General Information of the Compound
Compound ID
CP0706577
Compound Name
Exo-8-[bis(2-chorophenyl)methyl]-3-(6-methoxy-2-pyridinyl)-8-azabicyclo[3.2.1]octane
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Formula
C26H26Cl2N2O
Molecular Weight
453.413
Canonical SMILES
COc1cccc([C@H]2C[C@H]3CC[C@@H](C2)N3C(c2ccccc2Cl)c2ccccc2Cl)n1
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InChI
InChI=1S/C26H26Cl2N2O/c1-31-25-12-6-11-24(29-25)17-15-18-13-14-19(16-17)30(18)26(20-7-2-4-9-22(20)27)21-8-3-5-10-23(21)28/h2-12,17-19,26H,13-16H2,1H3/t17-,18+,19-
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InChIKey
ORTSEGKOUGBFOV-REPLKXPHSA-N
Physicochemical Property
logP
6.897
Rotatable Bonds
5
Heavy Atom Count
31
Polar Areas
25.36
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
3
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
SID: 85282830
ChEMBL ID
CHEMBL3084636
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 421 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 9 nM
   TI
   LI
   LO
   TS