General Information of the Compound
Compound ID
CP0573660
Compound Name
3-[5-amino-6-(2-methyl-1,3-thiazol-5-yl)pyrazin-2-yl]-N-(4,4-difluorocyclohexyl)-4-methylbenzenesulfonamide
    Show/Hide
Structure
Formula
C21H23F2N5O2S2
Molecular Weight
479.578
Canonical SMILES
Cc1ncc(s1)-c1nc(cnc1N)-c1cc(ccc1C)S(=O)(=O)NC1CCC(F)(F)CC1
    Show/Hide
InChI
InChI=1S/C21H23F2N5O2S2/c1-12-3-4-15(32(29,30)28-14-5-7-21(22,23)8-6-14)9-16(12)17-10-26-20(24)19(27-17)18-11-25-13(2)31-18/h3-4,9-11,14,28H,5-8H2,1-2H3,(H2,24,26)
    Show/Hide
InChIKey
NWOGAKBGRRKZPL-UHFFFAOYSA-N
Physicochemical Property
logP
4.32234
Rotatable Bonds
5
Heavy Atom Count
32
Polar Areas
110.86
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 118470493
ChEMBL ID
CHEMBL4867254
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01029, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 = 64 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 26 nM