General Information of the Compound
Compound ID
CP0891837
Compound Name
(2R,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-carboxylic acid methylamide
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Structure
Formula
C20H19N5O4
Molecular Weight
393.403
Canonical SMILES
CCC(=O)[C@H]1O[C@@H](n2cnc3c(N)nc(C#Cc4ccccc4)nc32)[C@H](O)[C@@H]1O
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InChI
InChI=1S/C20H19N5O4/c1-2-12(26)17-15(27)16(28)20(29-17)25-10-22-14-18(21)23-13(24-19(14)25)9-8-11-6-4-3-5-7-11/h3-7,10,15-17,20,27-28H,2H2,1H3,(H2,21,23,24)/t15-,16+,17+,20+/m0/s1
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InChIKey
MBXWXPUSFDNWKE-TVKQPGBESA-N
Physicochemical Property
logP
0.4066
Rotatable Bonds
3
Heavy Atom Count
29
Polar Areas
136.38
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
9
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 46905977
ChEMBL ID
CHEMBL1162942
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00840, Adenosine receptor A1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3920 nM
   TI
   LI
   LO
   TS
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1760 nM
   TI
   LI
   LO
   TS
Protein ID: PT01279, Adenosine receptor A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 7.3 nM
   TI
   LI
   LO
   TS