General Information of the Compound
Compound ID
CP0916304
Compound Name
N-((R)-1-{4-[3-(3-Chloro-4-fluoro-phenyl)-1-(3''-cyano-biphenyl-4-yl)-ureido]-butyl}-pyrrolidin-3-yl)-acetamide
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Structure
Formula
C30H31ClFN5O2
Molecular Weight
548.062
Canonical SMILES
CC(=O)N[C@@H]1CCN(CCCCN(C(=O)Nc2ccc(F)c(Cl)c2)c2ccc(-c3cccc(C#N)c3)cc2)C1
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InChI
InChI=1S/C30H31ClFN5O2/c1-21(38)34-26-13-16-36(20-26)14-2-3-15-37(30(39)35-25-9-12-29(32)28(31)18-25)27-10-7-23(8-11-27)24-6-4-5-22(17-24)19-33/h4-12,17-18,26H,2-3,13-16,20H2,1H3,(H,34,38)(H,35,39)/t26-/m1/s1
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InChIKey
JGPFRAZKWWKZBV-AREMUKBSSA-N
Physicochemical Property
logP
6.04688
Rotatable Bonds
9
Heavy Atom Count
39
Polar Areas
88.47
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
4
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10166038
SID: 15159191
ChEMBL ID
CHEMBL360006
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01027, Melanin-concentrating hormone receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki < 100 nM
   TI
   LI
   LO
   TS