Compound ID |
Compound Name |
Compound Formula |
CP0035405
|
7-[(3-hydroxypropyl)sulfanyl]-2-methyl-4-(2-methylpropyl)-6-(naphthalen-1-ylmethyl)-1H,2H,6H-pyrrolo[3,4-d]pyridazin-1-one
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|
C25H29N3O2S
|
1
|
1 |
Ki = 0.0955 nM
|
|
|
CP0159148
|
5-[(3-hydroxypropyl)sulfanyl]-3-methyl-1-(2-methylpropyl)-6-(naphthalen-1-ylmethyl)-1H,2H,3H,4H-thieno[2,3-d]pyrimidine-2,4-dione
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|
C25H28N2O3S2
|
1
|
1 |
Ki = 0.2754 nM
|
|
|
CP0255268
|
5-[(3-hydroxypropyl)sulfanyl]-3-methyl-1-(2-methylpropyl)-6-(naphthalen-1-ylmethyl)-1H,2H,3H,4H,6H-pyrrolo[3,4-d]pyrimidine-2,4-dione
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|
C25H29N3O3S
|
1
|
1 |
Ki = 0.3311 nM
|
|
|
CP0303011
|
5-[(3-hydroxypropyl)sulfanyl]-3-methyl-1-(2-methylpropyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H-thieno[2,3-d]pyrimidine-2,4-dione
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|
C22H25F3N2O3S2
|
1
|
1 |
Ki = 0.3548 nM
|
|
|
CP0172933
|
5-{[(3R)-3-hydroxypyrrolidin-1-yl]carbonyl}-6-(1H-indol-3-ylmethyl)-3-methyl-1-(2-methylpropyl)-1H,2H,3H,4H-thieno[2,3-d]pyrimidine-2,4-dione
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|
C25H28N4O4S
|
1
|
1 |
Ki = 3.162 nM
|
|
|
CP0384188
|
5-(2,5-dihydropyrrole-1-carbonyl)-3-methyl-1-(2-methylpropyl)-6-[[2-(trifluoromethyl)phenyl]methyl]thieno[2,3-d]pyrimidine-2,4-dione
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|
C24H24F3N3O3S
|
1
|
1 |
Ki = 3.388 nM
|
|
|
CP0159143
|
3-methyl-1-(2-methylpropyl)-5-(pyrrolidin-1-ylcarbonyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H-thieno[2,3-d]pyrimidine-2,4-dione
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|
C24H26F3N3O3S
|
1
|
1 |
Ki = 5.495 nM
|
|
|
CP0411900
|
1-Isobutyl-3-methyl-6-naphthalen-1-ylmethyl-1,6-dihydro-pyrrolo[3,4-d]pyrimidine-2,4-dione
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|
C22H23N3O2
|
1
|
1 |
Ki = 15.49 nM
|
|
|
CP0194005
|
5-{[(3R)-3-hydroxypyrrolidin-1-yl]carbonyl}-3-methyl-1-(2-methylpropyl)-6-(quinolin-4-ylmethyl)-1H,2H,3H,4H-thieno[2,3-d]pyrimidine-2,4-dione
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|
C26H28N4O4S
|
1
|
1 |
Ki = 30.9 nM
|
|
|
CP0402067
|
5-(azetidine-1-carbonyl)-1-(2-methylpropyl)-6-[[2-(trifluoromethyl)phenyl]methyl]thieno[2,3-d]pyrimidine-2,4-dione
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|
C22H22F3N3O3S
|
1
|
1 |
Ki > 199.53 nM
|
|
|