General Information of the Compound
Compound ID
CP0917640
Compound Name
N-[4-[(E)-2-(4-[[5-(Methoxymethyl)-1H-pyrazol-3-yl]amino]-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl)ethenyl]phenyl]prop-2-enamide
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Formula
C25H30N8O2
Molecular Weight
474.569
Canonical SMILES
C=CC(=O)Nc1ccc(/C=C/c2nc(Nc3cc(COC)[nH]n3)cc(N3CCN(C)CC3)n2)cc1
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InChI
InChI=1S/C25H30N8O2/c1-4-25(34)26-19-8-5-18(6-9-19)7-10-21-27-22(28-23-15-20(17-35-3)30-31-23)16-24(29-21)33-13-11-32(2)12-14-33/h4-10,15-16H,1,11-14,17H2,2-3H3,(H,26,34)(H2,27,28,29,30,31)/b10-7+
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InChIKey
QXBOYPMAXNKWLR-JXMROGBWSA-N
Physicochemical Property
logP
3.1364
Rotatable Bonds
9
Heavy Atom Count
35
Polar Areas
111.3
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
8
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4777595
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01411, Fibroblast growth factor receptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  2
1
GI50 = 1.3 nM
   TI
   LI
   LO
   TS
2
GI50 = 3.4 nM
   TI
   LI
   LO
   TS