General Information of the Compound
Compound ID
CP0868807
Compound Name
Rac-1-[3-(4-[4-[(5-Methyl-1H-pyrazol-3-yl)amino]-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl]phenyl)pyrrolidin-1-yl]prop-2-en-1-one
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Formula
C26H32N8O
Molecular Weight
472.597
Canonical SMILES
C=CC(=O)N1CCC(c2ccc(-c3nc(Nc4cc(C)[nH]n4)cc(N4CCN(C)CC4)n3)cc2)C1
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InChI
InChI=1S/C26H32N8O/c1-4-25(35)34-10-9-21(17-34)19-5-7-20(8-6-19)26-28-22(27-23-15-18(2)30-31-23)16-24(29-26)33-13-11-32(3)12-14-33/h4-8,15-16,21H,1,9-14,17H2,2-3H3,(H2,27,28,29,30,31)
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InChIKey
BHIGBIGJIDWVOR-UHFFFAOYSA-N
Physicochemical Property
logP
3.17242
Rotatable Bonds
6
Heavy Atom Count
35
Polar Areas
93.28
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4765110
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01411, Fibroblast growth factor receptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  2
1
GI50 = 5.2 nM
   TI
   LI
   LO
   TS
2
GI50 = 20 nM
   TI
   LI
   LO
   TS