Brief Information of the Cell Line and Protein
Cell Line ID: CL000206 , PANC-1
Synonyms
Panc-1
PANC.1
Panc 1
PanC1
Panc1
PANC1
Panc-1-P
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0480
Protein ID: PT01092 , Platelet-derived growth factor receptor alpha
Gene Name PDGFRA
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P16234
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000206  Protein ID: PT01092
 
Compound ID Compound Name Compound Formula
CP0085333
Amuvatinib
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C23H21N5O3S
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0690323
N-(benzo[d][1,3]dioxol-5-ylmethyl)-4-(6,7-dimethoxy-9H-pyrimido[4,5-b]indol-4-yl)piperazine-1-carbothioamide
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C25H26N6O4S
 1
1
IC50 = 16000 nM
   TI
   LI
   LO
   TS
CP0639448
Imatinib mesilate
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C30H35N7O4S
 1
1
IC50 = 24000 nM
   TI
   LI
   LO
   TS
CP0006232
4-(6,7-Dimethoxy-quinazolin-4-yl)-piperazine-1-carbothioic acid (benzo[1,3]dioxol-5-ylmethyl)-amide
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C23H25N5O4S
 1
1
IC50 = 26600 nM
   TI
   LI
   LO
   TS
CP0173802
4-(6,7-Dimethoxy-9H-pyrimido[4,5-b]indol-4-yl)-piperazine-1-carbothioic acid [4-(pyrimidin-2-ylsulfamoyl)-phenyl]-amide
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C27H27N9O4S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0881758
4-Pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-yl-piperazine-1-carbothioic acid(benzo[1,3]dioxol-5-ylmethyl)-amide
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C22H20N6O2S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0888241
4-(6,7-dimethoxyquinazolin-4-yl)-N-(4-(N-pyrimidin-2-ylsulfamoyl)phenyl)piperazine-1-carbothioamide
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C25H26N8O4S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0895676
4-Pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-yl-piperazine-1-carbothioic acid [4-(pyrimidin-2-ylsulfamoyl)-phenyl]-amide
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C24H21N9O2S3
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS