxy]phenyl]ethyl]acetamide

N-[1-[4-[[4-[3-(cyclopropylmethoxy)phenoxy]-2,6-difluorophenyl]methoxy]phenyl]ethyl]acetamide

N-[1-[5-[[4-[3-(cyclopropylmethoxy)phenoxy]-2,6-difluorophenyl]methoxy]pyridin-2-yl]ethyl]acetamide

N-[4-[2-(4-propan-2-ylphenoxy)-1,3-thiazol-5-yl]but-3-yn-2-yl]acetamide

N-{3-[2-(4-isopropoxy-phenoxy)-thiazol-4-yl]-1-methyl-prop-2-ynyl}-acetamide

N-[1-phenyl-3-[2-(4-propan-2-yloxyphenoxy)-1,3-thiazol-5-yl]prop-2-ynyl]acetamide

N-[1-[4-[4-[4-(2-methoxyethyl)phenoxy]phenyl]phenyl]ethyl]acetamide

3-fluoro-4-[8-(7-methyl-1H-indazole-5-carbonyl)-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile

8-(quinoline-7-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-(quinoline-6-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

4-[8-(7-methyl-1H-indazole-5-carbonyl)-3-oxo-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile

8-(1H-indole-5-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-(quinoline-3-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one

8-(1H-indole-6-carbonyl)-2-[4-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decan-3-one