General Information of the Compound
Compound ID
CP0868801
Compound Name
4-((2-((2R)-4-(5-(1,4-dioxan-2-yl)-1,2,4-oxadiazol-3-yl)-2-methylpiperazin-1-yl)pyrimidin-5-yloxy)methyl)nicotinonitrile
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Structure
Formula
C22H24N8O4
Molecular Weight
464.486
Canonical SMILES
C[C@@H]1CN(c2noc(C3COCCO3)n2)CCN1c1ncc(OCc2ccncc2C#N)cn1
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InChI
InChI=1S/C22H24N8O4/c1-15-12-29(22-27-20(34-28-22)19-14-31-6-7-32-19)4-5-30(15)21-25-10-18(11-26-21)33-13-16-2-3-24-9-17(16)8-23/h2-3,9-11,15,19H,4-7,12-14H2,1H3/t15-,19?/m1/s1
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InChIKey
BDCALHIYMZXLRA-NYRJJRHWSA-N
Physicochemical Property
logP
1.50828
Rotatable Bonds
6
Heavy Atom Count
34
Polar Areas
135.55
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
12
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 90666908
ChEMBL ID
CHEMBL3220233
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02455, Glucose-dependent insulinotropic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 100 nM
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   LI
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Protein ID: PT02398, Glucose-dependent insulinotropic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 630.96 nM
   TI
   LI
   LO
   TS