General Information of the Compound
Compound ID
CP0896986
Compound Name
(R)-1-(3-(4-Amino-3-(2-chloro-4-((3-fluorobenzyl)oxy)phenyl)-1Hpyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one
    Show/Hide
Structure
Formula
C26H24ClFN6O2
Molecular Weight
506.969
Canonical SMILES
C=CC(=O)N1CCC[C@@H](n2nc(-c3ccc(OCc4cccc(F)c4)cc3Cl)c3c(N)ncnc32)C1
    Show/Hide
InChI
InChI=1S/C26H24ClFN6O2/c1-2-22(35)33-10-4-7-18(13-33)34-26-23(25(29)30-15-31-26)24(32-34)20-9-8-19(12-21(20)27)36-14-16-5-3-6-17(28)11-16/h2-3,5-6,8-9,11-12,15,18H,1,4,7,10,13-14H2,(H2,29,30,31)/t18-/m1/s1
    Show/Hide
InChIKey
URKYUDFEWHAZBC-GOSISDBHSA-N
Physicochemical Property
logP
4.7965
Rotatable Bonds
6
Heavy Atom Count
36
Polar Areas
99.16
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
7
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 130203595
ChEMBL ID
CHEMBL4094291
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 170 nM
   TI
   LI
   LO
   TS