| Compound ID |
Compound Name |
Compound Formula |
|
CP0313905
|
(1R)-9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C24H27FN4O2
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0272055
|
(1R)-9-[(3R,4R)-1,3-dimethylpiperidin-4-yl]-8-(2-fluoro-4-methoxyphenyl)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C25H29FN4O3
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0545869
|
9-(azetidin-3-ylmethyl)-1-methyl-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C16H17F3N4O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0415131
|
(1R)-1-methyl-9-[(3-methylazetidin-3-yl)amino]-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C16H18F3N5O2
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0414992
|
(1R)-9-(azetidin-3-ylamino)-1-methyl-8-phenyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C20H21N5O2
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0379271
|
9-(azetidin-3-ylamino)-1-methyl-8-propan-2-yl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C17H23N5O2
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0536608
|
9-(azetidin-3-ylamino)-1-methyl-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H16F3N5O2
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0381408
|
(1S)-9-(azetidin-3-ylamino)-1-methyl-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H16F3N5O2
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0415465
|
9-(azetidin-3-yloxy)-1-methyl-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H15F3N4O3
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0536778
|
(1S)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H19N5O2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0548319
|
9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H19N5O2
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0379253
|
(1R)-9-(azetidin-3-ylamino)-1-methyl-8-(trifluoromethyl)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H16F3N5O2
|
1
|
| 1 |
IC50 = 4600 nM
|
|
|
|
CP0411801
|
(1R)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H19N5O2
|
1
|
| 1 |
IC50 = 5100 nM
|
|
|
|
CP0545878
|
9-(azetidin-3-ylamino)-1-ethyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C15H19N5O2
|
1
|
| 1 |
IC50 = 5400 nM
|
|
|
|
CP0548321
|
(1S)-9-(azetidin-3-ylamino)-1-methyl-8-phenyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C20H21N5O2
|
1
|
| 1 |
IC50 = 6600 nM
|
|
|
|
CP0410898
|
9-(azetidin-3-ylamino)-8-fluoro-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C14H16FN5O2
|
1
|
| 1 |
IC50 = 6900 nM
|
|
|
|
CP0550777
|
9-(azetidin-3-ylamino)-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C13H15N5O2
|
1
|
| 1 |
IC50 = 7100 nM
|
|
|
|
CP0414991
|
9-(azetidin-3-ylamino)-1-methyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C14H17N5O2
|
1
|
| 1 |
IC50 = 9400 nM
|
|
|
|
CP0361044
|
3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C10H9N3O2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
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CP0415466
|
9-(azetidin-3-ylamino)-1-phenyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C19H19N5O2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0548320
|
9-(azetidin-3-ylamino)-1-cyclopropyl-3,5-dihydro-1H-[1,2,4]triazino[3,4-c][1,4]benzoxazin-2-one
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|
C16H19N5O2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0012721
|
[3-[4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl]azetidin-1-yl]-[4-[[(2S)-2,3-dihydroxypropoxy]methyl]pyridin-2-yl]methanone
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|
C30H34N2O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
