General Information of the Compound
Compound ID
CP0953363
Compound Name
(S)-1-(4-(7-(5-Isopropyl-1H-indazol-4-yl)-2-((1-methylpyrrolidin-2-yl)methoxy)-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperazin-1-yl)prop-2-en-1-one
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Structure
Formula
C30H40N8O2
Molecular Weight
544.704
Canonical SMILES
C=CC(=O)N1CCN(c2nc(OC[C@@H]3CCCN3C)nc3c2CCN(c2c(C(C)C)ccc4[nH]ncc24)C3)CC1
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InChI
InChI=1S/C30H40N8O2/c1-5-27(39)36-13-15-37(16-14-36)29-23-10-12-38(28-22(20(2)3)8-9-25-24(28)17-31-34-25)18-26(23)32-30(33-29)40-19-21-7-6-11-35(21)4/h5,8-9,17,20-21H,1,6-7,10-16,18-19H2,2-4H3,(H,31,34)/t21-/m0/s1
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InChIKey
PQYZPEBTMDDKNX-NRFANRHFSA-N
Physicochemical Property
logP
3.3466
Rotatable Bonds
7
Heavy Atom Count
40
Polar Areas
93.72
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
40

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 134325886
ChEMBL ID
CHEMBL4642347
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03462, GTPase KRas
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000268 NCI-H358 Homo sapiens (Human)  1
1
IC50 = 1180 nM
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