General Information of the Compound
Compound ID
CP0859622
Compound Name
(rel)-8-(bis(2-chlorophenyl)methyl)-5'-fluoro-8-azaspiro[bicyclo[3.2.1]octane-3,3'-indoline]
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Formula
C27H25Cl2FN2
Molecular Weight
467.415
Canonical SMILES
Fc1ccc2c(c1)[C@]1(CN2)C[C@H]2CC[C@@H](C1)N2C(c1ccccc1Cl)c1ccccc1Cl
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InChI
InChI=1S/C27H25Cl2FN2/c28-23-7-3-1-5-20(23)26(21-6-2-4-8-24(21)29)32-18-10-11-19(32)15-27(14-18)16-31-25-12-9-17(30)13-22(25)27/h1-9,12-13,18-19,26,31H,10-11,14-16H2/t18-,19+,27-
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InChIKey
UJWRBOKPPNAWPV-MZNYFNKISA-N
Physicochemical Property
logP
7.2122
Rotatable Bonds
3
Heavy Atom Count
32
Polar Areas
15.27
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
2
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL3349284
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1706 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 39 nM
   TI
   LI
   LO
   TS