General Information of the Compound
Compound ID
CP0870485
Compound Name
N-[4-[(E)-2-[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl]ethenyl]phenyl]prop-2-enamide
    Show/Hide
Formula
C26H30N8O
Molecular Weight
470.581
Canonical SMILES
C=CC(=O)Nc1ccc(/C=C/c2nc(Nc3cc(C4CC4)[nH]n3)cc(N3CCN(C)CC3)n2)cc1
    Show/Hide
InChI
InChI=1S/C26H30N8O/c1-3-26(35)27-20-9-4-18(5-10-20)6-11-22-28-23(29-24-16-21(31-32-24)19-7-8-19)17-25(30-22)34-14-12-33(2)13-15-34/h3-6,9-11,16-17,19H,1,7-8,12-15H2,2H3,(H,27,35)(H2,28,29,30,31,32)/b11-6+
    Show/Hide
InChIKey
RPSAMANQENELCZ-IZZDOVSWSA-N
Physicochemical Property
logP
3.8674
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
102.07
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
ChEMBL ID
CHEMBL4756501
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01411, Fibroblast growth factor receptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 4 nM
   TI
   LI
   LO
   TS