General Information of the Compound
Compound ID
CP0969459
Compound Name
1-((1-acryloyl-3-fluoroazetidin-3-yl)methyl)-7-chloro-6-(2-fluorophenyl)-4-(2-isopropyl-4-methylpyridin-3-yl)pyrido[2,3-b]pyrazine-2,3(1H,4H)-dione
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Formula
C29H26ClF2N5O3
Molecular Weight
566.008
Canonical SMILES
C=CC(=O)N1CC(F)(Cn2c(=O)c(=O)n(-c3c(C)ccnc3C(C)C)c3nc(-c4ccccc4F)c(Cl)cc32)C1
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InChI
InChI=1S/C29H26ClF2N5O3/c1-5-22(38)35-13-29(32,14-35)15-36-21-12-19(30)24(18-8-6-7-9-20(18)31)34-26(21)37(28(40)27(36)39)25-17(4)10-11-33-23(25)16(2)3/h5-12,16H,1,13-15H2,2-4H3
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InChIKey
PMXJKTZZNXKQDL-UHFFFAOYSA-N
Physicochemical Property
logP
4.57022
Rotatable Bonds
6
Heavy Atom Count
40
Polar Areas
90.09
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
7
Complexity
40

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03462, GTPase KRas
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000207 MIA PaCa-2 Homo sapiens (Human)  1
1
IC50 <= 100 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 <= 100 nM