General Information of the Compound
Compound ID
CP0875557
Compound Name
1-[2-[2-[2-[4-[3-(6-chloro-2-guanidino-quinazolin-4-yl)phenyl]piperazin-1-yl]ethoxy]ethoxy]ethyl]-3-[2-[2-[2-[4-[2-[2-[2-[2-[2-[2-[4-[3-(6-chloro-2-guanidino-quinazolin-4-yl)phenyl]piperazin-1-yl]ethoxy]ethoxy]ethylcarbamoylamino]ethoxy]ethoxy]ethylcarbamoylamino]butylcarbamoylamino]ethoxy]ethoxy]ethyl]urea
    Show/Hide
Structure
Formula
C70H102Cl2N22O12
Molecular Weight
1514.634
Canonical SMILES
NC(N)=Nc1nc(-c2cccc(N3CCN(CCOCCOCCNC(=O)NCCOCCOCCNC(=O)NCCCCNC(=O)NCCOCCOCCNC(=O)NCCOCCOCCN4CCN(c5cccc(-c6nc(N=C(N)N)nc7ccc(Cl)cc67)c5)CC4)CC3)c2)c2cc(Cl)ccc2n1
    Show/Hide
InChI
InChI=1S/C70H102Cl2N22O12/c71-53-9-11-59-57(49-53)61(87-65(85-59)89-63(73)74)51-5-3-7-55(47-51)93-25-21-91(22-26-93)29-37-105-45-43-103-35-19-83-69(97)81-17-33-101-41-39-99-31-15-79-67(95)77-13-1-2-14-78-68(96)80-16-32-100-40-42-102-34-18-82-70(98)84-20-36-104-44-46-106-38-30-92-23-27-94(28-24-92)56-8-4-6-52(48-56)62-58-50-54(72)10-12-60(58)86-66(88-62)90-64(75)76/h3-12,47-50H,1-2,13-46H2,(H2,77,79,95)(H2,78,80,96)(H2,81,83,97)(H2,82,84,98)(H4,73,74,85,87,89)(H4,75,76,86,88,90)
    Show/Hide
InChIKey
RDFNWWCDBGKOFD-UHFFFAOYSA-N
Physicochemical Property
logP
3.0776
Rotatable Bonds
47
Heavy Atom Count
106
Polar Areas
431.68
Hydrogen Bond Donor Count
12
Hydrogen Bond Acceptor Count
22
Complexity
106

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 134155307
ChEMBL ID
CHEMBL3962344
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS