General Information of the Compound
Compound ID
CP0931560
Compound Name
SID49681549
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Synonyms
133073-73-1
4-Amino-10-methylfolic acid hydrate
6745-93-3
84DMZ3IHO0
AC1L4WT9
AC1Q5QR4
Abitrexate(Methotrexate)/
Antifolan hydrate
C20H22N8O5.xH2O
CH4474
L-Amethopterin hydrate
L-Amethopterin hydrate, 98%
L-Glutamic acid, N-[4-[[(2,4-diamino-6-pteridinyl)methyl]methylamino]benzoyl]- [CAS]
MLS000758248
MLS001401431
MTX hydrate
Methotrexate hydrate
Methotrexate hydrate(1:x)
Methotrexate monohydrate
Methotrexate trihydrate
Methylaminopterin hydrate
SCHEMBL1230252
SMR000449324
UNII-84DMZ3IHO0
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Structure
Formula
C20H24N8O6
Molecular Weight
472.462
Canonical SMILES
CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1.O
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InChI
InChI=1S/C20H22N8O5.H2O/c1-28(9-11-8-23-17-15(24-11)16(21)26-20(22)27-17)12-4-2-10(3-5-12)18(31)25-13(19(32)33)6-7-14(29)30;/h2-5,8,13H,6-7,9H2,1H3,(H,25,31)(H,29,30)(H,32,33)(H4,21,22,23,26,27);1H2/t13-;/m0./s1
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InChIKey
FPJYMUQSRFJSEW-ZOWNYOTGSA-N
CAS
6745-93-3
Physicochemical Property
logP
-0.5563
Rotatable Bonds
9
Heavy Atom Count
34
Polar Areas
242.04
Hydrogen Bond Donor Count
5
Hydrogen Bond Acceptor Count
10
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 165528
ChEMBL ID
CHEMBL1376974
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT06109, Geminin
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000015 SW480 Homo sapiens (Human)  1
1
Potency ~ 89.1 nM
   TI
   LI
   LO
   TS
Protein ID: PT06101, Latent membrane protein 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
AC50 = 16 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( CH4474 )
Drug Name CH4474
Target(s)
TNF alpha converting enzyme (ADAM17)
Inhibitor