General Information of the Compound
Compound ID
CP0883790
Compound Name
N1,N7-bis(2-(2-(2-(3-((S)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)phenylsulfonamido)ethoxy)ethoxy)ethyl)-4-(3-(2-(2-(2-(3-((S)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)phenylsulfonamido)ethoxy)ethoxy)ethylamino)-3-oxopropyl)-4-(4-(2-(2-hydroxyethoxy)ethyl)piperazine-1-carboxamido)heptanediamide
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Structure
Formula
C85H114Cl6N12O18S3
Molecular Weight
1900.832
Canonical SMILES
CN1Cc2c(Cl)cc(Cl)cc2[C@H](c2cccc(S(=O)(=O)NCCOCCOCCNC(=O)CCC(CCC(=O)NCCOCCOCCNS(=O)(=O)c3cccc([C@@H]4CN(C)Cc5c(Cl)cc(Cl)cc54)c3)(CCC(=O)NCCOCCOCCNS(=O)(=O)c3cccc([C@@H]4CN(C)Cc5c(Cl)cc(Cl)cc54)c3)NC(=O)N3CCN(CCOCCO)CC3)c2)C1
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InChI
InChI=1S/C85H114Cl6N12O18S3/c1-99-54-72(69-48-63(86)51-78(89)75(69)57-99)60-7-4-10-66(45-60)122(109,110)95-22-34-118-42-39-115-31-19-92-81(105)13-16-85(98-84(108)103-27-25-102(26-28-103)29-37-121-38-30-104,17-14-82(106)93-20-32-116-40-43-119-35-23-96-123(111,112)67-11-5-8-61(46-67)73-55-100(2)58-76-70(73)49-64(87)52-79(76)90)18-15-83(107)94-21-33-117-41-44-120-36-24-97-124(113,114)68-12-6-9-62(47-68)74-56-101(3)59-77-71(74)50-65(88)53-80(77)91/h4-12,45-53,72-74,95-97,104H,13-44,54-59H2,1-3H3,(H,92,105)(H,93,106)(H,94,107)(H,98,108)/t72-,73-,74-/m0/s1
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InChIKey
QKOPFAPFIMPUGO-GSWCZOIBSA-N
Physicochemical Property
logP
8.4379
Rotatable Bonds
51
Heavy Atom Count
124
Polar Areas
355.95
Hydrogen Bond Donor Count
8
Hydrogen Bond Acceptor Count
22
Complexity
124

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 86272547
ChEMBL ID
CHEMBL3979858
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS