General Information of the Compound
Compound ID
CP0862453
Compound Name
N-(4-chloro-2-hydroxy-3-{[(3-exo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl]sulfonyl}phenyl)-N'-(3-fluoro-2-methylphenyl)urea
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Formula
C22H25ClFN3O4S
Molecular Weight
481.977
Canonical SMILES
Cc1c(F)cccc1NC(=O)Nc1ccc(Cl)c(S(=O)(=O)[C@@H]2C[C@H]3CC[C@@H](C2)N3C)c1O
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InChI
InChI=1S/C22H25ClFN3O4S/c1-12-17(24)4-3-5-18(12)25-22(29)26-19-9-8-16(23)21(20(19)28)32(30,31)15-10-13-6-7-14(11-15)27(13)2/h3-5,8-9,13-15,28H,6-7,10-11H2,1-2H3,(H2,25,26,29)/t13-,14+,15-
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InChIKey
DUNGAEKWCMZUQI-QDMKHBRRSA-N
Physicochemical Property
logP
4.53602
Rotatable Bonds
4
Heavy Atom Count
32
Polar Areas
98.74
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
5
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL3941989
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01304, C-X-C chemokine receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 < 30000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01013, C-X-C chemokine receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 5 nM
   TI
   LI
   LO
   TS
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 < 30000 nM
   TI
   LI
   LO
   TS