General Information of the Compound
Compound ID
CP0882777
Compound Name
endo-8-(bis(2-chlorophenyl)methyl)-3-(5-carbamoylpyridin-2-yl)-8-azabicyclo[3.2.1]octane-3-carboxamide
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Formula
C27H26Cl2N4O2
Molecular Weight
509.437
Canonical SMILES
NC(=O)c1ccc([C@@]2(C(N)=O)C[C@H]3CC[C@@H](C2)N3C(c2ccccc2Cl)c2ccccc2Cl)nc1
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InChI
InChI=1S/C27H26Cl2N4O2/c28-21-7-3-1-5-19(21)24(20-6-2-4-8-22(20)29)33-17-10-11-18(33)14-27(13-17,26(31)35)23-12-9-16(15-32-23)25(30)34/h1-9,12,15,17-18,24H,10-11,13-14H2,(H2,30,34)(H2,31,35)/t17-,18+,27-
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InChIKey
ICMCDZNDWXJNGE-SCDHDWPVSA-N
Physicochemical Property
logP
4.6268
Rotatable Bonds
6
Heavy Atom Count
35
Polar Areas
102.31
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
4
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL3084538
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1315 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 401 nM
   TI
   LI
   LO
   TS