General Information of the Compound
Compound ID
CP0578416
Compound Name
(3R,4R)-4-fluoro-1-[6-fluoro-1-[(5-fluoropyrimidin-2-yl)methyl]benzimidazol-2-yl]piperidin-3-amine
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Structure
Formula
C17H17F3N6
Molecular Weight
362.359
Canonical SMILES
N[C@@H]1CN(CC[C@H]1F)c1nc2ccc(F)cc2n1Cc1ncc(F)cn1
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InChI
InChI=1S/C17H17F3N6/c18-10-1-2-14-15(5-10)26(9-16-22-6-11(19)7-23-16)17(24-14)25-4-3-12(20)13(21)8-25/h1-2,5-7,12-13H,3-4,8-9,21H2/t12-,13-/m1/s1
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InChIKey
DONHKZQWJGOSSY-CHWSQXEVSA-N
Physicochemical Property
logP
2.0283
Rotatable Bonds
3
Heavy Atom Count
26
Polar Areas
72.86
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
26

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 155193884
ChEMBL ID
CHEMBL4741505
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT04958, Short transient receptor potential channel 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 0.2 nM
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