General Information of the Compound
Compound ID
CP0906581
Compound Name
1-methylcyclopropyl 9-(5-fluoro-6-(2-fluoro-4-(1H-1,2,4-triazol-1-yl)phenylamino)pyrimidin-4-yloxy)-3-oxa-7-azabicyclo[3.3.1]nonane-7-carboxylate
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Structure
Formula
C24H25F2N7O4
Molecular Weight
513.505
Canonical SMILES
CC1(OC(=O)N2CC3COCC(C2)C3Oc2ncnc(Nc3ccc(-n4cncn4)cc3F)c2F)CC1
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InChI
InChI=1S/C24H25F2N7O4/c1-24(4-5-24)37-23(34)32-7-14-9-35-10-15(8-32)20(14)36-22-19(26)21(28-12-29-22)31-18-3-2-16(6-17(18)25)33-13-27-11-30-33/h2-3,6,11-15,20H,4-5,7-10H2,1H3,(H,28,29,31)
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InChIKey
AFFLSSIXCBCWOQ-UHFFFAOYSA-N
Physicochemical Property
logP
3.0938
Rotatable Bonds
6
Heavy Atom Count
37
Polar Areas
116.52
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
10
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 68036951
ChEMBL ID
CHEMBL4172962
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02455, Glucose-dependent insulinotropic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 19 nM
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