General Information of the Compound
Compound ID
CP0852726
Compound Name
3-{(2,3-dihydro-1'H-spiro[indene-1,4'-piperidin]-1'-yl)methyl}-1,2,3,4-tetrahydroisoquinolin-8-ol
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Structure
Formula
C23H28N2O
Molecular Weight
348.49
Canonical SMILES
Oc1cccc2c1CNC(CN1CCC3(CCc4ccccc43)CC1)C2
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InChI
InChI=1S/C23H28N2O/c26-22-7-3-5-18-14-19(24-15-20(18)22)16-25-12-10-23(11-13-25)9-8-17-4-1-2-6-21(17)23/h1-7,19,24,26H,8-16H2
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InChIKey
LSDHJVNCQHDVCX-UHFFFAOYSA-N
Physicochemical Property
logP
3.3865
Rotatable Bonds
2
Heavy Atom Count
26
Polar Areas
35.5
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
3
Complexity
26

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 11544795
SID: 16646977
ChEMBL ID
CHEMBL3785718
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 288 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 53.9 nM
   TI
   LI
   LO
   TS
2
Ki = 2.4 nM
   TI
   LI
   LO
   TS
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 940 nM
   TI
   LI
   LO
   TS