Brief Information of the Cell Line and Protein
Cell Line ID: CL000854 , GIST-5R
 Cell Line Info 
Synonyms
GIST-T1 T670I
GIST-5R
Category Cancer cell line
Organism
Homo sapiens (Human)
Protein ID: PT00888 , Mast/stem cell growth factor receptor Kit
 Protein Info 
Gene Name KIT
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P10721
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000854
 Cell Line Info 
 Protein ID: PT00888
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0421231
 Compound Info 
N-[[1-[4-[[3-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]carbamoylamino]-2-(trifluoromethyl)phenyl]piperidin-4-yl]methyl]propanamide
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C34H36F3N5O5
  2
1
EC50 < 100 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
GI50 = 26 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002211
 Compound Info 
N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
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C22H27FN4O2
  1
1
GI50 = 21 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002778
 Compound Info 
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide
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C29H31N7O
  1
1
GI50 = 8300 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS