General Information of the Compound
Compound ID
CP0574100
Compound Name
1'-[3-(dimethylamino)prop-2-ynoyl]-2-[2-(2-methoxyanilino)pyrimidin-4-yl]spiro[5,6-dihydro-1H-pyrrolo[3,2-c]pyridine-7,4'-piperidine]-4-one
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Structure
Formula
C27H29N7O3
Molecular Weight
499.575
Canonical SMILES
COc1ccccc1Nc1nccc(n1)-c1cc2c([nH]1)C1(CCN(CC1)C(=O)C#CN(C)C)CNC2=O
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InChI
InChI=1S/C27H29N7O3/c1-33(2)13-9-23(35)34-14-10-27(11-15-34)17-29-25(36)18-16-21(30-24(18)27)19-8-12-28-26(31-19)32-20-6-4-5-7-22(20)37-3/h4-8,12,16,30H,10-11,14-15,17H2,1-3H3,(H,29,36)(H,28,31,32)
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InChIKey
HXUNBLWPPKQBAN-UHFFFAOYSA-N
Physicochemical Property
logP
2.35
Rotatable Bonds
4
Heavy Atom Count
37
Polar Areas
115.48
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 166636348
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000157 NCI-H1975 Homo sapiens (Human)  1
1
EC50 = 2180 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2.8 nM
2 IC50 = 5.3 nM