General Information of the Compound
Compound ID
CP0576627
Compound Name
[4-[[2-amino-4-(butylamino)pyrido[3,2-d]pyrimidin-6-yl]methyl]phenyl]-pyrrolidin-1-ylmethanone
    Show/Hide
Structure
Formula
C23H28N6O
Molecular Weight
404.518
Canonical SMILES
CCCCNc1nc(N)nc2ccc(Cc3ccc(cc3)C(=O)N3CCCC3)nc12
    Show/Hide
InChI
InChI=1S/C23H28N6O/c1-2-3-12-25-21-20-19(27-23(24)28-21)11-10-18(26-20)15-16-6-8-17(9-7-16)22(30)29-13-4-5-14-29/h6-11H,2-5,12-15H2,1H3,(H3,24,25,27,28)
    Show/Hide
InChIKey
DKOULUBCLGBNCT-UHFFFAOYSA-N
Physicochemical Property
logP
3.6458
Rotatable Bonds
7
Heavy Atom Count
30
Polar Areas
97.03
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 166635334
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02160, Toll-like receptor 7
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 95 nM
   TI
   LI
   LO
   TS
Protein ID: PT02546, Toll-like receptor 8
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 67 nM
   TI
   LI
   LO
   TS