Compound ID |
Compound Name |
Compound Formula |
CP0488165
|
4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]-N-cyclopropylbenzenesulfonamide
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|
C20H20N4O3S
|
1
|
1 |
IC50 = 2100 nM
|
|
|
CP0534104
|
[4-[6-amino-5-[4-(trifluoromethyl)phenyl]pyridin-3-yl]phenyl]-morpholin-4-ylmethanone
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|
C23H20F3N3O2
|
1
|
1 |
IC50 = 3000 nM
|
|
|
CP0488164
|
[4-[6-amino-5-[4-(trifluoromethyl)phenyl]pyridin-3-yl]phenyl]-piperazin-1-ylmethanone
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|
C23H21F3N4O
|
1
|
1 |
IC50 = 5500 nM
|
|
|
CP0500295
|
[4-[6-amino-5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-3-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
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|
C23H22F3N5O
|
1
|
1 |
IC50 = 8200 nM
|
|
|
CP0443891
|
4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]-N,N-dimethylbenzenesulfonamide
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|
C19H20N4O3S
|
1
|
1 |
IC50 = 9700 nM
|
|
|
CP0462608
|
3-(6-methoxypyridin-3-yl)-5-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyridin-2-amine
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|
C22H25N5O3S
|
1
|
1 |
IC50 = 10400 nM
|
|
|
CP0405111
|
[4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]phenyl]-morpholin-4-ylmethanone
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|
C22H22N4O3
|
1
|
1 |
IC50 > 11000 nM
|
|
|
CP0443898
|
4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]-N,N-dimethylbenzamide
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|
C20H20N4O2
|
1
|
1 |
IC50 > 11000 nM
|
|
|
CP0481313
|
4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]-N-methylbenzenesulfonamide
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|
C18H18N4O3S
|
1
|
1 |
IC50 > 11000 nM
|
|
|
CP0488535
|
3-(6-methoxypyridin-3-yl)-5-(4-morpholin-4-ylsulfonylphenyl)pyridin-2-amine
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|
C21H22N4O4S
|
1
|
1 |
IC50 > 11000 nM
|
|
|
CP0455516
|
[4-[6-amino-5-[4-(trifluoromethyl)phenyl]pyridin-3-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
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|
C24H23F3N4O
|
1
|
1 |
IC50 = 16300 nM
|
|
|
CP0481309
|
[4-[6-amino-5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-3-yl]phenyl]-piperazin-1-ylmethanone
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|
C22H20F3N5O
|
1
|
1 |
IC50 = 19700 nM
|
|
|
CP0488528
|
[4-[6-amino-5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-3-yl]phenyl]-morpholin-4-ylmethanone
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|
C22H19F3N4O2
|
1
|
1 |
IC50 = 20200 nM
|
|
|
CP0462607
|
[4-[6-amino-5-(6-methoxypyridin-3-yl)pyridin-3-yl]phenyl]-(4-methylpiperazin-1-yl)methanone
Show/Hide
|
C23H25N5O2
|
1
|
1 |
IC50 = 20500 nM
|
|
|