General Information of the Compound
Compound ID
CP0955948
Compound Name
N-[4-[(E)-2-[4-[(5-Methyl-1,3-thiazol-2-yl)amino]-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl]ethenyl]phenyl]prop-2-enamide
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Formula
C24H27N7OS
Molecular Weight
461.595
Canonical SMILES
C=CC(=O)Nc1ccc(/C=C/c2nc(Nc3ncc(C)s3)cc(N3CCN(C)CC3)n2)cc1
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InChI
InChI=1S/C24H27N7OS/c1-4-23(32)26-19-8-5-18(6-9-19)7-10-20-27-21(29-24-25-16-17(2)33-24)15-22(28-20)31-13-11-30(3)12-14-31/h4-10,15-16H,1,11-14H2,2-3H3,(H,26,32)(H,25,27,28,29)/b10-7+
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InChIKey
LDOCDWKQVMOLLD-JXMROGBWSA-N
Physicochemical Property
logP
4.03182
Rotatable Bonds
7
Heavy Atom Count
33
Polar Areas
86.28
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4764283
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01411, Fibroblast growth factor receptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 1.2 nM
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