Brief Information of the Cell Line and Protein
Cell Line ID: CL001028 , CHO Pro-5
Synonyms
CHOpro-5
CHO-Pro5
CHO clone Pro-5
CHO, clone Pro5
Pro-5
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Protein ID: PT00943 , D(3) dopamine receptor
Gene Name DRD3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P35462
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL001028  Protein ID: PT00943
 
Compound ID Compound Name Compound Formula
CP0052483
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-ethyl}-amide
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C24H24BrCl2N3O2
 1
1
EC50 = 13 nM
   TI
   LI
   LO
   TS
CP0498321
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(3-chloro-phenyl)-piperazin-1-yl]-ethyl}-amide
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C24H25BrClN3O2
 1
1
EC50 = 28 nM
   TI
   LI
   LO
   TS
CP0448550
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2,3-dimethyl-phenyl)-piperazin-1-yl]-ethyl}-amide
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C26H30BrN3O2
 1
1
EC50 = 68 nM
   TI
   LI
   LO
   TS
CP0471100
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(4-phenyl-piperazin-1-yl)-ethyl]-amide
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C24H26BrN3O2
 1
1
EC50 = 68 nM
   TI
   LI
   LO
   TS
CP0458851
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2-chloro-phenyl)-piperazin-1-yl]-ethyl}-amide
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C24H25BrClN3O2
 1
1
EC50 = 83 nM
   TI
   LI
   LO
   TS
CP0406992
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(4-o-tolyl-piperazin-1-yl)-ethyl]-amide
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C25H28BrN3O2
 1
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS