General Information of the Compound
Compound ID
CP0915610
Compound Name
TTWEAWDRAIAEYAARIEALIR
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Structure
Formula
C118H181N33O34
Molecular Weight
2605.943
Canonical SMILES
CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@@H](N)[C@@H](C)O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@H](C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCCNC(=N)N)C(=O)O)[C@@H](C)CC)[C@@H](C)CC
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InChI
InChI=1S/C118H181N33O34/c1-17-55(6)90(148-99(168)63(14)134-100(169)74(31-24-44-126-116(120)121)139-108(177)84(51-88(161)162)146-107(176)82(49-67-52-129-72-29-22-20-27-70(67)72)144-98(167)61(12)132-101(170)76(38-41-85(155)156)140-106(175)83(50-68-53-130-73-30-23-21-28-71(68)73)147-114(183)93(65(16)153)151-110(179)89(119)64(15)152)111(180)136-62(13)96(165)138-78(40-43-87(159)160)103(172)145-81(48-66-34-36-69(154)37-35-66)105(174)135-58(9)94(163)131-59(10)95(164)137-75(32-25-45-127-117(122)123)104(173)149-91(56(7)18-2)112(181)141-77(39-42-86(157)158)102(171)133-60(11)97(166)143-80(47-54(4)5)109(178)150-92(57(8)19-3)113(182)142-79(115(184)185)33-26-46-128-118(124)125/h20-23,27-30,34-37,52-65,74-84,89-93,129-130,152-154H,17-19,24-26,31-33,38-51,119H2,1-16H3,(H,131,163)(H,132,170)(H,133,171)(H,134,169)(H,135,174)(H,136,180)(H,137,164)(H,138,165)(H,139,177)(H,140,175)(H,141,181)(H,142,182)(H,143,166)(H,144,167)(H,145,172)(H,146,176)(H,147,183)(H,148,168)(H,149,173)(H,150,178)(H,151,179)(H,155,156)(H,157,158)(H,159,160)(H,161,162)(H,184,185)(H4,120,121,126)(H4,122,123,127)(H4,124,125,128)/t55-,56-,57-,58-,59-,60-,61-,62-,63-,64+,65+,74-,75-,76-,77-,78-,79-,80-,81-,82-,83-,84-,89-,90-,91-,92-,93-/m0/s1
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InChIKey
RYIOERNWDZGPBY-GUWXJHCASA-N
Physicochemical Property
logP
-7.10029
Rotatable Bonds
82
Heavy Atom Count
185
Polar Areas
1101.59
Hydrogen Bond Donor Count
41
Hydrogen Bond Acceptor Count
33
Complexity
185

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 122184658
ChEMBL ID
CHEMBL3600955
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03571, Envelope glycoprotein gp160
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000291 HL2/3 Homo sapiens (Human)  1
1
IC50 > 2250 nM
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